Identification of Novel Purine and Pyrimidine Cyclin-Dependent Kinase Inhibitors with Distinct Molecular Interactions and Tumor Cell Growth Inhibition Profiles
Arris, Christine E, Boyle, F. Thomas, Calvert, A. Hilary, Curtin, Nicola J, Endicott, Jane A, Garman, Elspeth F, Gibson, Ashleigh E, Golding, Bernard T, Grant, Sharon, Griffin, Roger J, Jewsbury, Philip, Johnson, Louise N, Lawrie, Alison M, Newell, David R, Noble, Martin E. M, Sausville, Edward A, Schultz, Robert, Yu, Wyatt
Published in Journal of medicinal chemistry (27.07.2000)
Published in Journal of medicinal chemistry (27.07.2000)
Get full text
Journal Article
Resistance-modifying agents. 8. Inhibition of O(6)-alkylguanine-DNA alkyltransferase by O(6)-alkenyl-, O(6)-cycloalkenyl-, and O(6)-(2-oxoalkyl)guanines and potentiation of temozolomide cytotoxicity in vitro by O(6)-(1-cyclopentenylmethyl)guanine
Griffin, R J, Arris, C E, Bleasdale, C, Boyle, F T, Calvert, A H, Curtin, N J, Dalby, C, Kanugula, S, Lembicz, N K, Newell, D R, Pegg, A E, Golding, B T
Published in Journal of medicinal chemistry (02.11.2000)
Published in Journal of medicinal chemistry (02.11.2000)
Get full text
Journal Article
Probing the active site and mechanism of action of O6-methylguanine-DNA methyltransferase with substrate analogues (O6-substituted guanines)
Arris, C E, Bleasdale, C, Calvert, A H, Curtin, N J, Dalby, C, Golding, B T, Griffin, R J, Lunn, J M, Major, G N, Newell, D R
Published in Anti-cancer drug design (01.10.1994)
Get more information
Published in Anti-cancer drug design (01.10.1994)
Journal Article
Structure-based design of a potent purine-based cyclin-dependent kinase inhibitor
Newell, David R, Davies, Thomas G, Bentley, Johanne, Arris, Christine E, Boyle, F. Thomas, Curtin, Nicola J, Endicott, Jane A, Gibson, Ashleigh E, Golding, Bernard T, Griffin, Roger J, Hardcastle, Ian R, Jewsbury, Philip, Johnson, Louise N, Mesguiche, Veronique, Noble, Martin E.M, Tucker, Julie A, Wang, Lan, Whitfield, Hayley J
Published in Nature structural & molecular biology (01.10.2002)
Published in Nature structural & molecular biology (01.10.2002)
Get full text
Journal Article
N-2-substituted O-6-cyclohexylmethylguanine derivatives: Potent inhibitors of cyclin-dependent kinases 1 and 2
Hardcastle, IR, Arris, CE, Bentley, J, Boyle, FT, Chen, YH, Curtin, NJ, Endicott, JA, Gibson, AE, Golding, BT, Griffin, RJ, Jewsbury, P, Menyerol, J, Mesguiche, Newell, DR, Noble, MEM, Pratt, DJ, Wang, LZ, Whitfield, HJ
Published in Journal of medicinal chemistry (15.07.2004)
Published in Journal of medicinal chemistry (15.07.2004)
Get full text
Journal Article
Probing the ATP Ribose-Binding Domain of Cyclin-Dependent Kinases 1 and 2 with O6-Substituted Guanine Derivatives
GIBSON, Ashleigh E., ARRIS, Christine E., BENTLEY, Johanne, BOYLE, F. Thomas, CURTIN, Nicola J., DAVIES, Thomas G., ENDICOTT, Jane A., GOLDING, Bernard T., GRANT, Sharon, GRIFFIN, Roger J., JEWSBURY, Philip, JOHNSON, Louise N., MESGUICHE, Veronique, NEWELL, David R., NOBLE, Martin E. M., TUCKER, Julie A., WHITFIELD, Hayley J.
Published in Journal of medicinal chemistry (01.08.2002)
Published in Journal of medicinal chemistry (01.08.2002)
Get full text
Journal Article
4-Alkoxy-2,6-diaminopyrimidine derivatives: inhibitors of cyclin dependent kinases 1 and 2
Mesguiche, Veronique, Parsons, Rachel J, Arris, Christine E, Bentley, Johanne, Boyle, F.Thomas, Curtin, Nicola J, Davies, Thomas G, Endicott, Jane A, Gibson, Ashleigh E, Golding, Bernard T, Griffin, Roger J, Jewsbury, Philip, Johnson, Louise N, Newell, David R, Noble, Martin E.M, Wang, Lan Z, Hardcastle, Ian R
Published in Bioorganic & medicinal chemistry letters (20.01.2003)
Published in Bioorganic & medicinal chemistry letters (20.01.2003)
Get full text
Journal Article
Resistance-Modifying Agents. 8. Inhibition of O 6-Alkylguanine-DNA Alkyltransferase by O 6-Alkenyl-, O 6-Cycloalkenyl-, and O 6-(2-Oxoalkyl)guanines and Potentiation of Temozolomide Cytotoxicity in Vitro by O 6-(1-Cyclopentenylmethyl)guanine
Griffin, Roger J, Arris, Christine E, Bleasdale, Christine, Boyle, F. Thomas, Calvert, A. Hilary, Curtin, Nicola J, Dalby, Christine, Kanugula, Sreenivas, Lembicz, Nicola K, Newell, David R, Pegg, Anthony E, Golding, Bernard T
Published in Journal of medicinal chemistry (02.11.2000)
Published in Journal of medicinal chemistry (02.11.2000)
Get full text
Journal Article
DNA interstrand cross-linking and TP53 status as determinants of tumour cell sensitivity in vitro to the antibody-directed enzyme prodrug therapy ZD2767
Monks, Noel R., Blakey, David C., East, Simon J., Dowell, Robert I., Calvete, Joanne A., Curtin, Nicola J., Arris, Christine E., Newell, David R.
Published in European journal of cancer (1990) (01.07.2002)
Published in European journal of cancer (1990) (01.07.2002)
Get full text
Journal Article
Expression of mutant and wild-type TIMP3 in primary gingival fibroblasts from Sorsby's fundus dystrophy patients
Arris, Christine E., Bevitt, Debra J., Mohamed, Jeseem, Li, Zheng, Langton, Kevin P., Barker, Michael D., Clarke, Michael P., McKie, Norman
Published in Biochimica et biophysica acta (20.05.2003)
Published in Biochimica et biophysica acta (20.05.2003)
Get full text
Journal Article
Expression of ADAMTS metalloproteinases in the retinal pigment epithelium derived cell line ARPE-19: transcriptional regulation by TNFα
Bevitt, Debra J., Mohamed, Jeseem, Catterall, Jon B., Li, Zheng, Arris, Christine E., Hiscott, Paul, Sheridan, Carl, Langton, Kevin P., Barker, Michael D., Clarke, Michael P., McKie, Norman
Published in Biochimica et biophysica acta. Gene structure and expression (15.04.2003)
Published in Biochimica et biophysica acta. Gene structure and expression (15.04.2003)
Get full text
Journal Article