Fascaplysin-inspired diindolyls as selective inhibitors of CDK4/cyclin D1
Aubry, Carine, Wilson, A. James, Emmerson, Daniel, Murphy, Emma, Chan, Yu Yam, Dickens, Michael P., García, Marcos D., Jenkins, Paul R., Mahale, Sachin, Chaudhuri, Bhabatosh
Published in Bioorganic & medicinal chemistry (15.08.2009)
Published in Bioorganic & medicinal chemistry (15.08.2009)
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Journal Article
The design and synthesis of novel 3-[2-indol-1-yl-ethyl]-1H-indole derivatives as selective inhibitors of CDK4
Aubry, Carine, Patel, Asma, Mahale, Sachin, Chaudhuri, Bhabatosh, Maréchal, Jean-Didier, Sutcliffe, Michael J., Jenkins, Paul R.
Published in Tetrahedron letters (28.02.2005)
Published in Tetrahedron letters (28.02.2005)
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Journal Article
The design and synthesis of novel 3-[2-indol-1-yl-ethyl]-1 H-indole derivatives as selective inhibitors of CDK4
Aubry, Carine, Patel, Asma, Mahale, Sachin, Chaudhuri, Bhabatosh, Maréchal, Jean-Didier, Sutcliffe, Michael J., Jenkins, Paul R.
Published in Tetrahedron letters (28.02.2005)
Published in Tetrahedron letters (28.02.2005)
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Journal Article
Design, synthesis and biological activity of new CDK4-specific inhibitors, based on fascaplysin
Aubry, C, Wilson, AJ, Jenkins, PR, Mahale, S, Chaudhuri, B, Marechal, JD, Sutcliffe, MJ
Published in Organic & biomolecular chemistry (01.01.2006)
Published in Organic & biomolecular chemistry (01.01.2006)
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CA224, a non-planar analogue of fascaplysin, inhibits Cdk4 but not Cdk2 and arrests cells at G0/G1 inhibiting pRB phosphorylation
MAHALE, Sachin, AUBRY, Carine, WILSON, A. James, JENKINS, Paul R, MARECHAL, Jean-Didier, SUTCLIFFE, Michael J, CHAUDHURI, Bhabatosh
Published in Bioorganic & medicinal chemistry letters (15.08.2006)
Published in Bioorganic & medicinal chemistry letters (15.08.2006)
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Journal Article
New fascaplysin-based CDK4-specific inhibitors: design, synthesis and biological activity
Aubry, C, Jenkins, PR, Mahale, S, Chaudhuri, B, Marechal, JD, Sutcliffe, MJ
Published in Chemical communications (Cambridge, England) (01.01.2004)
Published in Chemical communications (Cambridge, England) (01.01.2004)
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Inhibition of cancer cell growth by cyclin dependent kinase 4 inhibitors synthesized based on the structure of fascaplysin
Mahale, Sachin, Aubry, Carine, Jenkins, Paul R., Maréchal, Jean-Didier, Sutcliffe, Michael J., Chaudhuri, Bhabatosh
Published in Bioorganic chemistry (01.10.2006)
Published in Bioorganic chemistry (01.10.2006)
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Journal Article
CA224, a non-planar analogue of fascaplysin, inhibits Cdk4 but not Cdk2 and arrests cells at G 0/G 1 inhibiting pRB phosphorylation
Mahale, Sachin, Aubry, Carine, James Wilson, A., Jenkins, Paul R., Maréchal, Jean-Didier, Sutcliffe, Michael J., Chaudhuri, Bhabatosh
Published in Bioorganic & medicinal chemistry letters (2006)
Published in Bioorganic & medicinal chemistry letters (2006)
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Journal Article
New synthesis ofcis 5-tert-butyl-L-proline via cuprate. Evaluation as acis proline mimetic in a biological active octapeptide
Aubry, Carine, Oulyadi, Hassan, Dutheuil, Guillaume, Leprince, Jérôme, Vaudry, Hubert, Pannecoucke, Xavier, Quirion, Jean-Charles
Published in Journal of peptide science (01.02.2006)
Published in Journal of peptide science (01.02.2006)
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Journal Article
New sythesis of cis 5-tert-butyl-L-proline via cuprate. Evaluation as a cis proline mimetic in a biological active octapeptide
Aubry, Carine, Oulyadi, Hassan, Dutheuil, Guillaume, Leprince, Jérôme, Vaudry, Hubert, Pannecoucke, Xavier, Quirion, Jean-Charles
Published in Journal of peptide science (2006)
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Published in Journal of peptide science (2006)
Journal Article
New synthesis of cis 5-tert-butyl-L-proline via cuprate. Evaluation as a cis proline mimetic in a biological active octapeptide
Aubry, Carine, Oulyadi, Hassan, Dutheuil, Guillaume, Leprince, Jerome, Vaudry, Hubert, Pannecoucke, Xavier, Quirion, Jean-Charles
Published in Journal of peptide science (01.02.2006)
Published in Journal of peptide science (01.02.2006)
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Journal Article
The Design and Synthesis of Novel 3-[2-Indol-1-yl-ethyl]-1H-indole Derivatives as Selective Inhibitors of CDK4
Aubry, Carine, Patel, Asma, Mahale, Sachin, Chaudhuri, Bhabatosh, Marechal, Jean-Didier, Sutcliffe, Michael J., Jenkins, Paul R.
Published in ChemInform (14.06.2005)
Published in ChemInform (14.06.2005)
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