PD-1 derived CA-170 is an oral immune checkpoint inhibitor that exhibits preclinical anti-tumor efficacy
Sasikumar, Pottayil G., Sudarshan, Naremaddepalli S., Adurthi, Srinivas, Ramachandra, Raghuveer K., Samiulla, Dodderi S., Lakshminarasimhan, Anirudha, Ramanathan, Anuradha, Chandrasekhar, Talapaneni, Dhudashiya, Amit A., Talapati, Sumalatha R., Gowda, Nagesh, Palakolanu, Sreenivasulareddy, Mani, Jiju, Srinivasrao, Bandi, Joseph, David, Kumar, Nigam, Nair, Rashmi, Atreya, Hanudatta S., Gowda, Nagaraj, Ramachandra, Murali
Published in Communications biology (08.06.2021)
Published in Communications biology (08.06.2021)
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Journal Article
Discovery of azetidine based ene-amides as potent bacterial enoyl ACP reductase (FabI) inhibitors
Takhi, Mohamed, Sreenivas, Kandepu, Reddy, Chandrashekar K., Munikumar, Mahadari, Praveena, Kolakota, Sudheer, Pabolu, Rao, Bandaru N.V.M., Ramakanth, Gollamudi, Sivaranjani, Jampala, Mulik, Shardaprasad, Reddy, Yeruva R., Narasimha Rao, Krishnamurthy, Pallavi, Rentala, Lakshminarasimhan, Anirudha, Panigrahi, Sunil K., Antony, Thomas, Abdullah, Iskandar, Lee, Yean K., Ramachandra, Murali, Yusof, Rohana, Rahman, Noorsaadah A., Subramanya, Hosahalli
Published in European journal of medicinal chemistry (12.09.2014)
Published in European journal of medicinal chemistry (12.09.2014)
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Journal Article
Sofosbuvir and its tri-phosphate metabolite inhibit the RNA-dependent RNA polymerase activity of non-structural protein 5 from the Kyasanur forest disease virus
Malik, Mansi, Vijayan, Parvathy, Jagannath, Deepak K., Mishra, Rakesh K., Lakshminarasimhan, Anirudha
Published in Biochemical and biophysical research communications (22.01.2023)
Published in Biochemical and biophysical research communications (22.01.2023)
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Journal Article
Nano-differential scanning fluorimetry as a tool for the assessment of refolded antibody fragments: A case study for anti-Pfs25 single-chain antibodies
Khera, Harvinder Kour, Valiyaparambil, Ashwathi, Jagannath, Deepak K., Viswanath, Vysakh K., Kumar, Naveen, Shukla, Jay Prakash, Pradhan, Sabyasachi, Lakshminarasimhan, Anirudha
Published in Biochemical engineering journal (01.06.2024)
Published in Biochemical engineering journal (01.06.2024)
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Journal Article
Refolding and characterization of a diabody against Pfs25, a vaccine candidate of Plasmodium falciparum
Jagannath, Deepak K., Valiyaparambil, Ashwathi, Viswanath, Vysakh K., Hurakadli, Manjunath A., Kamariah, Neelagandan, Jafer, Alifia C., Patole, Chhaya, Pradhan, Sabyasachi, Kumar, Naveen, Lakshminarasimhan, Anirudha
Published in Analytical biochemistry (15.10.2022)
Published in Analytical biochemistry (15.10.2022)
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Journal Article
Ternary complex formation of AFN‐1252 with Acinetobacter baumannii FabI and NADH: Crystallographic and biochemical studies
Rao, Narasimha K, Nataraj, Vijayashankar, Ravi, Mohan, Panchariya, Love, Palai, Kirttija, Talapati, Sumalatha R., Lakshminarasimhan, Anirudha, Ramachandra, Murali, Antony, Thomas
Published in Chemical biology & drug design (01.08.2020)
Published in Chemical biology & drug design (01.08.2020)
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Journal Article
Abstract B007: Potent antitumor activity of a novel and orally available small-molecule antagonist targeting the CD47/SIRPα pathway
Sasikumar, Pottayil G., Gundala, Chennakrishnareddy, Balasubramanian, Wesley R., Naremaddepalli, Sudarshan S., Bhumireddy, Archana, Patil, Sandeep S., Dhudashiya, Amit A., Rayavarapu, Vijaysai, Lakshminarasimhan, Anirudha, Samiulla, Dodheri S., Aithal, Kiran, Daginakatte, Girish, Ramachandra, Murali
Published in Molecular cancer therapeutics (01.01.2018)
Published in Molecular cancer therapeutics (01.01.2018)
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Journal Article
Abstract 1650: Targeting CD47- SIRPα interaction by novel peptide-based antagonists
Sasikumar, Pottayil G., Gundala, Chennakrishnareddy, Gowda, Nagaraj M., Naremaddepalli, Sudarshan S., Bhumireddy, Archana, Nair, Rashmi, Balasubramanian, Wesley Roy, Lakshminarasimhan, Anirudha, Dodheri, Samiulla S., Aithal, Kiran, Ramachandra, Raghuveer K., Daginakatte, Girish, Ramachandra, Murali
Published in Cancer research (Chicago, Ill.) (01.07.2017)
Published in Cancer research (Chicago, Ill.) (01.07.2017)
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Journal Article
Abstract 5108: Potent small molecule compounds that selectively inhibit proliferation of ABC-DLBCL cell lines
Satyam, Leena Khare, Chikkanna, Dinesh, Khairnar, Vinayak, Pothuganti, Manoj, Panigrahi, Sunil, Lakshminarasimhan, Anirudha, Rao, Narasimha, Balasubramanian, Wesley, Patil, Sandeep, Gopinath, Sreevalsam, Upendra, Gunta, Nagaraj, Jwala, Aithal, Kiran, Ahuja, Vijay, Giri, Sanjeev, Pandit, Chetan, Ramachandra, Murali
Published in Cancer research (Chicago, Ill.) (01.07.2017)
Published in Cancer research (Chicago, Ill.) (01.07.2017)
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Journal Article
Abstract 1392: Preclinical In vivo evaluation of efficacy, pharmacokinetics and pharmacodynamics of novel PRMT5 inhibitors in multiple tumor models
Chikkanna, Dinesh, Panigrahi, Sunil Kumar, Rajagopalan, Sujatha, Sammeta, Srinivasa Raju, Chawla, Darshan, S, Pavithra, D.S, Samiulla, Prasanna, Angelene, Chand, Priyabrata, Aithal, Kiran, Marri, Sai Sudheer, Kumar, Naveen, Ganipisetty, Srinivasa Rao, Mutyala, Raju, Rao, Kasieswara, Antony, Thomas, Daginakatte, Girish, Lakshminarasimhan, Anirudha, R, Mohan, K, Narasihmarao, Chelur, Shekar, Pandit, Chetan, Samajdar, Susanta, Ramachandra, Murali
Published in Cancer research (Chicago, Ill.) (01.07.2018)
Published in Cancer research (Chicago, Ill.) (01.07.2018)
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Journal Article
Abstract A174: Novel inhibitors of protein arginine methyltransferase 5 (PRMT5) for the treatment of solid tumors
Chikkanna, Dinesh, Panigrahi, Sunil Kumar, Rajagopalan, Sujatha, Sammeta, Srinivasa Raju, Lakshminarasimhan, Anirudha, R, Mohan, K, Narasihmarao, Chawla, Darshan, Bhat, Harsha, Kasturi, Venkateswarlu, D.S, Samiulla, Prasanna, Angelene, Aithal, Kiran, Chand, Priyabrata Chand, Kumar, Naveen, Marri, Sai Sudheer, Ganipisetty, Srinivasa Rao, N, Kasieswara Rao, Mutyala, Raju, Neerukattu, Nageswara Rao, K, Nithesh, Amin, Ramya, Gorade, Priyanka Machhindra, Antony, Thomas, Daginakatte, Girish, Chelur, Shekar, Pandit, Chetan, Samajdar, Susanta, Ramachandra, Murali
Published in Molecular cancer therapeutics (01.01.2018)
Published in Molecular cancer therapeutics (01.01.2018)
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Journal Article
Abstract A72: Novel NAMPT inhibitors for the treatment of Pancreatic cancer
Chikanna, Dinesh, Lakshminarasimhan, Anirudha, Khairnar, Vinayak, Panigrahi, Sunil, Ramanathan, Anuradha, Rao, Narasimha, Narayanan, Kishore, Gopinath, Sreevalsam, Ramachandra, Raghuveer, Chelur, Shekar, Pandit, Chetan, Ramachandra, Murali
Published in Molecular cancer research (01.01.2016)
Published in Molecular cancer research (01.01.2016)
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Journal Article
Structure-guided discovery of 2-aryl/pyridin-2-yl-1H-indole derivatives as potent and selective hepsin inhibitors
Goswami, Rajeev, Wohlfahrt, Gerd, Törmäkangas, Olli, Moilanen, Anu, Lakshminarasimhan, Anirudha, Nagaraj, Jwala, Arumugam, Karthikeyan N., Mukherjee, Subhendu, Chacko, Anita R., Krishnamurthy, Narasimha R., Jaleel, Mahaboobi, Palakurthy, Rajendra K., Samiulla, Dodheri S., Ramachandra, Murali
Published in Bioorganic & medicinal chemistry letters (15.11.2015)
Published in Bioorganic & medicinal chemistry letters (15.11.2015)
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Journal Article
AFN-1252 is a potent inhibitor of enoyl-ACP reductase from Burkholderia pseudomallei--Crystal structure, mode of action, and biological activity
Rao, Krishnamurthy Narasimha, Lakshminarasimhan, Anirudha, Joseph, Sarah, Lekshmi, Swathi U, Lau, Ming-Seong, Takhi, Mohammed, Sreenivas, Kandepu, Nathan, Sheila, Yusof, Rohana, Abd Rahman, Noorsaadah, Ramachandra, Murali, Antony, Thomas, Subramanya, Hosahalli
Published in Protein science (01.05.2015)
Published in Protein science (01.05.2015)
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Journal Article
Abstract 5367: Discovery of dihydro-isoxazole derivatives as novel inhibitors of NAMPT for the treatment of multiple myeloma
Chikkanna, Dinesh, Lakshminarasimhan, Anirudha, Khairnar, Vinayak, panigrahi, Sunil, Ramanathan, Anuradha, Rani, Sumalatha, Rao, Narasimha, S, Karthikeyan, Narayanan, Kishore, Gopinath, Sreevalsam, Ramachandra, Raghuveer, K B, Charamanna, Chelur, Shekar, Pandit, Chetan, Ramachandra, Murali
Published in Cancer research (Chicago, Ill.) (01.08.2015)
Published in Cancer research (Chicago, Ill.) (01.08.2015)
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Journal Article
Abstract C190: Potent and selective inhibition of CDK7 by novel covalent inhibitors
Poddutoori, Ramulu, Satyam, Leena K., Daginakatte, Girish, Mukherjee, Subhendu, Marappan, Sivapriya, Gopinath, Sreevalsam, Ramachandra, Raghuveer, Lakshminarasimhan, Anirudha, Pothuganti, Manoj, Nayak, Shilpa, C, Nandish, Naik, Chandranath, MV, Ravindra, Dabbeeru, Madhu, Antony, Thomas, Pandit, Chetan, Ramachandra, Murali, Chelur, Shekar, Samajdar, Susanta
Published in Molecular cancer therapeutics (01.12.2015)
Published in Molecular cancer therapeutics (01.12.2015)
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Journal Article
Abstract 339: Identification of novel covalent inhibitors of K-Ras G12C that are efficacious in a xenograft model of NSCLC
Satyam, Leena Khare, Chikkanna, Dinesh, G, Aswani K., Khairnar, Vinayak V., Reddy, Sreekanth, Durgaprasad, Vakkapatla, Radhakrishna, Kowju, Panigrahi, Sunil K., Ramanathan, Anuradha, Mahasweta, Kumari, Lakshminarasimhan, Anirudha, K, Narasimha R., R, Vinutha, Gopinath, Sreevalsam, Kumar, Suryakant, Shah, Mubarak H., Ramachandra, Raghuveer, B, Kiran A., Pandit, Chetan, Ramachandra, Murali
Published in Cancer research (Chicago, Ill.) (15.07.2016)
Published in Cancer research (Chicago, Ill.) (15.07.2016)
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