A screen against Leishmania intracellular amastigotes: comparison to a promastigote screen and identification of a host cell-specific hit
De Muylder, Geraldine, Ang, Kenny K H, Chen, Steven, Arkin, Michelle R, Engel, Juan C, McKerrow, James H
Published in PLoS neglected tropical diseases (01.07.2011)
Published in PLoS neglected tropical diseases (01.07.2011)
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Journal Article
Diverse inhibitor chemotypes targeting Trypanosoma cruzi CYP51
Gunatilleke, Shamila S, Calvet, Claudia M, Johnston, Jonathan B, Chen, Chiung-Kuang, Erenburg, Grigori, Gut, Jiri, Engel, Juan C, Ang, Kenny K H, Mulvaney, Joseph, Chen, Steven, Arkin, Michelle R, McKerrow, James H, Podust, Larissa M
Published in PLoS neglected tropical diseases (01.07.2012)
Published in PLoS neglected tropical diseases (01.07.2012)
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Journal Article
Mining a cathepsin inhibitor library for new antiparasitic drug leads
Ang, Kenny K H, Ratnam, Joseline, Gut, Jiri, Legac, Jennifer, Hansell, Elizabeth, Mackey, Zachary B, Skrzypczynska, Katarzyna M, Debnath, Anjan, Engel, Juan C, Rosenthal, Philip J, McKerrow, James H, Arkin, Michelle R, Renslo, Adam R
Published in PLoS neglected tropical diseases (01.05.2011)
Published in PLoS neglected tropical diseases (01.05.2011)
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Journal Article
An image-based assay for high throughput screening of Giardia lamblia
Gut, Jiri, Ang, Kenny K.H., Legac, Jennifer, Arkin, Michelle R., Rosenthal, Philip J., McKerrow, James H.
Published in Journal of microbiological methods (01.03.2011)
Published in Journal of microbiological methods (01.03.2011)
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Journal Article
UCSF Small Molecule Discovery Center: Innovation, Collaboration and Chemical Biology in the Bay Area
Arkin, Michelle R, Ang, Kenny K H, Chen, Steven, Davies, Julia, Merron, Connie, Tang, Yinyan, Wilson, Christopher G M, Renslo, Adam R
Published in Combinatorial chemistry & high throughput screening (01.05.2014)
Published in Combinatorial chemistry & high throughput screening (01.05.2014)
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Pharmacological brake-release of mRNA translation enhances cognitive memory
Sidrauski, Carmela, Acosta-Alvear, Diego, Khoutorsky, Arkady, Vedantham, Punitha, Hearn, Brian R, Li, Han, Gamache, Karine, Gallagher, Ciara M, Ang, Kenny K-H, Wilson, Chris, Okreglak, Voytek, Ashkenazi, Avi, Hann, Byron, Nader, Karim, Arkin, Michelle R, Renslo, Adam R, Sonenberg, Nahum, Walter, Peter
Published in eLife (28.05.2013)
Published in eLife (28.05.2013)
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Image-Based High-Throughput Drug Screening Targeting the Intracellular Stage of Trypanosoma cruzi, the Agent of Chagas' Disease
Engel, Juan C, Ang, Kenny K H, Chen, Steven, Arkin, Michelle R, McKerrow, James H, Doyle, Patricia S
Published in Antimicrobial Agents and Chemotherapy (01.08.2010)
Published in Antimicrobial Agents and Chemotherapy (01.08.2010)
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Journal Article
A gene-expression screen identifies a non-toxic sumoylation inhibitor that mimics SUMO-less human LRH-1 in liver
Suzawa, Miyuki, Miranda, Diego A, Ramos, Karmela A, Ang, Kenny K-H, Faivre, Emily J, Wilson, Christopher G, Caboni, Laura, Arkin, Michelle R, Kim, Yeong-Sang, Fletterick, Robert J, Diaz, Aaron, Schneekloth, John S, Ingraham, Holly A
Published in eLife (11.12.2015)
Published in eLife (11.12.2015)
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Journal Article
Novel non-peptidic vinylsulfones targeting the S2 and S3 subsites of parasite cysteine proteases
Bryant, Clifford, Kerr, Iain D., Debnath, Moumita, Ang, Kenny K.H., Ratnam, Joseline, Ferreira, Rafaela S., Jaishankar, Priyadarshini, Zhao, DongMei, Arkin, Michelle R., McKerrow, James H., Brinen, Linda S., Renslo, Adam R.
Published in Bioorganic & medicinal chemistry letters (01.11.2009)
Published in Bioorganic & medicinal chemistry letters (01.11.2009)
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Journal Article
Trypanosoma cruzi CYP51 inhibitor derived from a Mycobacterium tuberculosis screen hit
Chen, Chiung-Kuang, Doyle, Patricia S, Yermalitskaya, Liudmila V, Mackey, Zachary B, Ang, Kenny K H, McKerrow, James H, Podust, Larissa M
Published in PLoS neglected tropical diseases (2009)
Published in PLoS neglected tropical diseases (2009)
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Journal Article
In Vivo Antimalarial Activity of the Beta-Carboline Alkaloid Manzamine A
Ang, K K, Holmes, M J, Higa, T, Hamann, M T, Kara, U A
Published in Antimicrobial Agents and Chemotherapy (01.06.2000)
Published in Antimicrobial Agents and Chemotherapy (01.06.2000)
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Chemical-biological characterization of a cruzain inhibitor reveals a second target and a mammalian off-target
Choy, Jonathan W, Bryant, Clifford, Calvet, Claudia M, Doyle, Patricia S, Gunatilleke, Shamila S, Leung, Siegfried S F, Ang, Kenny K H, Chen, Steven, Gut, Jiri, Oses-Prieto, Juan A, Johnston, Jonathan B, Arkin, Michelle R, Burlingame, Alma L, Taunton, Jack, Jacobson, Matthew P, McKerrow, James M, Podust, Larissa M, Renslo, Adam R
Published in Beilstein journal of organic chemistry (04.01.2013)
Published in Beilstein journal of organic chemistry (04.01.2013)
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Journal Article
Guidelines for DNA recombination and repair studies: Mechanistic assays of DNA repair processes
Klein, Hannah L, Ang, Kenny K H, Arkin, Michelle R, Beckwitt, Emily C, Chang, Yi-Hsuan, Fan, Jun, Kwon, Youngho, Morten, Michael J, Mukherjee, Sucheta, Pambos, Oliver J, El Sayyed, Hafez, Thrall, Elizabeth S, Vieira-da-Rocha, João P, Wang, Quan, Wang, Shuang, Yeh, Hsin-Yi, Biteen, Julie S, Chi, Peter, Heyer, Wolf-Dietrich, Kapanidis, Achillefs N, Loparo, Joseph J, Strick, Terence R, Sung, Patrick, Van Houten, Bennett, Niu, Hengyao, Rothenberg, Eli
Published in Microbial cell (07.01.2019)
Published in Microbial cell (07.01.2019)
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New Antiinfective and Human 5-HT2 Receptor Binding Natural and Semisynthetic Compounds from the Jamaican Sponge Smenospongia aurea
HU, Jin-Feng, SCHETZ, John A., KELLY, Michelle, PENG, Jiang-Nan, ANG, Kenny K. H., FLOTOW, Horst, LEONG, Chung Yan, NG, Siew Bee, BUSS, Antony D., WILKINS, Scott P., HAMANN, Mark T.
Published in Journal of natural products (Washington, D.C.) (01.04.2002)
Published in Journal of natural products (Washington, D.C.) (01.04.2002)
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Journal Article
A benzopyrroloisoquinoline alkaloid from Ficus fistulosa
Subramaniam, G., Ang, Kenny K.H., Ng, Siewbee, Buss, Antony D., Butler, Mark S.
Published in Phytochemistry letters (29.04.2009)
Published in Phytochemistry letters (29.04.2009)
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