Search Results - "Andis, Sherri L." :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Synthesis, Pharmacological Characterization, and Molecular Modeling of Heterobicyclic Amino Acids Related to (+)-2-Aminobicyclo[3.1.0]hexane- 2,6-dicarboxylic Acid (LY354740): Identification of Two New Potent, Selective, and Systemically Active Agonists for Group II Metabotropic Glutamate Receptors

Synthesis, Pharmacological Characterization, and Molecular Modeling of Heterobicyclic Amino Acids Related to (+)-2-Aminobicyclo[3.1.0]hexane- 2,6-dicarboxylic Acid (LY354740): Identification of Two New Potent, Selective, and Systemically Active Agonists for Group II Metabotropic Glutamate Receptors

by Monn, James A, Valli, Matthew J, Massey, Steven M, Hansen, Marvin M, Kress, Thomas J, Wepsiec, James P, Harkness, Allen R, Grutsch, John L, Wright, Rebecca A, Johnson, Bryan G, Andis, Sherri L, Kingston, Ann, Tomlinson, Rosemarie, Lewis, Richard, Griffey, Kelly R, Tizzano, Joseph P, Schoepp, Darryle D
Published in Journal of medicinal chemistry (25.03.1999)

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Synthesis and Metabotropic Glutamate Receptor Activity of S-Oxidized Variants of (−)-4-Amino-2-thiabicyclo-[3.1.0]hexane-4,6-dicarboxylate: Identification of Potent, Selective, and Orally Bioavailable Agonists for mGlu2/3 Receptors

Synthesis and Metabotropic Glutamate Receptor Activity of S-Oxidized Variants of (−)-4-Amino-2-thiabicyclo-[3.1.0]hexane-4,6-dicarboxylate: Identification of Potent, Selective, and Orally Bioavailable Agonists for mGlu2/3 Receptors

by Monn, James A., Massey, Steven M., Valli, Matthew J., Henry, Steven S., Stephenson, Gregory A., Bures, Mark, Hérin, Marc, Catlow, John, Giera, Deborah, Wright, Rebecca A., Johnson, Bryan G., Andis, Sherri L., Kingston, Ann, Schoepp, Darryle D.
Published in Journal of medicinal chemistry (25.01.2007)

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LY231514, a pyrrolo[2,3-d]pyrimidine-based antifolate that inhibits multiple folate-requiring enzymes

LY231514, a pyrrolo[2,3-d]pyrimidine-based antifolate that inhibits multiple folate-requiring enzymes

by SHIH, C, CHEN, V. J, ANDIS, S. L, BEWLEY, J. R, RAYL, E. A, MOROSON, B. A, BEARDSLEY, G. P, KOHLER, W, RATNAM, M, SCHULTZ, R. M, GOSSETT, L. S, GATES, S. B, MACKELLAR, W. C, HABECK, L. L, SHACKELFORD, K. A, MENDELSOHN, L. G, SOOSE, D. J, PATEL, V. F
Published in Cancer research (Chicago, Ill.) (15.03.1997)

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Methyl Substitution of 2-Aminobicyclo[3.1.0]hexane 2,6-Dicarboxylate (LY354740) Determines Functional Activity at Metabotropic Glutamate Receptors: Identification of a Subtype Selective mGlu2 Receptor Agonist

Methyl Substitution of 2-Aminobicyclo[3.1.0]hexane 2,6-Dicarboxylate (LY354740) Determines Functional Activity at Metabotropic Glutamate Receptors: Identification of a Subtype Selective mGlu2 Receptor Agonist

by Dominguez, Carmen, Prieto, Lourdes, Valli, Matthew J, Massey, Steven M, Bures, Mark, Wright, Rebecca A, Johnson, Bryan G, Andis, Sherri L, Kingston, Ann, Schoepp, Darryle D, Monn, James A
Published in Journal of medicinal chemistry (19.05.2005)

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SAR study of a subtype selective allosteric potentiator of metabotropic glutamate 2 receptor, N-(4-phenoxyphenyl)- N-(3-pyridinylmethyl)ethanesulfonamide

SAR study of a subtype selective allosteric potentiator of metabotropic glutamate 2 receptor, N-(4-phenoxyphenyl)- N-(3-pyridinylmethyl)ethanesulfonamide

by Barda, David A., Wang, Zhao-Qing, Britton, Thomas C., Henry, Steven S., Jagdmann, G.Erik, Coleman, Darrell S., Johnson, Michael P., Andis, Sherri L., Schoepp, Darryle D.
Published in Bioorganic & medicinal chemistry letters (21.06.2004)

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A Convergent Approach to Cryptophycin 52 Analogues: Synthesis and Biological Evaluation of a Novel Series of Fragment A Epoxides and Chlorohydrins

A Convergent Approach to Cryptophycin 52 Analogues: Synthesis and Biological Evaluation of a Novel Series of Fragment A Epoxides and Chlorohydrins

by Al-awar, Rima S, Ray, James E, Schultz, Richard M, Andis, Sherri L, Kennedy, Joseph H, Moore, Richard E, Liang, Jian, Golakoti, Trimurtulu, Subbaraju, Gottumukkala V, Corbett, Thomas H
Published in Journal of medicinal chemistry (03.07.2003)

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C3′- cis-Substituted carboxycyclopropyl glycines as metabotropic glutamate 2/3 receptor agonists: Synthesis and SAR studies

C3′- cis-Substituted carboxycyclopropyl glycines as metabotropic glutamate 2/3 receptor agonists: Synthesis and SAR studies

by González, Rosario, Collado, Iván, López de Uralde, Beatriz, Marcos, Alicia, Martín-Cabrejas, Luisa M., Pedregal, Concepción, Blanco-Urgoiti, Jaime, Pérez-Castells, Javier, Alejandro Fernández, M., Andis, Sherri L., Johnson, Bryan G., Wright, Rebecca A., Schoepp, Darryle D., Monn, James A.
Published in Bioorganic & medicinal chemistry (01.12.2005)

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Total Synthesis of Cryptophycin Analogues. Isosteric Replacement of the C−D Ester

Total Synthesis of Cryptophycin Analogues. Isosteric Replacement of the C−D Ester

by Norman, Bryan H, Hemscheidt, Thomas, Schultz, Richard M, Andis, Sherri L
Published in Journal of organic chemistry (24.07.1998)

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Novel Cryptophycin Antitumor Agents: Synthesis and Cytotoxicity of Fragment “B” Analogues

Novel Cryptophycin Antitumor Agents: Synthesis and Cytotoxicity of Fragment “B” Analogues

by Patel, Vinod F, Andis, Sherri L, Kennedy, Joseph H, Ray, James E, Schultz, Richard M
Published in Journal of medicinal chemistry (15.07.1999)

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Total Synthesis of Seco (+)- and ent-(−)-Oxaduocarmycin SA: Construction of the (Chloromethyl)indoline Alkylating Subunit by a Novel Intramolecular Aryl Radical Cyclization onto a Vinyl Chloride

Total Synthesis of Seco (+)- and ent-(−)-Oxaduocarmycin SA: Construction of the (Chloromethyl)indoline Alkylating Subunit by a Novel Intramolecular Aryl Radical Cyclization onto a Vinyl Chloride

by Patel, Vinod F, Andis, Sherri L, Enkema, Julia K, Johnson, David A, Kennedy, Joseph H, Mohamadi, Fariborz, Schultz, Richard M, Soose, Daniel J, Spees, Michael M
Published in Journal of organic chemistry (12.12.1997)

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A novel class of monoglutamated antifolates exhibits tight-binding inhibition of human glycinamide ribonucleotide formyltransferase and potent activity against solid tumors

A novel class of monoglutamated antifolates exhibits tight-binding inhibition of human glycinamide ribonucleotide formyltransferase and potent activity against solid tumors

by Habeck, L L, Leitner, T A, Shackelford, K A, Gossett, L S, Schultz, R M, Andis, S L, Shih, C, Grindey, G B, Mendelsohn, L G
Published in Cancer research (Chicago, Ill.) (15.02.1994)

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Synthesis and biological evaluation of novel cryptophycin analogs with modification in the β-alanine region

Synthesis and biological evaluation of novel cryptophycin analogs with modification in the β-alanine region

by Shih, Chuan, Gossett, Lynn S., Gruber, Joseph M., Grossman, C.Sue, Andis, Sherri L., Schultz, Richard M., Worzalla, John F., Corbett, Tom H., Metz, James T.
Published in Bioorganic & medicinal chemistry letters (04.01.1999)

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Cell cycle effects of antifolate antimetabolites : implications for cytotoxicity and cytostasis

Cell cycle effects of antifolate antimetabolites : implications for cytotoxicity and cytostasis

by TONKINSON, J. L, MARDER, P, ANDIS, S. L, SCHULTZ, R. M, GOSSETT, L. S, SHIH, C, MENDELSOHN, L. G
Published in Cancer chemotherapy and pharmacology (1997)

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Substrate specificity of mammalian folylpolyglutamate synthetase for 5,10-dideazatetrahydrofolate analogs

Substrate specificity of mammalian folylpolyglutamate synthetase for 5,10-dideazatetrahydrofolate analogs

by Habeck, L L, Mendelsohn, L G, Shih, C, Taylor, E C, Colman, P D, Gossett, L S, Leitner, T A, Schultz, R M, Andis, S L, Moran, R G
Published in Molecular pharmacology (01.08.1995)

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Synthesis and biological evaluation of cryptophycin analogs with substitution at C-6 (fragment C region)

Synthesis and biological evaluation of cryptophycin analogs with substitution at C-6 (fragment C region)

by Varie, David L., Shih, Chuan, Hay, David A., Andis, Sherri L., Corbett, Tom H., Gossett, Lynn S., Janisse, Samantha K., Martinelli, Michael J., Moher, Eric D., Schultz, Richard M., Toth, John E.
Published in Bioorganic & medicinal chemistry letters (08.02.1999)

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The synthesis and biological activity of a series of 2,4-diaminopyrido[2,3- D]pyrimidine based antifolates as antineoplastic and antiarthritic agents

The synthesis and biological activity of a series of 2,4-diaminopyrido[2,3- D]pyrimidine based antifolates as antineoplastic and antiarthritic agents

by Gossett, Lynn S., Habeck, Lillian L., Shackelford, Katherine A., Mendelsohn, Laurane G., Gates, Susan B., Worzalla, John F., Self, Tracy D., Theobald, Karla S., Andis, Sherri L., Schultz, Richard M., Shih, Chuan
Published in Bioorganic & medicinal chemistry letters (04.01.1999)

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Synthesis and biological evaluation of a new series of dihydrofolate reductase inhibitors based on the 4-(2,6-diamino-5-pyrimidinyl)alkyl-L-glutamic acid structure

Synthesis and biological evaluation of a new series of dihydrofolate reductase inhibitors based on the 4-(2,6-diamino-5-pyrimidinyl)alkyl-L-glutamic acid structure

by Gossett, Lynn S., Habeck, Lillian L., Gates, Susan B., Andis, Sherri L., Worzalla, John F., Schultz, Richard M., Mendelsonn, Laurane G., Kohler, William, Ratnam, Manohar, Grindey, Gerald B., Shih, Chuan
Published in Bioorganic & medicinal chemistry letters (20.02.1996)

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Evaluation of new anticancer agents against the MIA PaCa-2 and PANC-1 human pancreatic carcinoma xenografts

Evaluation of new anticancer agents against the MIA PaCa-2 and PANC-1 human pancreatic carcinoma xenografts

by Schultz, R M, Merriman, R L, Toth, J E, Zimmermann, J E, Hertel, L W, Andis, S L, Dudley, D E, Rutherford, P G, Tanzer, L R, Grindey, G B
Published in Oncology research (1993)

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Role of membrane-associated folate binding protein in the cytotoxicity of antifolates in KB, IGROV1, and L1210A cells

Role of membrane-associated folate binding protein in the cytotoxicity of antifolates in KB, IGROV1, and L1210A cells

by Schultz, R M, Andis, S L, Shackelford, K A, Gates, S B, Ratnam, M, Mendelsohn, L G, Shih, C, Grindey, G B
Published in Oncology research (1995)

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SAR Study of a Subtype Selective Allosteric Potentiator of Metabotropic Glutamate 2 Receptor, N-(4-Phenoxyphenyl)-N-(3-pyridinylmethyl)ethanesulfonamide

SAR Study of a Subtype Selective Allosteric Potentiator of Metabotropic Glutamate 2 Receptor, N-(4-Phenoxyphenyl)-N-(3-pyridinylmethyl)ethanesulfonamide

by Barda, David A., Wang, Zhao-Qing, Britton, Thomas C., Henry, Steven S., Jagdmann, G. Erik, Coleman, Darrell S., Johnson, Michael P., Andis, Sherri L., Schoepp, Darryle D.
Published in ChemInform (28.09.2004)

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