Discovery of a series of imidazopyrazine small molecule inhibitors of the kinase MAPKAPK5, that show activity using in vitro and in vivo models of rheumatoid arthritis
Andrews, Martin J.I., Andrew Clase, J., Bar, Gregory, Tricarico, Giovanni, Edwards, Paul J., Brys, Reginald, Chambers, Mark, Schmidt, Wolfgang, MacLeod, Angus, Hirst, Kim, Allen, Vivienne, Birault, Veronique, Le, Joelle, Harris, John, Self, Andrew, Nash, Kevin, Dixon, Graham
Published in Bioorganic & medicinal chemistry letters (15.03.2012)
Published in Bioorganic & medicinal chemistry letters (15.03.2012)
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Journal Article
Design, synthesis, biological activity and structural analysis of cyclic peptide inhibitors targeting the substrate recruitment site of cyclin-dependent kinase complexes
Andrews, MJI, McInnes, C, Kontopidis, G, Innes, L, Cowan, A, Plater, A, Fischer, PM
Published in Organic & biomolecular chemistry (01.01.2004)
Published in Organic & biomolecular chemistry (01.01.2004)
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Journal Article
A large simple randomized trial of rocuronium versus succinylcholine in rapid-sequence induction of anaesthesia along with propofol
Andrews, J. I., Kumar, N., Van Den Brom, R. H. G., Olkkola, K. T., Roest, G. J., Wright, P. M. C.
Published in Acta anaesthesiologica Scandinavica (01.01.1999)
Published in Acta anaesthesiologica Scandinavica (01.01.1999)
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Journal Article
REPLACE: A Strategy for Iterative Design of Cyclin-Binding Groove Inhibitors
Andrews, Martin J.I, Kontopidis, George, McInnes, Campbell, Plater, Andy, Innes, Lorraine, Cowan, Angela, Jewsbury, Philip, Fischer, Peter M
Published in Chembiochem : a European journal of chemical biology (01.12.2006)
Published in Chembiochem : a European journal of chemical biology (01.12.2006)
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Journal Article
Obesity and prognosis in endometrial cancer
Anderson, Barrie, Connor, Joseph P., Andrews, Janet I., Davis, Charles S., Buller, Richard E., Sorosky, Joel I., Benda, Jo A.
Published in American journal of obstetrics and gynecology (01.04.1996)
Published in American journal of obstetrics and gynecology (01.04.1996)
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Journal Article
Computed tomography in endometrial carcinoma
Connor, Joseph P, Andrews, Janet I, Anderson, Barrie, Buller, Richard E
Published in Obstetrics and gynecology (New York. 1953) (01.05.2000)
Published in Obstetrics and gynecology (New York. 1953) (01.05.2000)
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Journal Article
West of Shetland revisited: the search for stratigraphic traps
Loizou, N., Andrews, I. J., Stoker, S. J., Cameron, D.
Published in Deliberate Search for the Stratigraphic Trap (2006)
Published in Deliberate Search for the Stratigraphic Trap (2006)
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Book Chapter
Journal Article
Group B streptococci causing neonatal bloodstream infection: Antimicrobial susceptibility and serotyping results from SENTRY centers in the Western Hemisphere
Andrews, Janet I., Diekema, Daniel J., Hunter, Stephen K., Rhomberg, Paul R., Pfaller, Michael A., Jones, Ronald N., Doern, Gary V.
Published in American journal of obstetrics and gynecology (01.10.2000)
Published in American journal of obstetrics and gynecology (01.10.2000)
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Journal Article
Conference Proceeding
The importance of stratigraphic plays in the undiscovered resources of the UK Continental Shelf
Stoker, S. J., Gray, J. C., Haile, P., Andrews, I. J., Cameron, T. D. J.
Published in Deliberate Search for the Stratigraphic Trap (2006)
Published in Deliberate Search for the Stratigraphic Trap (2006)
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Book Chapter
Journal Article
Spontaneous pneumomediastinum presenting as jaw pain during labor
Raley, Janice C., Andrews, Janet I.
Published in Obstetrics and gynecology (New York. 1953) (01.11.2001)
Published in Obstetrics and gynecology (New York. 1953) (01.11.2001)
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Journal Article
Peptides Constrained by an Aliphatic Linkage between Two C α Sites: Design, Synthesis, and Unexpected Conformational Properties of an i,(i + 4)-Linked Peptide
Alexander McNamara, Linda M, Andrews, Martin J. I, Mitzel, Frieder, Siligardi, Giuliano, Tabor, Alethea B
Published in Journal of organic chemistry (29.06.2001)
Published in Journal of organic chemistry (29.06.2001)
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Journal Article
The remaining hydrocarbon potential of the UK Continental Shelf
MUNNS, J. W., GRAY, J. C., STOKER, S. J., ANDREWS, I. J., CAMERON, T. D. J.
Published in Petroleum Geology: North-West Europe and Global Perspectives ‒ Proceedings of the 6th Petroleum Geology Conference (01.01.2005)
Published in Petroleum Geology: North-West Europe and Global Perspectives ‒ Proceedings of the 6th Petroleum Geology Conference (01.01.2005)
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Conference Proceeding
Expediting drug discovery: recent advances in fast medicinal chemistry--optimization of hits and leads
Edwards, Paul J, Allart, Brigitte, Andrews, Martin J I, Clase, J Andrew, Menet, Christel
Published in Current opinion in drug discovery & development (01.07.2006)
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Published in Current opinion in drug discovery & development (01.07.2006)
Journal Article
Insights into Cyclin Groove Recognition: Complex Crystal Structures and Inhibitor Design through Ligand Exchange
Kontopidis, George, Andrews, Martin J.I., McInnes, Campbell, Cowan, Angela, Powers, Helen, Innes, Lorraine, Plater, Andy, Griffiths, Gary, Paterson, Dougie, Zheleva, Daniella I., Lane, David P., Green, Stephen, Walkinshaw, Malcolm D., Fischer, Peter M.
Published in Structure (London) (01.12.2003)
Published in Structure (London) (01.12.2003)
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Journal Article
Molecular Epidemiology of Macrolide Resistance in Neonatal Bloodstream Isolates of Group B Streptococci
DIEKEMA, Daniel J, ANDREWS, Janet I, HUYNH, Holly, RHOMBERG, Paul R, DOKTOR, Stella R, BEYER, Jill, RIDGE, Virginia D, FLAMM, Robert K, JONES, Ronald N, PFALLER, Michael A
Published in Journal of Clinical Microbiology (01.06.2003)
Published in Journal of Clinical Microbiology (01.06.2003)
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Journal Article