Hydropersulfides inhibit lipid peroxidation and ferroptosis by scavenging radicals
Barayeu, Uladzimir, Schilling, Danny, Eid, Mohammad, Xavier da Silva, Thamara Nishida, Schlicker, Lisa, Mitreska, Nikolina, Zapp, Christopher, Gräter, Frauke, Miller, Aubry K, Kappl, Reinhard, Schulze, Almut, Friedmann Angeli, José Pedro, Dick, Tobias P
Published in Nature chemical biology (01.01.2023)
Published in Nature chemical biology (01.01.2023)
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Journal Article
Regulation of mitochondrial morphology and function by stearoylation of TFR1
Senyilmaz, Deniz, Virtue, Sam, Xu, Xiaojun, Tan, Chong Yew, Griffin, Julian L, Miller, Aubry K, Vidal-Puig, Antonio, Teleman, Aurelio A
Published in Nature (London) (03.09.2015)
Published in Nature (London) (03.09.2015)
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Journal Article
Practical synthesis of a phthalimide-based Cereblon ligand to enable PROTAC development
Lohbeck, Jasmin, Miller, Aubry K.
Published in Bioorganic & medicinal chemistry letters (01.11.2016)
Published in Bioorganic & medicinal chemistry letters (01.11.2016)
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Journal Article
Commonly Used Alkylating Agents Limit Persulfide Detection by Converting Protein Persulfides into Thioethers
Schilling, Danny, Barayeu, Uladzimir, Steimbach, Raphael R., Talwar, Deepti, Miller, Aubry K., Dick, Tobias P.
Published in Angewandte Chemie International Edition (25.07.2022)
Published in Angewandte Chemie International Edition (25.07.2022)
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Journal Article
Chemoproteomic target deconvolution reveals Histone Deacetylases as targets of (R)-lipoic acid
Lechner, Severin, Steimbach, Raphael R, Wang, Longlong, Deline, Marshall L, Chang, Yun-Chien, Fromme, Tobias, Klingenspor, Martin, Matthias, Patrick, Miller, Aubry K, Médard, Guillaume, Kuster, Bernhard
Published in Nature communications (15.06.2023)
Published in Nature communications (15.06.2023)
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Journal Article
Bioinspired Asymmetric Total Synthesis of Emeriones A–C
Jänner, Sven, Isak, Daniel, Li, Yuli, Houk, Kendall N., Miller, Aubry K.
Published in Angewandte Chemie International Edition (08.08.2022)
Published in Angewandte Chemie International Edition (08.08.2022)
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Journal Article
Stearic acid blunts growth-factor signaling via oleoylation of GNAI proteins
Nůsková, Hana, Serebryakova, Marina V., Ferrer-Caelles, Anna, Sachsenheimer, Timo, Lüchtenborg, Christian, Miller, Aubry K., Brügger, Britta, Kordyukova, Larisa V., Teleman, Aurelio A.
Published in Nature communications (28.07.2021)
Published in Nature communications (28.07.2021)
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Journal Article
Dual role of HDAC10 in lysosomal exocytosis and DNA repair promotes neuroblastoma chemoresistance
Ridinger, Johannes, Koeneke, Emily, Kolbinger, Fiona R, Koerholz, Katharina, Mahboobi, Siavosh, Hellweg, Lars, Gunkel, Nikolas, Miller, Aubry K, Peterziel, Heike, Schmezer, Peter, Hamacher-Brady, Anne, Witt, Olaf, Oehme, Ina
Published in Scientific reports (03.07.2018)
Published in Scientific reports (03.07.2018)
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Journal Article
Selective Inhibition of Histone Deacetylase 10: Hydrogen Bonding to the Gatekeeper Residue is Implicated
Géraldy, Magalie, Morgen, Michael, Sehr, Peter, Steimbach, Raphael R, Moi, Davide, Ridinger, Johannes, Oehme, Ina, Witt, Olaf, Malz, Mona, Nogueira, Mauro S, Koch, Oliver, Gunkel, Nikolas, Miller, Aubry K
Published in Journal of medicinal chemistry (09.05.2019)
Published in Journal of medicinal chemistry (09.05.2019)
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Journal Article
Target deconvolution of HDAC pharmacopoeia reveals MBLAC2 as common off-target
Lechner, Severin, Malgapo, Martin Ian P, Grätz, Christian, Steimbach, Raphael R, Baron, Agnes, Rüther, Patrick, Nadal, Simon, Stumpf, Carmen, Loos, Christina, Ku, Xin, Prokofeva, Polina, Lautenbacher, Ludwig, Heimburg, Tino, Würf, Vivian, Meng, Chen, Wilhelm, Mathias, Sippl, Wolfgang, Kleigrewe, Karin, Pauling, Josch K, Kramer, Karl, Miller, Aubry K, Pfaffl, Michael W, Linder, Maurine E, Kuster, Bernhard, Médard, Guillaume
Published in Nature chemical biology (01.08.2022)
Published in Nature chemical biology (01.08.2022)
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Journal Article
A KLK6 Activity-Based Probe Reveals a Role for KLK6 Activity in Pancreatic Cancer Cell Invasion
Zhang, Leran, Lovell, Scott, De Vita, Elena, Jagtap, Pravin Kumar Ankush, Lucy, Daniel, Goya Grocin, Andrea, Kjær, Svend, Borg, Annabel, Hennig, Janosch, Miller, Aubry K., Tate, Edward W.
Published in Journal of the American Chemical Society (14.12.2022)
Published in Journal of the American Chemical Society (14.12.2022)
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Journal Article
A potent, proteolysis-resistant inhibitor of kallikrein-related peptidase 6 (KLK6) for cancer therapy, developed by combinatorial engineering
Sananes, Amiram, Cohen, Itay, Shahar, Anat, Hockla, Alexandra, De Vita, Elena, Miller, Aubry K., Radisky, Evette S., Papo, Niv
Published in The Journal of biological chemistry (17.08.2018)
Published in The Journal of biological chemistry (17.08.2018)
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Journal Article
Frontispiece: Commonly Used Alkylating Agents Limit Persulfide Detection by Converting Protein Persulfides into Thioethers
Schilling, Danny, Barayeu, Uladzimir, Steimbach, Raphael R., Talwar, Deepti, Miller, Aubry K., Dick, Tobias P.
Published in Angewandte Chemie International Edition (25.07.2022)
Published in Angewandte Chemie International Edition (25.07.2022)
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Journal Article
Tetrahydro-β-carboline derivatives as potent histone deacetylase 6 inhibitors with broad-spectrum antiproliferative activity
Chen, Xin, Wang, Jiayun, Zhao, Peng, Dang, Baiyun, Liang, Ting, Steimbach, Raphael R., Miller, Aubry K., Liu, Jia, Wang, Xin, Zhang, Tongtong, Luan, Xiaofa, Hu, Jiadong, Gao, Jinming
Published in European journal of medicinal chemistry (15.11.2023)
Published in European journal of medicinal chemistry (15.11.2023)
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Journal Article
Decrypting lysine deacetylase inhibitor action and protein modifications by dose-resolved proteomics
Chang, Yun-Chien, Gnann, Christian, Steimbach, Raphael R., Bayer, Florian P., Lechner, Severin, Sakhteman, Amirhossein, Abele, Miriam, Zecha, Jana, Trendel, Jakob, The, Matthew, Lundberg, Emma, Miller, Aubry K., Kuster, Bernhard
Published in Cell reports (Cambridge) (25.06.2024)
Published in Cell reports (Cambridge) (25.06.2024)
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Journal Article
Histone deacetylase-10 liberates spermidine to support polyamine homeostasis and tumor cell growth
Stewart, Tracy Murray, Foley, Jackson R., Holbert, Cassandra E., Klinke, Glynis, Poschet, Gernot, Steimbach, Raphael R., Miller, Aubry K., Casero, Robert A.
Published in The Journal of biological chemistry (01.10.2022)
Published in The Journal of biological chemistry (01.10.2022)
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Journal Article
Scalable synthesis and structural characterization of reversible KLK6 inhibitors
Baumann, Andreas, Isak, Daniel, Lohbeck, Jasmin, Jagtap, Pravin Kumar Ankush, Hennig, Janosch, Miller, Aubry K
Published in RSC advances (21.09.2022)
Published in RSC advances (21.09.2022)
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