New applications of disease genetics and pharmacogenetics to drug development
Roses, Allen D, Saunders, Ann M, Lutz, Michael W, Zhang, Nanyin, Hariri, Ahmad R, Asin, Karen E, Crenshaw, Donna G, Budur, Kumar, Burns, Daniel K, Brannan, Stephen K
Published in Current opinion in pharmacology (01.02.2014)
Published in Current opinion in pharmacology (01.02.2014)
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The application of electrophysiological methods to characterize AMPA receptors in dissociated adult rat and non-human primate cerebellar neurons for use in neuronal safety pharmacology assessments of the central nervous system
Miraucourt, Loïs S., Accardi, Michael V., Asin, Karen E., Pugsley, Michael K., Curtis, Michael J., Authier, Simon
Published in Journal of pharmacological and toxicological methods (01.09.2020)
Published in Journal of pharmacological and toxicological methods (01.09.2020)
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Substituted Hexahydrobenzo[f]thieno[c]quinolines as Dopamine D1-Selective Agonists: Synthesis and Biological Evaluation in Vitro and in Vivo
Michaelides, Michael R, Hong, Yufeng, DiDomenico, Stanley, Bayburt, Erol K, Asin, Karen E, Britton, Donald R, Lin, Chun Wel, Shiosaki, Kazumi
Published in Journal of medicinal chemistry (23.05.1997)
Published in Journal of medicinal chemistry (23.05.1997)
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Synthesis and dopaminergic activity of 3-substituted 1-(aminomethyl)-3,4-dihydro-5,6-dihydroxy-1H-2-benzopyrans: characterization of an auxiliary binding region in the D1 receptor
DeNinno, Michael P, Schoenleber, Robert, Perner, Richard J, Lijewski, Linda, Asin, Karen E, Britton, Donald R, MacKenzie, Robert, Kebabian, John W
Published in Journal of medicinal chemistry (01.08.1991)
Published in Journal of medicinal chemistry (01.08.1991)
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Hyperactivity and behavioral seizures in rodents following treatment with the dopamine D1 receptor agonists A-86929 and ABT-431
SHIOSAKI, K, ASIN, K. E, BRITTON, D. R, GIARDINA, W. J, BEDNARZ, L, MAHAN, L, MIKUSA, J, NIKKEL, A, WISMER, C
Published in European journal of pharmacology (19.12.1996)
Published in European journal of pharmacology (19.12.1996)
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(5aR,11bS)-4,5,5a,6,7,11b-Hexahydro-2-propyl-3-thia-5-azacyclopent-1-ena[c]phenanthrene-9,10-diol (A-86929): a potent and selective dopamine D1 agonist that maintain behavioral efficacy following repeated administration and characterization of its diacetyl prodrug (ABT-431)
Michaelides, Michael R, Hong, Yufeng, DiDomenico, Stanley, Asin, Karen E, Britton, Donald R, Lin, Chun Wel, Williams, Michael, Shiosaki, Kazumi
Published in Journal of medicinal chemistry (01.09.1995)
Published in Journal of medicinal chemistry (01.09.1995)
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Synthesis and biological activity of CCK heptapeptide analogs. Effects of conformational constraints and standard modifications on receptor subtype selectivity, functional activity in vitro, and appetite suppression in vivo
Holladay, Mark W, Bennett, Michael J, Tufano, Michael D, Lin, C. W, Asin, Karen E, Witte, David G, Miller, Thomas R, Bianchi, Bruce R, Nikkel, A. L
Published in Journal of medicinal chemistry (01.08.1992)
Published in Journal of medicinal chemistry (01.08.1992)
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