Magnesium Chelating 2-Hydroxyisoquinoline-1,3(2H,4H)-diones, as Inhibitors of HIV-1 Integrase and/or the HIV-1 Reverse Transcriptase Ribonuclease H Domain: Discovery of a Novel Selective Inhibitor of the Ribonuclease H Function
Billamboz, Muriel, Bailly, Fabrice, Lion, Cédric, Touati, Nadia, Vezin, Hervé, Calmels, Christina, Andréola, Marie-Line, Christ, Frauke, Debyser, Zeger, Cotelle, Philippe
Published in Journal of medicinal chemistry (24.03.2011)
Published in Journal of medicinal chemistry (24.03.2011)
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Design, Synthesis, and Biological Evaluation of a Series of 2-Hydroxyisoquinoline-1,3(2H,4H)-diones as Dual Inhibitors of Human Immunodeficiency Virus Type 1 Integrase and the Reverse Transcriptase RNase H Domain
Billamboz, Muriel, Bailly, Fabrice, Barreca, Maria Letizia, De Luca, Laura, Mouscadet, Jean-François, Calmels, Christina, Andréola, Marie-Line, Witvrouw, Myriam, Christ, Frauke, Debyser, Zeger, Cotelle, Philippe
Published in Journal of medicinal chemistry (25.12.2008)
Published in Journal of medicinal chemistry (25.12.2008)
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4‑Substituted 2‑Hydroxyisoquinoline-1,3(2H,4H)‑diones as a Novel Class of HIV‑1 Integrase Inhibitors
Billamboz, Muriel, Suchaud, Virginie, Bailly, Fabrice, Lion, Cedric, Demeulemeester, Jonas, Calmels, Christina, Andréola, Marie-Line, Christ, Frauke, Debyser, Zeger, Cotelle, Philippe
Published in ACS medicinal chemistry letters (11.07.2013)
Published in ACS medicinal chemistry letters (11.07.2013)
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Journal Article
An Interlocked Dimeric Parallel-Stranded DNA Quadruplex: A Potent Inhibitor of HIV-1 Integrase
Phan, Anh Tuân, Kuryavyi, Vitaly, Ma, Jin-Biao, Faure, Aurélie, Andréola, Marie-Line, Patel, Dinshaw J., Doudna, Jennifer A.
Published in Proceedings of the National Academy of Sciences - PNAS (18.01.2005)
Published in Proceedings of the National Academy of Sciences - PNAS (18.01.2005)
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Journal Article
2-Hydroxyisoquinoline-1,3(2 H,4 H)-diones as inhibitors of HIV-1 integrase and reverse transcriptase RNase H domain: Influence of the alkylation of position 4
Billamboz, Muriel, Bailly, Fabrice, Lion, Cédric, Calmels, Christina, Andréola, Marie-Line, Witvrouw, Myriam, Christ, Frauke, Debyser, Zeger, De Luca, Laura, Chimirri, Alba, Cotelle, Philippe
Published in European journal of medicinal chemistry (01.02.2011)
Published in European journal of medicinal chemistry (01.02.2011)
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Exploring the impact of the side-chain length on peptide/RNA binding events
Sbicca, Lola, González, Alejandro López, Gresika, Alexandra, Di Giorgio, Audrey, Closa, Jordi Teixido, Tejedor, Roger Estrada, Andréola, Marie-Line, Azoulay, Stéphane, Patino, Nadia
Published in Physical chemistry chemical physics : PCCP (19.07.2017)
Published in Physical chemistry chemical physics : PCCP (19.07.2017)
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Activation of GCN2 upon HIV-1 infection and inhibition of translation
Cosnefroy, Ophélie, Jaspart, Anaïs, Calmels, Christina, Parissi, Vincent, Fleury, Hervé, Ventura, Michel, Reigadas, Sandrine, Andréola, Marie-Line
Published in Cellular and molecular life sciences : CMLS (01.07.2013)
Published in Cellular and molecular life sciences : CMLS (01.07.2013)
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Evaluation of selected South African medicinal plants for inhibitory properties against human immunodeficiency virus type 1 reverse transcriptase and integrase
Bessong, Pascal Obong, Obi, Chikwelu Larry, Andréola, Marie-Line, Rojas, Luis B., Pouységu, Laurent, Igumbor, Eunice, Meyer, J.J. Marion, Quideau, Stéphane, Litvak, Simon
Published in Journal of ethnopharmacology (13.05.2005)
Published in Journal of ethnopharmacology (13.05.2005)
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Journal Article
Evolution of 2-long terminal repeat (2-LTR) episomal HIV-1 DNA in raltegravir-treated patients and in in vitro infected cells
Reigadas, Sandrine, Andréola, Marie-Line, Wittkop, Linda, Cosnefroy, Ophélie, Anies, Guerric, Recordon-Pinson, Patricia, Thiébaut, Rodolphe, Masquelier, Bernard, Fleury, Hervé
Published in Journal of antimicrobial chemotherapy (01.03.2010)
Published in Journal of antimicrobial chemotherapy (01.03.2010)
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RNA synthesis is modulated by G-quadruplex formation in Hepatitis C virus negative RNA strand
Jaubert, Chloé, Bedrat, Amina, Bartolucci, Laura, Di Primo, Carmelo, Ventura, Michel, Mergny, Jean-Louis, Amrane, Samir, Andreola, Marie-Line
Published in Scientific reports (25.05.2018)
Published in Scientific reports (25.05.2018)
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Journal Article
Structure of a DNA G-quadruplex that Modulates SP1 Binding Sites Architecture in HIV-1 Promoter
De Rache, Aurore, Marquevielle, Julien, Bouaziz, Serge, Vialet, Brune, Andreola, Marie-Line, Mergny, Jean-Louis, Amrane, Samir
Published in Journal of molecular biology (15.01.2024)
Published in Journal of molecular biology (15.01.2024)
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Journal Article
Targeting HIV-1 integrase with aptamers selected against the purified RNase H domain of HIV-1 RT
Métifiot, Mathieu, Leon, Oscar, Tarrago-Litvak, Laura, Litvak, Simon, Andréola, Marie-Line
Published in Biochimie (01.09.2005)
Published in Biochimie (01.09.2005)
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Journal Article
Investigation of a Novel Series of 2‑Hydroxyisoquinoline-1,3(2H,4H)‑diones as Human Immunodeficiency Virus Type 1 Integrase Inhibitors
Suchaud, Virginie, Bailly, Fabrice, Lion, Cedric, Calmels, Christina, Andréola, Marie-Line, Christ, Frauke, Debyser, Zeger, Cotelle, Philippe
Published in Journal of medicinal chemistry (12.06.2014)
Published in Journal of medicinal chemistry (12.06.2014)
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2-hydroxyisoquinoline-1,3(2H,4H)-diones (HIDs) as human immunodeficiency virus type 1 integrase inhibitors: Influence of the alkylcarboxamide substitution of position 4
Billamboz, Muriel, Suchaud, Virginie, Bailly, Fabrice, Lion, Cedric, Andréola, Marie-Line, Christ, Frauke, Debyser, Zeger, Cotelle, Philippe
Published in European journal of medicinal chemistry (19.07.2016)
Published in European journal of medicinal chemistry (19.07.2016)
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Journal Article
De novo RNA synthesis catalyzed by the Zika Virus RNA polymerase domain
Calmels, Christina, Ventura, Michel, Aknin, Cindy, Métifiot, Mathieu, Andreola, Marie-Line
Published in Scientific reports (02.06.2017)
Published in Scientific reports (02.06.2017)
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Modulation of chromatin structure by the FACT histone chaperone complex regulates HIV-1 integration
Matysiak, Julien, Lesbats, Paul, Mauro, Eric, Lapaillerie, Delphine, Dupuy, Jean-William, Lopez, Angelica P, Benleulmi, Mohamed Salah, Calmels, Christina, Andreola, Marie-Line, Ruff, Marc, Llano, Manuel, Delelis, Olivier, Lavigne, Marc, Parissi, Vincent
Published in Retrovirology (28.07.2017)
Published in Retrovirology (28.07.2017)
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Journal Article
Intasome architecture and chromatin density modulate retroviral integration into nucleosome
Benleulmi, Mohamed Salah, Matysiak, Julien, Henriquez, Daniel Rodrigo, Vaillant, Cédric, Lesbats, Paul, Calmels, Christina, Naughtin, Monica, Leon, Oscar, Skalka, Anna Marie, Ruff, Marc, Lavigne, Marc, Andreola, Marie-Line, Parissi, Vincent
Published in Retrovirology (07.02.2015)
Published in Retrovirology (07.02.2015)
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