Levomilnacipran (F2695), a norepinephrine-preferring SNRI: Profile in vitro and in models of depression and anxiety
Auclair, A.L., Martel, J.C., Assié, M.B., Bardin, L., Heusler, P., Cussac, D., Marien, M., Newman-Tancredi, A., O'Connor, J.A., Depoortère, R.
Published in Neuropharmacology (01.07.2013)
Published in Neuropharmacology (01.07.2013)
Get full text
Journal Article
Signal transduction and functional selectivity of F15599, a preferential post‐synaptic 5‐HT1A receptor agonist
Newman‐Tancredi, A, Martel, J‐C, Assié, M‐B, Buritova, J, Lauressergues, E, Cosi, C, Heusler, P, Bruins Slot, L, Colpaert, FC, Vacher, B, Cussac, D
Published in British journal of pharmacology (01.01.2009)
Published in British journal of pharmacology (01.01.2009)
Get full text
Journal Article
Rapid desensitization of somatodendritic 5‐HT1A receptors by chronic administration of the high‐efficacy 5‐HT1A agonist, F13714: a microdialysis study in the rat
Assié, M‐B, Lomenech, H, Ravailhe, V, Faucillon, V, Newman‐Tancredi, A
Published in British journal of pharmacology (01.09.2006)
Published in British journal of pharmacology (01.09.2006)
Get full text
Journal Article
F15063, a potential antipsychotic with D2/D3 antagonist, 5‐HT1A agonist and D4 partial agonist properties: (I) in vitro receptor affinity and efficacy profile
Newman‐Tancredi, A, Assié, M‐B, Martel, J‐C, Cosi, C, Slot, L Bruins, Palmier, C, Rauly‐Lestienne, I, Colpaert, F, Vacher, B, Cussac, D
Published in British journal of pharmacology (01.05.2007)
Published in British journal of pharmacology (01.05.2007)
Get full text
Journal Article
Signal transduction and functional selectivity of F15599, a preferential post‐synaptic 5‐HT 1A receptor agonist
Newman‐Tancredi, A, Martel, J‐C, Assié, M‐B, Buritova, J, Lauressergues, E, Cosi, C, Heusler, P, Bruins Slot, L, Colpaert, FC, Vacher, B, Cussac, D
Published in British journal of pharmacology (01.01.2009)
Published in British journal of pharmacology (01.01.2009)
Get full text
Journal Article
Rapid desensitization of somatodendritic 5‐HT 1A receptors by chronic administration of the high‐efficacy 5‐HT 1A agonist, F13714: a microdialysis study in the rat
Assié, M‐B, Lomenech, H, Ravailhe, V, Faucillon, V, Newman‐Tancredi, A
Published in British journal of pharmacology (29.01.2009)
Published in British journal of pharmacology (29.01.2009)
Get full text
Journal Article
F15063, a potential antipsychotic with D 2 /D 3 antagonist, 5‐HT 1A agonist and D 4 partial agonist properties: (I) in vitro receptor affinity and efficacy profile
Newman‐Tancredi, A, Assié, M‐B, Martel, J‐C, Cosi, C, Slot, L Bruins, Palmier, C, Rauly‐Lestienne, I, Colpaert, F, Vacher, B, Cussac, D
Published in British journal of pharmacology (29.01.2009)
Published in British journal of pharmacology (29.01.2009)
Get full text
Journal Article
Large-amplitude 5-HT1A receptor activation: a new mechanism of profound, central analgesia
Colpaert, F C, Tarayre, J P, Koek, W, Pauwels, P J, Bardin, L, Xu, X-J, Wiesenfeld-Hallin, Z, Cosi, C, Carilla-Durand, E, Assié, M B, Vacher, B
Published in Neuropharmacology (01.11.2002)
Published in Neuropharmacology (01.11.2002)
Get full text
Journal Article
Neuropharmacology of a new potential anxiolytic compound, F 2692, 1-(3'-trifluoromethyl phenyl) 1, 4-dihydro 3-amino 4-oxo 6-methyl pyridazine. 2. Evaluation of its tolerance and dependence producing potential and of its effects on benzodiazepine withdrawal in the elevated plus-maze test in rats
Get more information
Journal Article
Novel Derivatives of 2-Pyridinemethylamine as Selective, Potent, and Orally Active Agonists at 5-HT1A Receptors
Vacher, Bernard, Bonnaud, Bernard, Funes, Philippe, Jubault, Nathalie, Koek, Wouter, Assié, Marie-Bernadette, Cosi, Cristina, Kleven, Mark
Published in Journal of medicinal chemistry (06.05.1999)
Published in Journal of medicinal chemistry (06.05.1999)
Get full text
Journal Article