Novel Therapeutic Approaches Targeting the Renin-Angiotensin System and Associated Peptides in Hypertension and Heart Failure
Arendse, Lauren B, Danser, A H Jan, Poglitsch, Marko, Touyz, Rhian M, Burnett, Jr, John C, Llorens-Cortes, Catherine, Ehlers, Mario R, Sturrock, Edward D
Published in Pharmacological reviews (01.10.2019)
Published in Pharmacological reviews (01.10.2019)
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Journal Article
Structural Basis for Inhibitor Potency and Selectivity of Plasmodium falciparum Phosphatidylinositol 4‑Kinase Inhibitors
Fienberg, Stephen, Eyermann, Charles J, Arendse, Lauren B, Basarab, Gregory S, McPhail, Jacob A, Burke, John E, Chibale, Kelly
Published in ACS infectious diseases (13.11.2020)
Published in ACS infectious diseases (13.11.2020)
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Journal Article
Developing kinase inhibitors for malaria: an opportunity or liability?
Mogwera, Koketso S.P., Chibale, Kelly, Arendse, Lauren B.
Published in Trends in parasitology (01.09.2023)
Published in Trends in parasitology (01.09.2023)
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Journal Article
Inhibition of Resistance-Refractory P. falciparum Kinase PKG Delivers Prophylactic, Blood Stage, and Transmission-Blocking Antiplasmodial Activity
Vanaerschot, Manu, Murithi, James M., Pasaje, Charisse Flerida A., Ghidelli-Disse, Sonja, Dwomoh, Louis, Bird, Megan, Spottiswoode, Natasha, Mittal, Nimisha, Arendse, Lauren B., Owen, Edward S., Wicht, Kathryn J., Siciliano, Giulia, Bösche, Markus, Yeo, Tomas, Kumar, T.R. Santha, Mok, Sachel, Carpenter, Emma F., Giddins, Marla J., Sanz, Olalla, Ottilie, Sabine, Alano, Pietro, Chibale, Kelly, Llinás, Manuel, Uhlemann, Anne-Catrin, Delves, Michael, Tobin, Andrew B., Doerig, Christian, Winzeler, Elizabeth A., Lee, Marcus C.S., Niles, Jacquin C., Fidock, David A.
Published in Cell chemical biology (16.07.2020)
Published in Cell chemical biology (16.07.2020)
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Selective Inhibition of the C-Domain of ACE (Angiotensin-Converting Enzyme) Combined With Inhibition of NEP (Neprilysin): A Potential New Therapy for Hypertension
Alves-Lopes, Rhéure, Montezano, Augusto C, Neves, Karla B, Harvey, Adam, Rios, Francisco J, Skiba, Dominik S, Arendse, Lauren B, Guzik, Tomasz J, Graham, Delyth, Poglitsch, Marko, Sturrock, Edward, Touyz, Rhian M
Published in Hypertension (Dallas, Tex. 1979) (01.09.2021)
Published in Hypertension (Dallas, Tex. 1979) (01.09.2021)
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Journal Article
Probing the Requirements for Dual Angiotensin-Converting Enzyme C‑Domain Selective/Neprilysin Inhibition
Arendse, Lauren B, Cozier, Gyles E, Eyermann, Charles J, Basarab, Gregory S, Schwager, Sylva L, Chibale, Kelly, Acharya, K. Ravi, Sturrock, Edward D
Published in Journal of medicinal chemistry (24.02.2022)
Published in Journal of medicinal chemistry (24.02.2022)
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Structural basis for the C-domain-selective angiotensin-converting enzyme inhibition by bradykinin-potentiating peptide b (BPPb)
Sturrock, Edward D, Lubbe, Lizelle, Cozier, Gyles E, Schwager, Sylva L U, Arowolo, Afolake T, Arendse, Lauren B, Belcher, Emma, Acharya, K Ravi
Published in Biochemical journal (31.05.2019)
Published in Biochemical journal (31.05.2019)
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Journal Article
The anticancer human mTOR inhibitor sapanisertib potently inhibits multiple Plasmodium kinases and life cycle stages
Arendse, Lauren B, Murithi, James M, Qahash, Tarrick, Pasaje, Charisse Flerida A, Godoy, Luiz C, Dey, Sumanta, Gibhard, Liezl, Ghidelli-Disse, Sonja, Drewes, Gerard, Bantscheff, Marcus, Lafuente-Monasterio, Maria J, Fienberg, Stephen, Wambua, Lynn, Gachuhi, Samuel, Coertzen, Dina, van der Watt, Mariëtte, Reader, Janette, Aswat, Ayesha S, Erlank, Erica, Venter, Nelius, Mittal, Nimisha, Luth, Madeline R, Ottilie, Sabine, Winzeler, Elizabeth A, Koekemoer, Lizette L, Birkholtz, Lyn-Marie, Niles, Jacquin C, Llinás, Manuel, Fidock, David A, Chibale, Kelly
Published in Science translational medicine (19.10.2022)
Published in Science translational medicine (19.10.2022)
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Journal Article
Advances in malaria pharmacology and the online guide to MALARIA PHARMACOLOGY: IUPHAR review 38
Armstrong, Jane F., Campo, Brice, Alexander, Stephen P. H., Arendse, Lauren B., Cheng, Xiu, Davenport, Anthony P., Faccenda, Elena, Fidock, David A., Godinez‐Macias, Karla P., Harding, Simon D., Kato, Nobutaka, Lee, Marcus C. S., Luth, Madeline R., Mazitschek, Ralph, Mittal, Nimisha, Niles, Jacquin C., Okombo, John, Ottilie, Sabine, Pasaje, Charisse Flerida A., Probst, Alexandra S., Rawat, Mukul, Rocamora, Frances, Sakata‐Kato, Tomoyo, Southan, Christopher, Spedding, Michael, Tye, Mark A., Yang, Tuo, Zhao, Na, Davies, Jamie A.
Published in British journal of pharmacology (01.08.2023)
Published in British journal of pharmacology (01.08.2023)
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Journal Article
Plasmodium Kinases as Potential Drug Targets for Malaria: Challenges and Opportunities
Arendse, Lauren B, Wyllie, Susan, Chibale, Kelly, Gilbert, Ian H
Published in ACS infectious diseases (12.03.2021)
Published in ACS infectious diseases (12.03.2021)
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Journal Article
New Amidated 3,6-Diphenylated Imidazopyridazines with Potent Antiplasmodium Activity Are Dual Inhibitors of Plasmodium Phosphatidylinositol-4-kinase and cGMP-Dependent Protein Kinase
Cheuka, Peter Mubanga, Centani, Luyanda, Arendse, Lauren B, Fienberg, Stephen, Wambua, Lynn, Renga, Shoneeze S, Dziwornu, Godwin Akpeko, Kumar, Malkeet, Lawrence, Nina, Taylor, Dale, Wittlin, Sergio, Coertzen, Dina, Reader, Janette, van der Watt, Mariette, Birkholtz, Lyn-Marie, Chibale, Kelly
Published in ACS infectious diseases (08.01.2021)
Published in ACS infectious diseases (08.01.2021)
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