Discovery of 2‑[1-(4,4-Difluorocyclohexyl)piperidin-4-yl]-6-fluoro-3-oxo-2,3-dihydro‑1H‑isoindole-4-carboxamide (NMS-P118): A Potent, Orally Available, and Highly Selective PARP‑1 Inhibitor for Cancer Therapy
Papeo, Gianluca, Posteri, Helena, Borghi, Daniela, Busel, Alina A., Caprera, Francesco, Casale, Elena, Ciomei, Marina, Cirla, Alessandra, Corti, Emiliana, D’Anello, Matteo, Fasolini, Marina, Forte, Barbara, Galvani, Arturo, Isacchi, Antonella, Khvat, Alexander, Krasavin, Mikhail Y., Lupi, Rosita, Orsini, Paolo, Perego, Rita, Pesenti, Enrico, Pezzetta, Daniele, Rainoldi, Sonia, Riccardi-Sirtori, Federico, Scolaro, Alessandra, Sola, Francesco, Zuccotto, Fabio, Felder, Eduard R., Donati, Daniele, Montagnoli, Alessia
Published in Journal of medicinal chemistry (10.09.2015)
Published in Journal of medicinal chemistry (10.09.2015)
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Journal Article
Cdc7 Kinase Inhibitors: 5-Heteroaryl-3-Carboxamido-2-Aryl Pyrroles as Potential Antitumor Agents. 1. Lead Finding
Menichincheri, Maria, Albanese, Clara, Alli, Cristina, Ballinari, Dario, Bargiotti, Alberto, Caldarelli, Marina, Ciavolella, Antonella, Cirla, Alessandra, Colombo, Maristella, Colotta, Francesco, Croci, Valter, D’Alessio, Roberto, D’Anello, Matteo, Ermoli, Antonella, Fiorentini, Francesco, Forte, Barbara, Galvani, Arturo, Giordano, Patrizia, Isacchi, Antonella, Martina, Katia, Molinari, Antonio, Moll, Jürgen K, Montagnoli, Alessia, Orsini, Paolo, Orzi, Fabrizio, Pesenti, Enrico, Pillan, Antonio, Roletto, Fulvia, Scolaro, Alessandra, Tatò, Marco, Tibolla, Marcellino, Valsasina, Barbara, Varasi, Mario, Vianello, Paola, Volpi, Daniele, Santocanale, Corrado, Vanotti, Ermes
Published in Journal of medicinal chemistry (28.10.2010)
Published in Journal of medicinal chemistry (28.10.2010)
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Discovery and optimization of pyrrolo[1,2-a]pyrazinones leads to novel and selective inhibitors of PIM kinases
Casuscelli, Francesco, Ardini, Elena, Avanzi, Nilla, Casale, Elena, Cervi, Giovanni, D’Anello, Matteo, Donati, Daniele, Faiardi, Daniela, Ferguson, Ronald D., Fogliatto, Gianpaolo, Galvani, Arturo, Marsiglio, Aurelio, Mirizzi, Danilo G., Montemartini, Marisa, Orrenius, Christian, Papeo, Gianluca, Piutti, Claudia, Salom, Barbara, Felder, Eduard R.
Published in Bioorganic & medicinal chemistry (01.12.2013)
Published in Bioorganic & medicinal chemistry (01.12.2013)
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Thieno[3,2- c]pyrazoles: A novel class of Aurora inhibitors with favorable antitumor activity
Bindi, Simona, Fancelli, Daniele, Alli, Cristina, Berta, Daniela, Bertrand, Jay A., Cameron, Alexander D., Cappella, Paolo, Carpinelli, Patrizia, Cervi, Giovanni, Croci, Valter, D’Anello, Matteo, Forte, Barbara, Laura Giorgini, M., Marsiglio, Aurelio, Moll, Juergen, Pesenti, Enrico, Pittalà, Valeria, Pulici, Maurizio, Riccardi-Sirtori, Federico, Roletto, Fulvia, Soncini, Chiara, Storici, Paola, Varasi, Mario, Volpi, Daniele, Zugnoni, Paola, Vianello, Paola
Published in Bioorganic & medicinal chemistry (01.10.2010)
Published in Bioorganic & medicinal chemistry (01.10.2010)
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Application of computer vision systems for assessing bergamot fruit external features
Benalia, S, Calogero, V, Anello, M, Zimbalatti, G, Bernardi, B
Published in Advances in horticultural science (01.03.2023)
Published in Advances in horticultural science (01.03.2023)
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Abstract 4785: NMS-E668, a highly potent orally available RET inhibitor with selectivity towards VEGFR2 and demonstrated antitumor efficacy in multiple RET-driven cancer models
Ardini, Elena, Banfi, Patrizia, Avanzi, Nilla, Ciomei, Marina, Polucci, Paolo, Cirla, Alessandra, D'Anello, Matteo, Borgia, Andrea Lombardi, Motto, Ilaria, Cristiani, Cinzia, Ballinari, Dario, Felder, Eduard, Donati, Daniele, Galvani, Arturo, Isacchi, Antonella, Menichincheri, Maria
Published in Cancer research (Chicago, Ill.) (01.07.2018)
Published in Cancer research (Chicago, Ill.) (01.07.2018)
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Journal Article
Discovery of 2-[1-(4,4-Difluorocyclohexyl)piperidin-4-yl]-6-fluoro-3-oxo-2,3-dihydro-1 H -isoindole-4-carboxamide (NMS-P118): A Potent, Orally Available, and Highly Selective PARP-1 Inhibitor for Cancer Therapy
Papeo, Gianluca, Posteri, Helena, Borghi, Daniela, Busel, Alina A., Caprera, Francesco, Casale, Elena, Ciomei, Marina, Cirla, Alessandra, Corti, Emiliana, D’Anello, Matteo, Fasolini, Marina, Forte, Barbara, Galvani, Arturo, Isacchi, Antonella, Khvat, Alexander, Krasavin, Mikhail Y., Lupi, Rosita, Orsini, Paolo, Perego, Rita, Pesenti, Enrico, Pezzetta, Daniele, Rainoldi, Sonia, Riccardi-Sirtori, Federico, Scolaro, Alessandra, Sola, Francesco, Zuccotto, Fabio, Felder, Eduard R., Donati, Daniele, Montagnoli, Alessia
Published in Journal of medicinal chemistry (10.09.2015)
Published in Journal of medicinal chemistry (10.09.2015)
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Journal Article
Compuestos derivados de 3-fenil-isoquinolin-1(2h)-ona, inhibidores de parp-1; procedimiento de preparacion; composicion farmaceutica; y uso en el tratamiento del cancer
CIRLA, ALESSANDRA, D´ANELLO, MATTEO, PAPEO, GIANLUCA MARIANO ENRICO, SCOLARO, ALESSANDRA, ZUCCOTTO, FABIO
Year of Publication 05.09.2014
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Year of Publication 05.09.2014
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New salt of N-(2,6-diethylphenyl)-8-({4-(4-(dimethylamino)piperidin-1-yl)-2-methoxyphenyl}am ino)-1-methyl-4,5-dihydro-1H-pyrazolo(4,3-h)quinazoline-3-carboxamide, its preparation and formulations containing it
CANDIANI, Ilaria, D'ANELLO, Matteo, CALDARELLI, Marina, ZAMPIERI, Massimo, D'ARASMO, Germano
Year of Publication 14.07.2022
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Year of Publication 14.07.2022
Patent
NEW SALT OF N-(2,6-DIETHYLPHENYL)-8-({4-[4-(DIMETHYLAMINO)PIPERIDIN-1-YL]-2-METHOXYPHENYL}AMINO)-1-METHYL-4,5-DIHYDRO-1H-PYRAZOLO[4,3-H]QUINAZOLINE-3-CARBOXAMIDE, ITS PREPARATION AND FORMULATIONS CONTAINING IT
CALDARELLI, MARINA, ZAMPIERI, MASSIMO, D'ARASMO, GERMANO, CANDIANI, ILARIA, D'ANELLO, MATTEO
Year of Publication 19.04.2022
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Year of Publication 19.04.2022
Patent
SALT OF N-(2,6-DIETHYLPHENYL)-8-({4-[4-(DIMETHYLAMINO)PIPERIDIN-1-YL]-2-METHOXYPHENYL}AMINO)-1-METHYL-4,5-DIHYDRO-1H-PYRAZOLO[4,3-h]QUINAZOLINE-3-CARBOXAMIDE, ITS PREPARATION AND FORMULATIONS CONTAINING IT
CANDIANI, Ilaria, D'ANELLO, Matteo, CALDARELLI, Marina, ZAMPIERI, Massimo, D'ARASMO, Germano
Year of Publication 11.03.2022
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Year of Publication 11.03.2022
Patent
New salt of N-(2,6-diethylphenyl)-8-({4-(4-(dimethylamino)piperidin-1-yl)-2-methoxyphenyl}am ino)-1-methyl-4,5-dihydro-1H-pyrazolo(4,3-h)quinazoline-3-carboxamide, its preparation and formulations containing it
CANDIANI, Ilaria, D'ANELLO, Matteo, CALDARELLI, Marina, ZAMPIERI, Massimo, D'ARASMO, Germano
Year of Publication 10.03.2022
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Year of Publication 10.03.2022
Patent
SALT OF N-(2,6-DIETHYLPHENYL)-8-({4-[4-(DIMETHYLAMINO) PIPERIDIN-1-YL]-2-METHOXYPHENYL}AMINO)-1-METHYL-4,5-DIHYDRO-1H-PYRAZOLO[4,3-h]QUINAZOLINE-3-CARBOXAMIDE, ITS PREPARATION, AND FORMULATIONS CONTAINING IT
CANDIANI, Ilaria, D'ANELLO, Matteo, CALDARELLI, Marina, ZAMPIERI, Massimo, D'ARASMO, Germano
Year of Publication 20.01.2022
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Year of Publication 20.01.2022
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SUBSTITUTED 3-AMINO INDAZOLE DERIVATIVES AS KINASE INHIBITORS
POLUCCI, Paolo, SALSA, Matteo, MENICHINCHERI, Maria, D'ANELLO, Matteo, FAIARDI, Daniela, MOTTO, Ilaria
Year of Publication 05.10.2023
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Year of Publication 05.10.2023
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Salt of N-(2,6-diethylphenyl)-8-({4-[4-(dimethylamino) piperidin-1-yl]-2-methoxyphenyl}amino)-1-methyl-4,5-dihydro-1H-pyrazolo[4,3-h]quinazoline-3-carboxamide, its preparation, and formulations containing it
D'Arasmo, Germano, Candiani, Ilaria, Caldarelli, Marina, Zampieri, Massimo, D'Anello, Matteo
Year of Publication 02.11.2021
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Year of Publication 02.11.2021
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NEW SALT OF N-(2,6-DIETHYLPHENYL)-8-({4-[4-(DIMETHYLAMINO)PIPERIDIN-1-YL]-2-METHOXYPHENYL}AMINO)-1-METHYL-4,5-DIHYDRO-1H-PYRAZOLO[4,3-H]QUINAZOLINE-3-CARBOXAMIDE, ITS PREPARATION AND FORMULATIONS CONTAINING IT
CANDIANI, Ilaria, D'ANELLO, Matteo, CALDARELLI, Marina, ZAMPIERI, Massimo, D'ARASMO, Germano
Year of Publication 08.09.2021
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Year of Publication 08.09.2021
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NOUVEAU SEL DE N-(2,6-DIÉTHYLPHÉNYL)-8-((4-4-(DIMÉTHYLAMINO)PIPÉRIDINE-1-YL]-2-MÉTHOXYPHÉNYL)AMINO)-1-MÉTHYL-4,5-DIHYDRO-1H-PYRAZOLO[4,3-H]QUINAZOLINE-3-CARBOXAMIDE, SA PRÉPARATION ET FORMULATIONS LE CONTENANT
CANDIANI, Ilaria, D'ANELLO, Matteo, CALDARELLI, Marina, D'ARASMO, Germano, ZAMPIERI, Massimo
Year of Publication 26.05.2021
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Year of Publication 26.05.2021
Patent