Aggrecan Protects Cartilage Collagen from Proteolytic Cleavage
Pratta, Michael A., Yao, Wenqing, Decicco, Carl, Tortorella, Micky D., Liu, Riu-Qin, Copeland, Robert A., Magolda, Ronald, Newton, Robert C., Trzaskos, James M., Arner, Elizabeth C.
Published in The Journal of biological chemistry (14.11.2003)
Published in The Journal of biological chemistry (14.11.2003)
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Journal Article
Proprotein convertase activation of aggrecanases in cartilage in situ
Malfait, Anne-Marie, Arner, Elizabeth C., Song, Ruo-Hua, Alston, James T., Markosyan, Stella, Staten, Nicholas, Yang, Zhiyong, Griggs, David W., Tortorella, Micky D.
Published in Archives of biochemistry and biophysics (01.10.2008)
Published in Archives of biochemistry and biophysics (01.10.2008)
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Journal Article
Proprotein Convertase Furin Interacts with and Cleaves Pro-ADAMTS4 (Aggrecanase-1) in the trans-Golgi Network
Wang, Ping, Tortorella, Micky, England, Kristen, Malfait, Anne-Marie, Thomas, Gary, Arner, Elizabeth C., Pei, Duanqing
Published in The Journal of biological chemistry (09.04.2004)
Published in The Journal of biological chemistry (09.04.2004)
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Journal Article
High Resolution Crystal Structure of the Catalytic Domain of ADAMTS-5 (Aggrecanase-2)
Shieh, Huey-Sheng, Mathis, Karl J., Williams, Jennifer M., Hills, Robert L., Wiese, Joe F., Benson, Timothy E., Kiefer, James R., Marino, Margaret H., Carroll, Jeffery N., Leone, Joseph W., Malfait, Anne-Marie, Arner, Elizabeth C., Tortorella, Micky D., Tomasselli, Alfredo
Published in The Journal of biological chemistry (18.01.2008)
Published in The Journal of biological chemistry (18.01.2008)
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Journal Article
The Thrombospondin Motif of Aggrecanase-1 (ADAMTS-4) Is Critical for Aggrecan Substrate Recognition and Cleavage
Tortorella, Micky, Pratta, Michael, Liu, Rui-Qin, Abbaszade, Ilgar, Ross, Harold, Burn, Timothy, Arner, Elizabeth
Published in The Journal of biological chemistry (18.08.2000)
Published in The Journal of biological chemistry (18.08.2000)
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Journal Article
Sites of Aggrecan Cleavage by Recombinant Human Aggrecanase-1 (ADAMTS-4)
Tortorella, Micky D., Pratta, Michael, Liu, Rui-Qin, Austin, Julian, Ross, O.Harold, Abbaszade, Ilgar, Burn, Tim, Arner, Elizabeth
Published in The Journal of biological chemistry (16.06.2000)
Published in The Journal of biological chemistry (16.06.2000)
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Journal Article
Identification of an ADAMTS-4 Cleavage Motif Using Phage Display Leads to the Development of Fluorogenic Peptide Substrates and Reveals Matrilin-3 as a Novel Substrate
Hills, Robert, Mazzarella, Richard, Fok, Kam, Liu, Min, Nemirovskiy, Olga, Leone, Joseph, Zack, Marc D., Arner, Elizabeth C., Viswanathan, Malini, Abujoub, Aida, Muruganandam, Arumugam, Sexton, Daniel J., Bassill, Gary J., Sato, Aaron K., Malfait, Anne-Marie, Tortorella, Micky D.
Published in The Journal of biological chemistry (13.04.2007)
Published in The Journal of biological chemistry (13.04.2007)
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Journal Article
ADAMTS-4 (aggrecanase-1): N-Terminal activation mechanisms
Tortorella, Micky D., Arner, Elizabeth C., Hills, Robert, Gormley, Jennifer, Fok, Kam, Pegg, Lyle, Munie, Grace, Malfait, Anne-Marie
Published in Archives of biochemistry and biophysics (01.12.2005)
Published in Archives of biochemistry and biophysics (01.12.2005)
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Journal Article
Substrate-Dependent Inhibition Kinetics of an Active Site-Directed Inhibitor of ADAMTS-4 (Aggrecanase 1)
Wittwer, Arthur J, Hills, Robert L, Keith, Robert H, Munie, Grace E, Arner, Elizabeth C, Anglin, Charles P, Malfait, Anne-Marie, Tortorella, Micky D
Published in Biochemistry (Easton) (29.05.2007)
Published in Biochemistry (Easton) (29.05.2007)
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Journal Article
Cloning and Characterization of ADAMTS11 , an Aggrecanase from the ADAMTS Family
Abbaszade, Ilgar, Liu, Rui-Qin, Yang, Fude, Rosenfeld, Stuart A., Ross, O. Harold, Link, John R., Ellis, Dawn M., Tortorella, Micky D., Pratta, Michael A., Hollis, Jeannine M., Wynn, Richard, Duke, Jodie L., George, Henry J., Hillman, Milton C., Murphy, Kathleen, Wiswall, Barbara H., Copeland, Robert A., Decicco, Carl P., Bruckner, Robert, Nagase, Hideaki, Itoh, Yoshifumi, Newton, Robert C., Magolda, Ronald L., Trzaskos, James M., Hollis, Gregory F., Arner, Elizabeth C., Burn, Timothy C.
Published in The Journal of biological chemistry (13.08.1999)
Published in The Journal of biological chemistry (13.08.1999)
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Journal Article
Brain-enriched Hyaluronan Binding (BEHAB)/Brevican Cleavage in a Glioma Cell Line Is Mediated by a Disintegrin and Metalloproteinase with Thrombospondin Motifs (ADAMTS) Family Member
Matthews, Russell T., Gary, Sydney C., Zerillo, Cynthia, Pratta, Michael, Solomon, Kimberly, Arner, Elizabeth C., Hockfield, Susan
Published in The Journal of biological chemistry (28.07.2000)
Published in The Journal of biological chemistry (28.07.2000)
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Journal Article
Aggrecan degradation in human articular cartilage explants is mediated by both ADAMTS‐4 and ADAMTS‐5
Song, Ruo‐Hua, D. Tortorella, Micky, Malfait, Anne‐Marie, Alston, James T., Yang, Zhiyong, Arner, Elizabeth C., Griggs, David W.
Published in Arthritis and rheumatism (01.02.2007)
Published in Arthritis and rheumatism (01.02.2007)
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Journal Article
Potent and selective aggrecanase inhibitors containing cyclic P1 substituents
Cherney, Robert J, Mo, Ruowei, Meyer, Dayton T, Wang, Li, Yao, Wenqing, Wasserman, Zelda R, Liu, Rui-Qin, Covington, Maryanne B, Tortorella, Micky D, Arner, Elizabeth C, Qian, Mingxin, Christ, David D, Trzaskos, James M, Newton, Robert C, Magolda, Ron L, Decicco, Carl P
Published in Bioorganic & medicinal chemistry letters (07.04.2003)
Published in Bioorganic & medicinal chemistry letters (07.04.2003)
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Journal Article
Age-related Changes in Aggrecan Glycosylation Affect Cleavage by Aggrecanase
Pratta, Michael A., Tortorella, Micky D., Arner, Elizabeth C.
Published in The Journal of biological chemistry (15.12.2000)
Published in The Journal of biological chemistry (15.12.2000)
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Journal Article
Chondrocyte Extracellular Matrix Synthesis and Turnover Are Influenced by Static Compression in a New Alginate Disk Culture System
Ragan, Paula M., Chin, Vicki I., Hung, Han-Hwa K., Masuda, Koichi, Thonar, Eugene J.-M.A., Arner, Elizabeth C., Grodzinsky, Alan J., Sandy, John D.
Published in Archives of biochemistry and biophysics (15.11.2000)
Published in Archives of biochemistry and biophysics (15.11.2000)
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Journal Article
Amide surrogates of matrix metalloproteinase inhibitors: Urea and sulfonamide mimics
Decicco, Carl P, Seng, Jennifer L, Kennedy, Kenneth E, Covington, Maryanne B, Welch, Patty K, Arner, Elizabeth C, Magolda, Ronald L, Nelson, David J
Published in Bioorganic & medicinal chemistry letters (23.09.1997)
Published in Bioorganic & medicinal chemistry letters (23.09.1997)
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Journal Article
Design and Synthesis of a Series of (2R)-N 4-Hydroxy-2-(3-hydroxybenzyl)-N - [(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden- 1-yl]butanediamide Derivatives as Potent, Selective, and Orally Bioavailable Aggrecanase Inhibitors
Yao, Wenqing, Wasserman, Zelda R, Chao, Michael, Reddy, Gade, Shi, Eric, Liu, Rui-Qin, Covington, Maryanne B, Arner, Elizabeth C, Pratta, Michael A, Tortorella, Micky, Magolda, Ronald L, Newton, Robert, Qian, MingXin, Ribadeneira, Maria D, Christ, David, Wexler, Ruth R, Decicco, Carl P
Published in Journal of medicinal chemistry (11.10.2001)
Published in Journal of medicinal chemistry (11.10.2001)
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Journal Article
Macrocyclic Amino Carboxylates as Selective MMP-8 Inhibitors
Cherney, Robert J, Wang, Li, Meyer, Dayton T, Xue, Chu-Baio, Wasserman, Zelda R, Hardman, Karl D, Welch, Patty K, Covington, Maryanne B, Copeland, Robert A, Arner, Elizabeth C, DeGrado, William F, Decicco, Carl P
Published in Journal of medicinal chemistry (21.05.1998)
Published in Journal of medicinal chemistry (21.05.1998)
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