Discovery of AZD-2098 and AZD-1678, Two Potent and Bioavailable CCR4 Receptor Antagonists
Kindon, Nicholas, Andrews, Glen, Baxter, Andrew, Cheshire, David, Hemsley, Paul, Johnson, Timothy, Liu, Yu-Zhen, McGinnity, Dermot, McHale, Mark, Mete, Antonio, Reuberson, James, Roberts, Bryan, Steele, John, Teobald, Barry, Unitt, John, Vaughan, Deborah, Walters, Iain, Stocks, Michael J
Published in ACS medicinal chemistry letters (14.09.2017)
Published in ACS medicinal chemistry letters (14.09.2017)
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discovery of AZD9164, a novel muscarinic M₃ antagonist
Mete, Antonio, Bowers, Keith, Chevalier, Eric, Donald, David K, Edwards, Helen, Escott, Katherine J, Ford, Rhonan, Grime, Ken, Millichip, Ian, Teobald, Barry, Russell, Vince
Published in Bioorganic & medicinal chemistry letters (15.12.2011)
Published in Bioorganic & medicinal chemistry letters (15.12.2011)
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Design and Synthesis of a Novel and Potent Series of Inhibitors of Cytosolic Phospholipase A2 Based on a 1,3-Disubstituted Propan-2-one Skeleton
Connolly, Stephen, Bennion, Colin, Botterell, Sarah, Croshaw, Pamela J, Hallam, Catherine, Hardy, Kim, Hartopp, Paul, Jackson, Clive G, King, Sarah J, Lawrence, Louise, Mete, Antonio, Murray, David, Robinson, David H, Smith, Gillian M, Stein, Linda, Walters, Iain, Wells, Edward, Withnall, W. John
Published in Journal of medicinal chemistry (14.03.2002)
Published in Journal of medicinal chemistry (14.03.2002)
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The relative rate of kill of the MMV Malaria Box compounds provides links to the mode of antimalarial action and highlights scaffolds of medicinal chemistry interest
Ullah, Imran, Sharma, Raman, Mete, Antonio, Biagini, Giancarlo A, Wetzel, Dawn M, Horrocks, Paul D
Published in Journal of antimicrobial chemotherapy (01.02.2020)
Published in Journal of antimicrobial chemotherapy (01.02.2020)
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Anchored plasticity opens doors for selective inhibitor design in nitric oxide synthase
Garcin, Elsa D, Getzoff, Elizabeth D, Arvai, Andrew S, Rosenfeld, Robin J, Kroeger, Matt D, Crane, Brian R, Andersson, Gunilla, Andrews, Glen, Hamley, Peter J, Mallinder, Philip R, Nicholls, David J, St-Gallay, Stephen A, Tinker, Alan C, Gensmantel, Nigel P, Mete, Antonio, Cheshire, David R, Connolly, Stephen, Stuehr, Dennis J, Åberg, Anders, Wallace, Alan V, Tainer, John A
Published in Nature chemical biology (01.11.2008)
Published in Nature chemical biology (01.11.2008)
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Cathepsin C Inhibitors: Property Optimization and Identification of a Clinical Candidate
Furber, Mark, Tiden, Anna-Karin, Gardiner, Philip, Mete, Antonio, Ford, Rhonan, Millichip, Ian, Stein, Linda, Mather, Andrew, Kinchin, Elizabeth, Luckhurst, Christopher, Barber, Simon, Cage, Peter, Sanganee, Hitesh, Austin, Rupert, Chohan, Kamaldeep, Beri, Raj, Thong, Bob, Wallace, Alan, Oreffo, Victor, Hutchinson, Ray, Harper, Steve, Debreczeni, Judit, Breed, Jason, Wissler, Lisa, Edman, Karl
Published in Journal of medicinal chemistry (27.03.2014)
Published in Journal of medicinal chemistry (27.03.2014)
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Asymmetric synthesis of azidotetrahydropyranols via Sharpless epoxidation
Ong, Quyen, Handa, Sheetal, Mete, Antonio, Hill, Alison M., Jones, Keith
Published in ARKIVOC (28.03.2002)
Published in ARKIVOC (28.03.2002)
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The discovery of AZD9164, a novel muscarinic M 3 antagonist
Mete, Antonio, Bowers, Keith, Chevalier, Eric, Donald, David K., Edwards, Helen, Escott, Katherine J., Ford, Rhonan, Grime, Ken, Millichip, Ian, Teobald, Barry, Russell, Vince
Published in Bioorganic & medicinal chemistry letters (15.12.2011)
Published in Bioorganic & medicinal chemistry letters (15.12.2011)
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The design of a novel series of muscarinic receptor antagonists leading to AZD8683, a potential inhaled treatment for COPD
Mete, Antonio, Bowers, Keith, Bull, Richard J., Coope, Helen, Donald, David K., Escott, Katherine J., Ford, Rhonan, Grime, Ken, Mather, Andrew, Ray, Nicholas C., Russell, Vince
Published in Bioorganic & medicinal chemistry letters (01.12.2013)
Published in Bioorganic & medicinal chemistry letters (01.12.2013)
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The discovery of novel, potent and highly selective inhibitors of inducible nitric oxide synthase (iNOS)
Cheshire, David R., Åberg, Anders, Andersson, Gunilla M.K., Andrews, Glen, Beaton, Haydn G., Birkinshaw, Timothy N., Boughton-Smith, Nigel, Connolly, Stephen, Cook, Tony R., Cooper, Anne, Cooper, Sally L., Cox, David, Dixon, John, Gensmantel, Nigel, Hamley, Peter J., Harrison, Richard, Hartopp, Paul, Käck, Helena, Leeson, Paul D., Luker, Timothy, Mete, Antonio, Millichip, Ian, Nicholls, David J., Pimm, Austen D., St-Gallay, Steve A., Wallace, Alan V.
Published in Bioorganic & medicinal chemistry letters (15.04.2011)
Published in Bioorganic & medicinal chemistry letters (15.04.2011)
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