Enhanced brain delivery of liposomal methylprednisolone improved therapeutic efficacy in a model of neuroinflammation
Gaillard, Pieter J., Appeldoorn, Chantal C.M., Rip, Jaap, Dorland, Rick, van der Pol, Susanne M.A., Kooij, Gijs, de Vries, Helga E., Reijerkerk, Arie
Published in Journal of controlled release (28.12.2012)
Published in Journal of controlled release (28.12.2012)
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Journal Article
Targeted blood-to-brain drug delivery --10 key development criteria
Gaillard, Pieter J, Visser, Corine C, Appeldoorn, Chantal C M, Rip, Jaap
Published in Current pharmaceutical biotechnology (01.09.2012)
Published in Current pharmaceutical biotechnology (01.09.2012)
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Journal Article
Glutathione PEGylated liposomal methylprednisolone (2B3-201) attenuates CNS inflammation and degeneration in murine myelin oligodendrocyte glycoprotein induced experimental autoimmune encephalomyelitis
Lee, De-Hyung, Rötger, Caroline, Appeldoorn, Chantal C.M, Reijerkerk, Arie, Gladdines, Werner, Gaillard, Pieter J, Linker, Ralf A
Published in Journal of neuroimmunology (15.09.2014)
Published in Journal of neuroimmunology (15.09.2014)
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Journal Article
Targeted CRM197-PEG-PEI/siRNA Complexes for Therapeutic RNAi in Glioblastoma
Höbel, Sabrina, Appeldoorn, Chantal C M, Gaillard, Pieter J, Aigner, Achim
Published in Pharmaceuticals (Basel, Switzerland) (16.12.2011)
Published in Pharmaceuticals (Basel, Switzerland) (16.12.2011)
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Journal Article
Gallic acid antagonizes p-selectin-mediated platelet-leukocyte interactions: Implications for the French paradox
APPELDOORN, Chantal C. M, BONNEFOY, Arnaud, LUTTERS, Bianca C. H, DAENENS, Kim, VAN BERKEL, Theo J. C, HOYLAERTS, Marc F, BIESSEN, Erik A. L
Published in Circulation (New York, N.Y.) (04.01.2005)
Published in Circulation (New York, N.Y.) (04.01.2005)
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Journal Article
Rational Optimization of a Short Human P-selectin-binding Peptide Leads to Nanomolar Affinity Antagonists
Appeldoorn, Chantal C M, Molenaar, Tom J M, Bonnefoy, Arnaud, van Leeuwen, Steven H, Vandervoort, Petra A H, Hoylaerts, Marc F, van Berkel, Theo J C, Biessen, Erik A L
Published in The Journal of biological chemistry (21.03.2003)
Published in The Journal of biological chemistry (21.03.2003)
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Journal Article
Pharmacokinetics, brain delivery, and efficacy in brain tumor-bearing mice of glutathione pegylated liposomal doxorubicin (2B3-101)
Gaillard, Pieter J, Appeldoorn, Chantal C M, Dorland, Rick, van Kregten, Joan, Manca, Francesca, Vugts, Danielle J, Windhorst, Bert, van Dongen, Guus A M S, de Vries, Helga E, Maussang, David, van Tellingen, Olaf
Published in PloS one (08.01.2014)
Published in PloS one (08.01.2014)
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Journal Article
Systemic treatment with glutathione PEGylated liposomal methylprednisolone (2B3-201) improves therapeutic efficacy in a model of ocular inflammation
Reijerkerk, Arie, Appeldoorn, Chantal C M, Rip, Jaap, de Boer, Marco, Gaillard, Pieter J
Published in Investigative ophthalmology & visual science (28.04.2014)
Published in Investigative ophthalmology & visual science (28.04.2014)
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Journal Article
Abstract 5687: Development of glutathione pegylated liposomal doxorubicin (2B3-101) for the treatment of brain cancer
Gaillard, Pieter J., Gladdines, Werner, Appeldoorn, Chantal C.M., Rip, Jaap, Boogerd, Willem J., Beijnen, Jos H., Brandsma, Dieta, van Tellingen, Olaf
Published in Cancer research (Chicago, Ill.) (15.04.2012)
Published in Cancer research (Chicago, Ill.) (15.04.2012)
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Journal Article
Inhibition of Streptococcus suis Adhesion by Dendritic Galabiose Compounds at Low Nanomolar Concentration
JOOSTEN, John A. F., LOIMARANTA, Vuokko, APPELDOORN, Chantal C. M., HAATAJA, Sauli, EL MAATE, Fatna Ait, LISKAMP, Rob M. J., FINNE, Jukka, PIETERS, Roland J.
Published in Journal of medicinal chemistry (16.12.2004)
Published in Journal of medicinal chemistry (16.12.2004)
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Journal Article
Abstract 5537: GSH-conjugation improves efficacy of Doxil against intracranial xenografts
van Tellingen, Olaf, Brandsma, Dieta, Appeldoorn, Chantal C.M., Manca, M Francesca, Rip, Jaap, Dorland, Rick, van Kregten, Joan M.R, Boogerd, Willem J., Beijnen, Jos H., Gaillard, Pieter J.
Published in Cancer research (Chicago, Ill.) (15.04.2010)
Published in Cancer research (Chicago, Ill.) (15.04.2010)
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Journal Article
Novel multivalent mannose compounds and their inhibition of the adhesion of type 1 fimbriated uropathogenic E. coli
Appeldoorn, Chantal C.M., Joosten, John A.F., Ait el Maate, Fatna, Dobrindt, Ulrich, Hacker, Jörg, Liskamp, Rob M.J., Khan, A. Salam, Pieters, Roland J.
Published in Tetrahedron: asymmetry (24.01.2005)
Published in Tetrahedron: asymmetry (24.01.2005)
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Journal Article
Specific inhibition of P-selectin–mediated cell adhesion by phage display–derived peptide antagonists
Molenaar, Tom J.M., Appeldoorn, Chantal C.M., de Haas, Sonja A.M., Michon, Ingrid N., Bonnefoy, Arnaud, Hoylaerts, Marc F., Pannekoek, Hans, van Berkel, Theo J.C., Kuiper, Johan, Biessen, Erik A.L.
Published in Blood (15.11.2002)
Published in Blood (15.11.2002)
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Journal Article
Blocking endothelial adhesion molecules: a potential therapeutic strategy to combat atherogenesis
Lutters, Bianca C H, Leeuwenburgh, Michiel A, Appeldoorn, Chantal C M, Molenaar, Tom J M, Van Berkel, Theo J C, Biessen, Erik A L
Published in Current opinion in lipidology (01.10.2004)
Published in Current opinion in lipidology (01.10.2004)
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Journal Article
Efficient degradation-aided selection of protease inhibitors by phage display
Hawinkels, Lukas J.A.C., van Rossenberg, Sabine M.W., de Jonge-Muller, Eveline S.M., Molenaar, Tom J.M., Appeldoorn, Chantal C.M., van Berkel, Theo J.C., Sier, Cornelis F.M., Biessen, Erik A.L.
Published in Biochemical and biophysical research communications (21.12.2007)
Published in Biochemical and biophysical research communications (21.12.2007)
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Journal Article
Synthesis of Highly Functionalised Carbohydrate-Derived Spiroacetals by Ring-Closing Metathesis and Pauson-Khand Reaction of Ketoglycosidic Enynes
Leeuwenburgh, Michiel A., Appeldoorn, Chantal C. M., van Hooft, Peter A. V., Overkleeft, Herman S., van der Marel, Gijsbert A., van Boom, Jacques H.
Published in European journal of organic chemistry (01.03.2000)
Published in European journal of organic chemistry (01.03.2000)
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Journal Article
Compounds binding to p-selectin
MOLENAAR THOMAS J.M, BIESSEN ERIK ANNA L, VAN BERKEL THEODORUS J.C, KUIPER JOHAN, APPELDOORN CHANTAL C.M
Year of Publication 28.09.2006
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Year of Publication 28.09.2006
Patent
Glucose-based compounds with affinity to p-selectin
MOLENAAR THOMAS J.M, VAN BERKEL THEODORUS JOSEPHUS C, APPELDOORN CHANTAL C.M, BIESSEN ERIK A.L
Year of Publication 24.11.2005
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Year of Publication 24.11.2005
Patent