Importance of the Azole Moiety of Cimetidine Derivatives for the Inhibition of Human Multidrug and Toxin Extrusion Transporter 1 (hMATE1)
Shinya, Susumu, Kawai, Kentaro, Tarui, Atsushi, Karuo, Yukiko, Sato, Kazuyuki, Matsuda, Masaya, Kitatani, Kazuyuki, Kobayashi, Naoki, Nabe, Takeshi, Otsuka, Masato, Omote, Masaaki
Published in Chemical & pharmaceutical bulletin (01.09.2021)
Published in Chemical & pharmaceutical bulletin (01.09.2021)
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Journal Article
Pentafluorosulfanyl-substituted biaryl derivatives as MATE-type transporter inhibitors targeting drug-resistant bacteria
Shinya, Susumu, Kawai, Kentaro, Kobayashi, Naoki, Karuo, Yukiko, Tarui, Atsushi, Sato, Kazuyuki, Otsuka, Masato, Omote, Masaaki
Published in Bioorganic & medicinal chemistry (01.02.2024)
Published in Bioorganic & medicinal chemistry (01.02.2024)
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Journal Article
Identification and Synthesis of DDI-6, a Quinolinol Analog Capable of Activating Both Caenorhabditis elegans and Mouse Spermatozoa
Karuo, Yukiko, Shiraki, Riona, Yoshida, Ayaka, Tsunokawa, Ryo, Nakahara-Yamada, Mayuko, Tarui, Atsushi, Sato, Kazuyuki, Kawai, Kentaro, Omote, Masaaki, Nishimura, Hitoshi
Published in Chemical & pharmaceutical bulletin (01.06.2021)
Published in Chemical & pharmaceutical bulletin (01.06.2021)
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Journal Article
Fluorophenylalkyl-substituted cyanoguanidine derivatives as bacteria-selective MATE transporter inhibitors for the treatment of antibiotic-resistant infections
Shinya, Susumu, Kawai, Kentaro, Kobayashi, Naoki, Karuo, Yukiko, Tarui, Atsushi, Sato, Kazuyuki, Otsuka, Masato, Omote, Masaaki
Published in Bioorganic & medicinal chemistry (15.11.2022)
Published in Bioorganic & medicinal chemistry (15.11.2022)
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Journal Article
Synthesis of aryl 2-bromo-2-chloro-1,1-difluoroethyl ethers through the base-mediated reaction between phenols and halothane
Karuo, Yukiko, Kametani, Ayaka, Tarui, Atsushi, Sato, Kazuyuki, Kawai, Kentaro, Omote, Masaaki
Published in Beilstein journal of organic chemistry (11.01.2021)
Published in Beilstein journal of organic chemistry (11.01.2021)
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Journal Article
Synthesis of new fluorescent molecules having an aggregation-induced emission property derived from 4-fluoroisoxazoles
Sato, Kazuyuki, Kawasaki, Akira, Karuo, Yukiko, Tarui, Atsushi, Kawai, Kentaro, Omote, Masaaki
Published in Beilstein journal of organic chemistry (22.06.2020)
Published in Beilstein journal of organic chemistry (22.06.2020)
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Journal Article
LCP: Simple Representation of Docking Poses for Machine Learning: A Case Study on Xanthine Oxidase Inhibitors
Kawai, Kentaro, Asanuma, Yoshitaka, Kato, Toshiki, Karuo, Yukiko, Tarui, Atsushi, Sato, Kazuyuki, Omote, Masaaki
Published in Molecular informatics (01.05.2022)
Published in Molecular informatics (01.05.2022)
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Journal Article
Rhodium-catalyzed homo-coupling reaction of aryl Grignard reagents and its application for the synthesis of an integrin inhibitor
Sato, Kazuyuki, Teranishi, Satoki, Sakaue, Atsushi, Karuo, Yukiko, Tarui, Atsushi, Kawai, Kentaro, Takeda, Hiroyuki, Kinashi, Tatsuo, Omote, Masaaki
Published in Beilstein journal of organic chemistry (12.06.2024)
Published in Beilstein journal of organic chemistry (12.06.2024)
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Journal Article
Decarboxylative Aldol Reaction of α,α-Difluoro-β-keto Esters: Easy Access to Difluoroenolate
Tarui, Atsushi, Shimomura, Hiroshi, Yasuno, Yohei, Karuo, Yukiko, Sato, Kazuyuki, Kawai, Kentaro, Omote, Masaaki
Published in ACS omega (18.06.2024)
Published in ACS omega (18.06.2024)
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Journal Article
Ligand-Promoted Asymmetric Imino-Reformatsky Reaction of Ethyl Dibromofluoroacetate
Tarui, Atsushi, Nishimura, Haruka, Ikebata, Takeshi, Tahira, Asuka, Sato, Kazuyuki, Omote, Masaaki, Minami, Hideki, Miwa, Yoshihisa, Ando, Akira
Published in Organic letters (18.04.2014)
Published in Organic letters (18.04.2014)
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Journal Article
Synthesis of Small Fluorescent Molecules and Evaluation of Photophysical Properties
Ogawa, Futa, Karuo, Yukiko, Yamazawa, Ryuji, Miyanaga, Kanae, Hori, Kazushige, Tani, Keita, Yamada, Kengo, Saito, Yuki, Funabiki, Kazumasa, Tarui, Atsushi, Sato, Kazuyuki, Ito, Kiyoshi, Kawai, Kentaro, Omote, Masaaki
Published in Journal of organic chemistry (17.01.2020)
Published in Journal of organic chemistry (17.01.2020)
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Journal Article
Synthesis of 2,2-difluoro-2-arylethylamines as fluorinated analogs of octopamine and noradrenaline
Tarui Atsushi, Kamata Erika, Ebisu Koji, Kawai Yui, Araki Ryota, Yabe Takeshi, Karuo Yukiko, Sato Kazuyuki, Kawai Kentaro, Omote Masaaki
Published in Heterocyclic Communications (19.03.2022)
Published in Heterocyclic Communications (19.03.2022)
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Journal Article
Development of a fluorogenic small substrate for dipeptidyl peptidase-4
Ogawa, Futa, Takeda, Masanori, Miyanaga, Kanae, Tani, Keita, Yamazawa, Ryuji, Ito, Kiyoshi, Tarui, Atsushi, Sato, Kazuyuki, Omote, Masaaki
Published in Beilstein journal of organic chemistry (14.12.2017)
Published in Beilstein journal of organic chemistry (14.12.2017)
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Journal Article
Rh-Catalyzed reductive Mannich-type reaction and its application towards the synthesis of (±)-ezetimibe
Isoda, Motoyuki, Sato, Kazuyuki, Kunugi, Yurika, Tokonishi, Satsuki, Tarui, Atsushi, Omote, Masaaki, Minami, Hideki, Ando, Akira
Published in Beilstein journal of organic chemistry (27.07.2016)
Published in Beilstein journal of organic chemistry (27.07.2016)
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Journal Article
Diastereoselective synthesis of 2-fluoroaziridine-2-carboxylates by Reformatsky-type aza-Darzens reaction
Tarui, Atsushi, Kawashima, Naoto, Sato, Kazuyuki, Omote, Masaaki, Ando, Akira
Published in Tetrahedron letters (11.08.2010)
Published in Tetrahedron letters (11.08.2010)
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Journal Article
Csp3–Csp3 Homocoupling Reaction of Benzyl Halides Catalyzed by Rhodium
Sato, Kazuyuki, Inoue, Yuichi, Mori, Tomohisa, Sakaue, Atsushi, Tarui, Atsushi, Omote, Masaaki, Kumadaki, Itsumaro, Ando, Akira
Published in Organic letters (18.07.2014)
Published in Organic letters (18.07.2014)
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