Clinical Probes and Endogenous Biomarkers as Substrates for Transporter Drug-Drug Interaction Evaluation: Perspectives From the International Transporter Consortium
Chu, Xiaoyan, Liao, Mingxiang, Shen, Hong, Yoshida, Kenta, Zur, Arik A, Arya, Vikram, Galetin, Aleksandra, Giacomini, Kathleen M, Hanna, Imad, Kusuhara, Hiroyuki, Lai, Yurong, Rodrigues, David, Sugiyama, Yuichi, Zamek-Gliszczynski, Maciej J, Zhang, Lei
Published in Clinical pharmacology and therapeutics (01.11.2018)
Published in Clinical pharmacology and therapeutics (01.11.2018)
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Journal Article
OCT1 is a high-capacity thiamine transporter that regulates hepatic steatosis and is a target of metformin
Chen, Ligong, Shu, Yan, Liang, Xiaomin, Chen, Eugene C., Yee, Sook Wah, Zur, Arik A., Li, Shuanglian, Xu, Lu, Keshari, Kayvan R., Lin, Michael J., Chien, Huan-Chieh, Zhang, Youcai, Morrissey, Kari M., Liu, Jason, Ostrem, Jonathan, Younger, Noah S., Kurhanewicz, John, Shokat, Keven M., Ashrafi, Kaveh, Giacomini, Kathleen M.
Published in Proceedings of the National Academy of Sciences - PNAS (08.07.2014)
Published in Proceedings of the National Academy of Sciences - PNAS (08.07.2014)
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Journal Article
Discovery of Potent, Selective Multidrug and Toxin Extrusion Transporter 1 (MATE1, SLC47A1) Inhibitors Through Prescription Drug Profiling and Computational Modeling
Wittwer, Matthias B, Zur, Arik A, Khuri, Natalia, Kido, Yasuto, Kosaka, Alan, Zhang, Xuexiang, Morrissey, Kari M, Sali, Andrej, Huang, Yong, Giacomini, Kathleen M
Published in Journal of medicinal chemistry (14.02.2013)
Published in Journal of medicinal chemistry (14.02.2013)
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Journal Article
Reevaluating the Substrate Specificity of the L‑Type Amino Acid Transporter (LAT1)
Chien, Huan-Chieh, Colas, Claire, Finke, Karissa, Springer, Seth, Stoner, Laura, Zur, Arik A., Venteicher, Brooklynn, Campbell, Jerome, Hall, Colton, Flint, Andrew, Augustyn, Evan, Hernandez, Christopher, Heeren, Nathan, Hansen, Logan, Anthony, Abby, Bauer, Justine, Fotiadis, Dimitrios, Schlessinger, Avner, Giacomini, Kathleen M., Thomas, Allen A.
Published in Journal of medicinal chemistry (23.08.2018)
Published in Journal of medicinal chemistry (23.08.2018)
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Journal Article
LAT-1 activity of meta-substituted phenylalanine and tyrosine analogs
Augustyn, Evan, Finke, Karissa, Zur, Arik A., Hansen, Logan, Heeren, Nathan, Chien, Huan-Chieh, Lin, Lawrence, Giacomini, Kathleen M., Colas, Claire, Schlessinger, Avner, Thomas, Allen A.
Published in Bioorganic & medicinal chemistry letters (01.06.2016)
Published in Bioorganic & medicinal chemistry letters (01.06.2016)
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Journal Article
Drug Metabolites Potently Inhibit Renal Organic Anion Transporters, OAT1 and OAT3
Zou, Ling, Matsson, Pär, Stecula, Adrian, Ngo, Huy X., Zur, Arik A., Giacomini, Kathleen M.
Published in Journal of pharmaceutical sciences (01.01.2021)
Published in Journal of pharmaceutical sciences (01.01.2021)
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Journal Article
LAT1 activity of carboxylic acid bioisosteres: Evaluation of hydroxamic acids as substrates
Zur, Arik A., Chien, Huan-Chieh, Augustyn, Evan, Flint, Andrew, Heeren, Nathan, Finke, Karissa, Hernandez, Christopher, Hansen, Logan, Miller, Sydney, Lin, Lawrence, Giacomini, Kathleen M., Colas, Claire, Schlessinger, Avner, Thomas, Allen A.
Published in Bioorganic & medicinal chemistry letters (15.10.2016)
Published in Bioorganic & medicinal chemistry letters (15.10.2016)
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Journal Article
The Effect of Famotidine, a MATE1-Selective Inhibitor, on the Pharmacokinetics and Pharmacodynamics of Metformin
Hibma, Jennifer E., Zur, Arik A., Castro, Richard A., Wittwer, Matthias B., Keizer, Ron J., Yee, Sook Wah, Goswami, Srijib, Stocker, Sophie L., Zhang, Xuexiang, Huang, Yong, Brett, Claire M., Savic, Radojka M., Giacomini, Kathleen M.
Published in Clinical pharmacokinetics (01.06.2016)
Published in Clinical pharmacokinetics (01.06.2016)
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Journal Article
Arcuate nucleus neuropeptide coexpression and connections to gonadotrophin‐releasing hormone neurones in the female rhesus macaque
True, C., Takahashi, D., Kirigiti, M., Lindsley, S. R., Moctezuma, C., Arik, A., Smith, M. S., Kievit, P., Grove, K. L.
Published in Journal of neuroendocrinology (01.06.2017)
Published in Journal of neuroendocrinology (01.06.2017)
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Journal Article
The effect of laquinimod, a novel immuno-modulator in development to treat Huntington disease, on the pharmacokinetics of ethinylestradiol and levonorgestrel in healthy young women
Elgart, Anna, Zur, Arik A., Mimrod, Dorit, Dror, Vered, Bar-Ilan, Oren, Korver, Tjeerd, Spiegelstein, Ofer
Published in European journal of clinical pharmacology (01.01.2019)
Published in European journal of clinical pharmacology (01.01.2019)
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Journal Article
Computational Discovery and Experimental Validation of Inhibitors of the Human Intestinal Transporter OATP2B1
Khuri, Natalia, Zur, Arik A, Wittwer, Matthias B, Lin, Lawrence, Yee, Sook Wah, Sali, Andrej, Giacomini, Kathleen M
Published in Journal of chemical information and modeling (26.06.2017)
Published in Journal of chemical information and modeling (26.06.2017)
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Journal Article
Rapid Method To Determine Intracellular Drug Concentrations in Cellular Uptake Assays: Application to Metformin in Organic Cation Transporter 1-Transfected Human Embryonic Kidney 293 Cells
Chien, Huan-Chieh, Zur, Arik A, Maurer, Tristan S, Yee, Sook Wah, Tolsma, John, Jasper, Paul, Scott, Dennis O, Giacomini, Kathleen M
Published in Drug metabolism and disposition (01.03.2016)
Published in Drug metabolism and disposition (01.03.2016)
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Journal Article
Use of multiparametric magnetic resonance imaging as a screening tool for the determination of acute ischemic stroke duration
Taner Bulut, H, Altun, Y, Arik, A, Oktay, C, Çorapli, M
Published in European review for medical and pharmacological sciences (01.02.2022)
Published in European review for medical and pharmacological sciences (01.02.2022)
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AGI-134: a fully synthetic α-Gal glycolipid that converts tumors into in situ autologous vaccines, induces anti-tumor immunity and is synergistic with an anti-PD-1 antibody in mouse melanoma models
Shaw, Stephen M, Middleton, Jenny, Wigglesworth, Kim, Charlemagne, Amber, Schulz, Oliver, Glossop, Melanie S, Whalen, Giles F, Old, Robert, Westby, Mike, Pickford, Chris, Tabakman, Rinat, Carmi-Levy, Irit, Vainstein, Abi, Sorani, Ella, Zur, Arik A, Kristian, Sascha A
Published in Cancer cell international (19.12.2019)
Published in Cancer cell international (19.12.2019)
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Journal Article
The Effect of CYP3A Induction and Inhibition on the Pharmacokinetics of Laquinimod, a Novel Neuroimmunomodulator
Elgart, Anna, Greenblatt, David J., Loupe, Pippa S., Zur, Arik A., Weiss, Sivan, Mimrod, Dorit, Spiegelstein, Ofer
Published in Clinical pharmacology in drug development (01.11.2020)
Published in Clinical pharmacology in drug development (01.11.2020)
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Journal Article
Shade estimation over streams using distributed temperature sensing
Petrides, A. C., Huff, J., Arik, A., van de Giesen, N., Kennedy, A. M., Thomas, C. K., Selker, J. S.
Published in Water resources research (01.07.2011)
Published in Water resources research (01.07.2011)
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