Bromodomain protein BRD4 controls HOTAIR, a long noncoding RNA essential for glioblastoma proliferation
Pastori, Chiara, Philipp Kapranov, Clara Penas, Veronica Peschansky, Claude-Henry Volmar, Jann N. Sarkaria, Amade Bregy, Ricardo Komotar, Georges St. Laurent, Nagi G. Ayad, Claes Wahlestedt
Published in Proceedings of the National Academy of Sciences - PNAS (07.07.2015)
Published in Proceedings of the National Academy of Sciences - PNAS (07.07.2015)
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Journal Article
An overview of human single-cell RNA sequencing studies in neurobiological disease
Walter, T. Jordan, Suter, Robert K., Ayad, Nagi G.
Published in Neurobiology of disease (01.08.2023)
Published in Neurobiology of disease (01.08.2023)
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Journal Article
Epigenetic pathways and plasticity in brain tumors
Suter, Robert K., Rodriguez-Blanco, Jezabel, Ayad, Nagi G.
Published in Neurobiology of disease (01.11.2020)
Published in Neurobiology of disease (01.11.2020)
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Journal Article
Organoid Models of Glioblastoma and Their Role in Drug Discovery
Rybin, Matthew J, Ivan, Michael E, Ayad, Nagi G, Zeier, Zane
Published in Frontiers in cellular neuroscience (05.02.2021)
Published in Frontiers in cellular neuroscience (05.02.2021)
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Journal Article
Neuroinflammation Treatment via Targeted Delivery of Nanoparticles
Cerqueira, Susana R, Ayad, Nagi G, Lee, Jae K
Published in Frontiers in cellular neuroscience (30.09.2020)
Published in Frontiers in cellular neuroscience (30.09.2020)
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Journal Article
Glutaminase 2 as a therapeutic target in glioblastoma
Veeramachaneni, Rithvik K., Suter, Robert K., Rowland, Emma, Jermakowicz, Anna, Ayad, Nagi G.
Published in Biochimica et biophysica acta. Reviews on cancer (01.11.2024)
Published in Biochimica et biophysica acta. Reviews on cancer (01.11.2024)
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Journal Article
Drug and disease signature integration identifies synergistic combinations in glioblastoma
Stathias, Vasileios, Jermakowicz, Anna M, Maloof, Marie E, Forlin, Michele, Walters, Winston, Suter, Robert K, Durante, Michael A, Williams, Sion L, Harbour, J William, Volmar, Claude-Henry, Lyons, Nicholas J, Wahlestedt, Claes, Graham, Regina M, Ivan, Michael E, Komotar, Ricardo J, Sarkaria, Jann N, Subramanian, Aravind, Golub, Todd R, Schürer, Stephan C, Ayad, Nagi G
Published in Nature communications (14.12.2018)
Published in Nature communications (14.12.2018)
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Journal Article
Kinome-Wide Virtual Screening by Multi-Task Deep Learning
Hu, Jiaming, Allen, Bryce K, Stathias, Vasileios, Ayad, Nagi G, Schürer, Stephan C
Published in International journal of molecular sciences (22.02.2024)
Published in International journal of molecular sciences (22.02.2024)
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Journal Article
The BET Bromodomain Inhibitor I-BET151 Acts Downstream of Smoothened Protein to Abrogate the Growth of Hedgehog Protein-driven Cancers
Long, Jun, Li, Bin, Rodriguez-Blanco, Jezabel, Pastori, Chiara, Volmar, Claude-Henry, Wahlestedt, Claes, Capobianco, Anthony, Bai, Feng, Pei, Xin-Hai, Ayad, Nagi G., Robbins, David J.
Published in The Journal of biological chemistry (19.12.2014)
Published in The Journal of biological chemistry (19.12.2014)
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Journal Article
392 Targeting One-Carbon Metabolism in Brain Cancer
Rowland, Emma, Ayad, Nagi G.
Published in Journal of clinical and translational science (01.04.2024)
Published in Journal of clinical and translational science (01.04.2024)
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Journal Article
The novel BET inhibitor UM-002 reduces glioblastoma cell proliferation and invasion
Jermakowicz, Anna M, Rybin, Matthew J, Suter, Robert K, Sarkaria, Jann N, Zeier, Zane, Feng, Yangbo, Ayad, Nagi G
Published in Scientific reports (03.12.2021)
Published in Scientific reports (03.12.2021)
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Journal Article
Drug Repositioning in Glioblastoma: A Pathway Perspective
Tan, Sze Kiat, Jermakowicz, Anna, Mookhtiar, Adnan K, Nemeroff, Charles B, Schürer, Stephan C, Ayad, Nagi G
Published in Frontiers in pharmacology (16.03.2018)
Published in Frontiers in pharmacology (16.03.2018)
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Journal Article
Identifying glioblastoma gene networks based on hypergeometric test analysis
Stathias, Vasileios, Pastori, Chiara, Griffin, Tess Z, Komotar, Ricardo, Clarke, Jennifer, Zhang, Ming, Ayad, Nagi G
Published in PloS one (31.12.2014)
Published in PloS one (31.12.2014)
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Journal Article
RAPID resistance to BET inhibitors is mediated by FGFR1 in glioblastoma
Jermakowicz, Anna M, Kurimchak, Alison M, Johnson, Katherine J, Bourgain-Guglielmetti, Florence, Kaeppeli, Simon, Affer, Maurizio, Pradhyumnan, Hari, Suter, Robert K, Walters, Winston, Cepero, Maria, Duncan, James S, Ayad, Nagi G
Published in Scientific reports (23.04.2024)
Published in Scientific reports (23.04.2024)
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Journal Article
BET bromodomain proteins are required for glioblastoma cell proliferation
Pastori, Chiara, Daniel, Mark, Penas, Clara, Volmar, Claude-Henry, Johnstone, Andrea L, Brothers, Shaun P, Graham, Regina M, Allen, Bryce, Sarkaria, Jann N, Komotar, Ricardo J, Wahlestedt, Claes, Ayad, Nagi G
Published in Epigenetics (01.04.2014)
Published in Epigenetics (01.04.2014)
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Journal Article
The E3 ubiquitin ligase component, Cereblon, is an evolutionarily conserved regulator of Wnt signaling
Shen, Chen, Nayak, Anmada, Neitzel, Leif R., Adams, Amber A., Silver-Isenstadt, Maya, Sawyer, Leah M., Benchabane, Hassina, Wang, Huilan, Bunnag, Nawat, Li, Bin, Wynn, Daniel T., Yang, Fan, Garcia-Contreras, Marta, Williams, Charles H., Dakshanamurthy, Sivanesan, Hong, Charles C., Ayad, Nagi G., Capobianco, Anthony J., Ahmed, Yashi, Lee, Ethan, Robbins, David J.
Published in Nature communications (06.09.2021)
Published in Nature communications (06.09.2021)
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Journal Article
A dual aurora and lim kinase inhibitor reduces glioblastoma proliferation and invasion
Rybin, Matthew J., Laverde-Paz, Mayra Juliana, Suter, Robert K., Affer, Maurizio, Ayad, Nagi G., Feng, Yangbo, Zeier, Zane
Published in Bioorganic & medicinal chemistry letters (01.04.2022)
Published in Bioorganic & medicinal chemistry letters (01.04.2022)
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