Discovery and Preclinical Characterization of GSK1278863 (Daprodustat), a Small Molecule Hypoxia Inducible Factor-Prolyl Hydroxylase Inhibitor for Anemia
Ariazi, Jennifer L, Duffy, Kevin J, Adams, David F, Fitch, Duke M, Luo, Lusong, Pappalardi, Melissa, Biju, Mangatt, DiFilippo, Erin Hugger, Shaw, Tony, Wiggall, Ken, Erickson-Miller, Connie
Published in The Journal of pharmacology and experimental therapeutics (01.12.2017)
Published in The Journal of pharmacology and experimental therapeutics (01.12.2017)
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Chronic inhibition of hypoxia-inducible factor prolyl 4-hydroxylase improves ventricular performance, remodeling, and vascularity after myocardial infarction in the rat
Bao, Weike, Qin, Pu, Needle, Saul, Erickson-Miller, Connie L, Duffy, Kevin J, Ariazi, Jennifer L, Zhao, Shufang, Olzinski, Alan R, Behm, David J, Pipes, G C Teg, Jucker, Beat M, Hu, Erding, Lepore, John J, Willette, Robert N
Published in Journal of cardiovascular pharmacology (01.08.2010)
Published in Journal of cardiovascular pharmacology (01.08.2010)
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Journal Article
Discovery of Tetralones as Potent and Selective Inhibitors of Acyl-CoA:Diacylglycerol Acyltransferase 1
Cheung, Mui, Tangirala, Raghuram S, Bethi, Sridhar R, Joshi, Hemant V, Ariazi, Jennifer L, Tirunagaru, Vijaya G, Kumar, Sanjay
Published in ACS medicinal chemistry letters (08.02.2018)
Published in ACS medicinal chemistry letters (08.02.2018)
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Journal Article
Mammary glands of sexually immature rats are more susceptible than those of mature rats to the carcinogenic, lethal, and mutagenic effects of N-nitroso-N-methylurea
Ariazi, Jennifer L., Haag, Jill D., Lindstrom, Mary J., Gould, Michael N.
Published in Molecular carcinogenesis (01.07.2005)
Published in Molecular carcinogenesis (01.07.2005)
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Estrogen receptors as therapeutic targets in breast cancer
Ariazi, Eric A, Ariazi, Jennifer L, Cordera, Fernando, Jordan, V Craig
Published in Current topics in medicinal chemistry (01.02.2006)
Published in Current topics in medicinal chemistry (01.02.2006)
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Rational Design, Synthesis, and SAR of a Novel Thiazolopyrimidinone Series of Selective PI3K-beta Inhibitors
Lin, Hong, Schulz, Mark J, Xie, Ren, Zeng, Jin, Luengo, Juan I, Squire, Michael D, Tedesco, Rosanna, Qu, Junya, Erhard, Karl, Mack, James F, Raha, Kaushik, Plant, Ramona, Rominger, Cynthia M, Ariazi, Jennifer L, Sherk, Christian S, Schaber, Michael D, McSurdy-Freed, Jeanelle, Spengler, Michael D, Davis, Charles B, Hardwicke, Mary Ann, Rivero, Ralph A
Published in ACS medicinal chemistry letters (12.07.2012)
Published in ACS medicinal chemistry letters (12.07.2012)
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Emerging principles for the development of resistance to antihormonal therapy: Implications for the clinical utility of fulvestrant
Ariazi, Eric A., Lewis-Wambi, Joan S., Gill, Shaun D., Pyle, Jennifer R., Ariazi, Jennifer L., Kim, Helen R., Sharma, Catherine G.N., Cordera, Fernando, Shupp, Heather A., Li, Tianyu, Jordan, V. Craig
Published in Journal of steroid biochemistry and molecular biology (01.12.2006)
Published in Journal of steroid biochemistry and molecular biology (01.12.2006)
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Conference Proceeding
Discovery of Tetralones as Potent and Selective Inhibitors of AcylCoA:Diacylglycerol Acy-ltransferase 1
Cheung, Mui, Tangirala, Raihuram S., Bethi, Sridhar R., Joshi, Hemant V., Ariazi, Jennifer L., Tirunagaru, Vijaya G., Kumar, Sanjay
Published in ACS medicinal chemistry letters (01.02.2018)
Published in ACS medicinal chemistry letters (01.02.2018)
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