Improving potency and selectivity of a new class of non-Zn-chelating MMP-13 inhibitors
Heim-Riether, Alexander, Taylor, Steven J., Liang, Shuang, Gao, Donghong Amy, Xiong, Zhaoming, Michael August, E., Collins, Brandon K., Farmer, Bennett T., Haverty, Kathleen, Hill-Drzewi, Melissa, Junker, Hans-Dieter, Mariana Margarit, S., Moss, Neil, Neumann, Thomas, Proudfoot, John R., Keenan, Lana Smith, Sekul, Renate, Zhang, Qiang, Li, Jun, Farrow, Neil A.
Published in Bioorganic & medicinal chemistry letters (15.09.2009)
Published in Bioorganic & medicinal chemistry letters (15.09.2009)
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Benzimidazolone as potent chymase inhibitor: Modulation of reactive metabolite formation in the hydrophobic (P 1) region
Lo, Ho Yin, Nemoto, Peter A., Kim, Jin Mi, Hao, Ming-Hong, Qian, Kevin C., Farrow, Neil A., Albaugh, Daniel R., Fowler, Danielle M., Schneiderman, Richard D., Michael August, E., Martin, Leslie, Hill-Drzewi, Melissa, Pullen, Steven S., Takahashi, Hidenori, De Lombaert, Stéphane
Published in Bioorganic & medicinal chemistry letters (01.08.2011)
Published in Bioorganic & medicinal chemistry letters (01.08.2011)
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Reversal of H3K9me2 by a Small-Molecule Inhibitor for the G9a Histone Methyltransferase
Kubicek, Stefan, O'Sullivan, Roderick J., August, E. Michael, Hickey, Eugene R., Zhang, Qiang, Teodoro, Miguel L., Rea, Stephen, Mechtler, Karl, Kowalski, Jennifer A., Homon, Carol Ann, Kelly, Terence A., Jenuwein, Thomas
Published in Molecular cell (09.02.2007)
Published in Molecular cell (09.02.2007)
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SAR studies of non-zinc-chelating MMP-13 inhibitors: Improving selectivity and metabolic stability
Gao, Donghong Amy, Xiong, Zhaoming, Heim-Riether, Alexander, Amodeo, Laura, August, E. Michael, Cao, Xianhua, Ciccarelli, Leonard, Collins, Brandon K., Harrington, Kyle, Haverty, Kathleen, Hill-Drzewi, Melissa, Li, Xiang, Liang, Shuang, Margarit, Steluta Mariana, Moss, Neil, Nagaraja, Nelamangala, Proudfoot, John, Roman, Rene, Schlyer, Sabine, Keenan, Lana Smith, Taylor, Steven, Wellenzohn, Bernd, Wiedenmayer, Dieter, Li, Jun, Farrow, Neil A.
Published in Bioorganic & medicinal chemistry letters (01.09.2010)
Published in Bioorganic & medicinal chemistry letters (01.09.2010)
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Bioluminescent method for assaying multiple semicarbazide-sensitive amine oxidase (SSAO) family members in both 96- and 384-well formats
Peet, Gregory W, Lukas, Susan, Hill-Drzewi, Melissa, Martin, Leslie, Rybina, Irina V, Roma, Teresa, Shoultz, Alycia, Zhu, Xiang, Cazacu, Daniela, Kronkaitis, Anthony, Baptiste, Alistair, Raudenbush, Brian C, August, E Michael, Modis, Louise Kelly
Published in Journal of biomolecular screening (01.10.2011)
Published in Journal of biomolecular screening (01.10.2011)
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Development of a high-throughput assay to measure histidine decarboxylase activity
August, E Michael, Patnaude, Lori, Hopkins, Jerry, Studts, Joey, Gautschi, Elda, Shrutkowski, Anthony, Kronkaitis, Anthony, Brown, Martha, Kabcenell, Alisa, Rajotte, Daniel
Published in Journal of biomolecular screening (01.10.2006)
Published in Journal of biomolecular screening (01.10.2006)
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Abstract 5590: Screening of pediatric and adult sarcoma cell lines reveals novel patterns of sensitivity toward approved oncology drugs and investigational agents
August, E. Michael, Delosh, Rene, Laudeman, Julie, Ogle, Chad, Reinhart, Russell, Selby, Michael, Silvers, Thomas, Morris, Joel, Teicher, Beverly A.
Published in Cancer research (Chicago, Ill.) (15.04.2013)
Published in Cancer research (Chicago, Ill.) (15.04.2013)
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Abstract 4361: Target and drug discovery for recalcitrant, rare and neglected cancers
Monks, Anne, Rapisarda, Annamaria, Wrzeszczynski, Kazimierz O., August, E. Michael, Polley, Eric C., Kondapaka, Sudhir B., Kaur, Gurmeet, Newton, Dianne, Teicher, Beverley A.
Published in Cancer research (Chicago, Ill.) (15.04.2013)
Published in Cancer research (Chicago, Ill.) (15.04.2013)
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1-(2,3-Dideoxy-.beta.-D-glycero-pent-2-enofuranosyl)thymine. A highly potent and selective anti-HIV agent
Mansuri, Muzammil M, Starrett, John E, Ghazzouli, Ismail, Hitchcock, Michael J. M, Sterzycki, Roman Z, Brankovan, Vera, Lin, Tai Shun, August, E. Michael, Prusoff, William H
Published in Journal of medicinal chemistry (01.02.1989)
Published in Journal of medicinal chemistry (01.02.1989)
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Driver status display
DANIEL S. GLASER, GILL PATRICE, LORE JOSEPH V, SZERBA JOSEPH F, AUGUST MICHAEL E, GLASER DANIEL G
Year of Publication 18.07.2023
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Year of Publication 18.07.2023
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