Incarvillateine produces antinociceptive and motor suppressive effects via adenosine receptor activation
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Published in PloS one (25.06.2019)
Published in PloS one (25.06.2019)
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Journal Article
SAR study on Novel truxillic acid monoester-Based inhibitors of fatty acid binding proteins as Next-Generation antinociceptive agents
Wang, Hehe, Taouil, Adam, Awwa, Monaf, Clement, Timothy, Zhu, Chuanzhou, Kim, Jinwoo, Rendina, Dominick, Jayanetti, Kalani, Maharaj, Atri, Wang, Liqun, Bogdan, Diane, Pepe, Antonella, Kaczocha, Martin, Ojima, Iwao
Published in Bioorganic chemistry (01.12.2022)
Published in Bioorganic chemistry (01.12.2022)
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Targeting the Hemopexin-like Domain of Latent Matrix Metalloproteinase‑9 (proMMP-9) with a Small Molecule Inhibitor Prevents the Formation of Focal Adhesion Junctions
Alford, Vincent M, Kamath, Anushree, Ren, Xiaodong, Kumar, Kunal, Gan, Qianwen, Awwa, Monaf, Tong, Michael, Seeliger, Markus A, Cao, Jian, Ojima, Iwao, Sampson, Nicole S
Published in ACS chemical biology (17.11.2017)
Published in ACS chemical biology (17.11.2017)
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Journal Article
SAR studies on truxillic acid mono esters as a new class of antinociceptive agents targeting fatty acid binding proteins
Yan, Su, Elmes, Matthew W., Tong, Simon, Hu, Kongzhen, Awwa, Monaf, Teng, Gary Y.H., Jing, Yunrong, Freitag, Matthew, Gan, Qianwen, Clement, Timothy, Wei, Longfei, Sweeney, Joseph M., Joseph, Olivia M., Che, Joyce, Carbonetti, Gregory S., Wang, Liqun, Bogdan, Diane M., Falcone, Jerome, Smietalo, Norbert, Zhou, Yuchen, Ralph, Brian, Hsu, Hao-Chi, Li, Huilin, Rizzo, Robert C., Deutsch, Dale G., Kaczocha, Martin, Ojima, Iwao
Published in European journal of medicinal chemistry (25.06.2018)
Published in European journal of medicinal chemistry (25.06.2018)
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Journal Article
Structure-activity relationship studies on 2,5,6-trisubstituted benzimidazoles targeting Mtb -FtsZ as antitubercular agents
Haranahalli, Krupanandan, Tong, Simon, Kim, Saerom, Awwa, Monaf, Chen, Lei, Knudson, Susan E, Slayden, Richard A, Singleton, Eric, Russo, Riccardo, Connell, Nancy, Ojima, Iwao
Published in MedChemComm (01.01.2021)
Published in MedChemComm (01.01.2021)
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Journal Article
Structure-activity relationship studies on 2,5,6-trisubstituted benzimidazoles targeting -FtsZ as antitubercular agents
Haranahalli, Krupanandan, Tong, Simon, Kim, Saerom, Awwa, Monaf, Chen, Lei, Knudson, Susan E, Slayden, Richard A, Singleton, Eric, Russo, Riccardo, Connell, Nancy, Ojima, Iwao
Published in RSC medicinal chemistry (04.02.2021)
Published in RSC medicinal chemistry (04.02.2021)
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Journal Article
Substituted pyrimidines as matrix metalloproteinase-9 hemopexin domain inhibitors
Awwa, Monaf, Ren, Xiadong, Ojima, Iwao, Alford, Vincent, Sampson, Nicole, Kamath, Anushree, Cao, Jian
Year of Publication 25.06.2024
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Year of Publication 25.06.2024
Patent
SUBSTITUTED QUINAZOLINES AS MATRIX METALLOPROTEINASE-9 HEMOPEXIN DOMAIN INHIBITORS
OJIMA, Iwao, REN, Xiadong, CAO, Jian, ALFORD, Vincent, KAMATH, Anushree, AWWA, Monaf, SAMPSON, Nicole
Year of Publication 07.10.2021
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Year of Publication 07.10.2021
Patent
Substituted quinazolines as matrix metalloproteinase-9 hemopexin domain inhibitors
Awwa, Monaf, Ren, Xiadong, Ojima, Iwao, Alford, Vincent, Sampson, Nicole, Kamath, Anushree, Cao, Jian
Year of Publication 22.06.2021
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Year of Publication 22.06.2021
Patent
MATRIX METALLOPROTEINASE-9 HEMOPEXIN DOMAIN INHIBITORS AND METHODS OF TREATMENT USING SAME
OJIMA, Iwao, REN, Xiadong, CAO, Jian, ALFORD, Vincent, KAMATH, Anushree, AWWA, Monaf, SAMPSON, Nicole
Year of Publication 16.01.2020
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Year of Publication 16.01.2020
Patent