439 Comparison of Dielectrophoretic Field Flow Fractionation (DEP-FFF) with ApoStream™, an Antibody Independent Platform, with Immunomagnetic Capture Using CellSearch™ for Enumeration of Circulating Tumor Cells in Patients with Metastatic Prostate Cancer
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Published in European journal of cancer (1990) (01.11.2012)
Published in European journal of cancer (1990) (01.11.2012)
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214 Androgen Receptor Expression in in Circulating Tumor Cells, Archival and Metastatic Tissue in Prostate Cancer Patients
Anderes, K, Melnikova, V, Pace, M, Sukumaran, S, Garza, M, Redden, B, Woo, J, Davis, D, Amato, R
Published in European journal of cancer (1990) (01.11.2012)
Published in European journal of cancer (1990) (01.11.2012)
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215 Circulating Tumor Cells as Surrogate Biomarkers of Epithelial Mesenchymal Transition and Metastatic Phenotype in Prostate Cancer Patients
Amato, R, Melnikova, V, Pace, M, Sukumaran, S, Garza, M, Redden, B, Woo, J, Anderes, K, Davis, D
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Published in European journal of cancer (1990) (01.11.2012)
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414 Clinical pharmacokinetics and pharmacodynamics of CX-4945, a novel inhibitor of protein kinase CK2: Interim report from the phase 1 clinical trial
Padgett, C.S, Lim, J.K.C, Marschke, R.F, Northfelt, D.W, Andreopoulou, E, Hoff, D.D. Von, Anderes, K, Ryckman, D.M, Chen, T.K, O'Brien, S.E
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Published in European journal of cancer supplements (01.11.2010)
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Identification of Alkylidene Hydrazides as Glucagon Receptor Antagonists
Ling, Anthony, Hong, Yufeng, Gonzalez, Javier, Gregor, Vlad, Polinsky, Alex, Kuki, Atsuo, Shi, Shenghua, Teston, Kimberly, Murphy, Douglas, Porter, John, Kiel, Dan, Lakis, James, Anderes, Kenna, May, John, Knudsen, Lotte Bjerre, Lau, Jesper
Published in Journal of medicinal chemistry (13.09.2001)
Published in Journal of medicinal chemistry (13.09.2001)
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633 The contribution of dysregulated ribosomal gene transcription to malignant transformation
Hannan, R.D, Bywater, M.J, Poortinga, G, Cullinane, C, Stanley, K, Walker, R, Drygin, D, Anderes, K, Pearson, R, McArthur, G.A
Published in European journal of cancer supplements (2010)
Published in European journal of cancer supplements (2010)
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518 CX-4945, an inhibitor of protein kinase CK2, disrupts DNA damage repair, potentiates apoptosis and enhances antitumor activity of gemcitabine in a model of ovarian cancer
Anderes, K, Bliesath, J, Ho, C, Omori, M, Huser, N, Siddiqui-Jain, A, Streiner, N, Proffitt, C, O'Brien, S, Drygin, D
Published in European journal of cancer supplements (2010)
Published in European journal of cancer supplements (2010)
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99 Combined inhibition of EGFR and protein kinase CK2 synergistically blocks phosphorylation of ribosomal protein S6, induces apoptosis in cancer cells and displays enhanced antitumor activity in xenograft models
Drygin, D, Bliesath, J, Siddiqui-Jain, A, Huser, N, Omori, M, Streiner, N, Proffitt, C, Ho, C, O'Brien, S, Anderes, K
Published in European journal of cancer supplements (2010)
Published in European journal of cancer supplements (2010)
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549O Adagrasib with or without cetuximab in patients with KRASG12C-mutated colorectal cancer (CRC): Analysis of tumor biomarkers and genomic alterations
Pelster, M.S., Yaeger, R., Klempner, S.J., Ou, S-H.I., Spira, A.I., Jänne, P.A., Uboha, N.V., Gaffar, Y.A., Newman, G., Paweletz, C.P., Heavey, G.A., Alejandro, L., Kheoh, T., Anderes, K., Der Torossian, H., Christensen, J.G., Weiss, J.
Published in Annals of oncology (01.10.2023)
Published in Annals of oncology (01.10.2023)
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526P Pharmacodynamic evidence for WEE1 target engagement in surrogate and tumor tissues from a phase I study of the WEE1 inhibitor ZN-c3
Chalasani, P., Tolcher, A., Meric-Bernstam, F., Mamdani, H., de Jong, P.R., Anderes, K., Samatar, A.A., Sergeeva, M., Gazdoiu, M., Viana, M.R., Pultar, P., Voliotis, D., Donate, F.
Published in Annals of oncology (01.09.2021)
Published in Annals of oncology (01.09.2021)
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8MO Adagrasib (MRTX849) in patients with advanced/metastatic KRAS G12C-mutated non-small cell lung cancer (NSCLC): Preliminary analysis of mutation allele frequency
Jänne, P.A., Spira, A., Riely, G.J., Gadgeel, S., Heist, R., Ou, S-H.I., Johnson, M.L., Sabari, J., Velastegui, K., Christensen, J.G., Yang, W., Anderes, K., Chao, R., Paweletz, C.
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Published in Journal of thoracic oncology (01.04.2023)
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Effect of testosterone suppression on the pharmacokinetics of a potent GnRH receptor antagonist
IATSIMIRSKAIA, Eugenia A, GREGORY, Margaret L, MAY, John M, ANDERES, Kenna L, CASTILLO, Rosemary, MILGRAM, K. Eric, LUTHIN, David R, PATHAK, Ved P, CHRISTIE, Lance C, VAZIR, Haresh, ANDERSON, Mark B
Published in Pharmaceutical research (01.02.2002)
Published in Pharmaceutical research (01.02.2002)
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Effect of CX-4945, a selective bioavailable small molecule inhibitor of protein kinase CK2, on gemcitabine antitumor activity in A2780 ovarian cancer
Anderes, K. L., Streiner, N., Omori, M., Huser, N., Ho, C., Siddiqui-Jain, A., Bliesath, J., O'Brien, S., Drygin, D., Rice, W. G.
Published in Journal of clinical oncology (20.05.2010)
Published in Journal of clinical oncology (20.05.2010)
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Optimization of Alkylidene Hydrazide Based Human Glucagon Receptor Antagonists. Discovery of the Highly Potent and Orally Available 3-Cyano-4-hydroxybenzoic Acid [1-(2,3,5,6-Tetramethylbenzyl)-1H-indol-4-ylmethylene]hydrazide
Madsen, Peter, Ling, Anthony, Plewe, Michael, Sams, Christian K, Knudsen, Lotte B, Sidelmann, Ulla G, Ynddal, Lars, Brand, Christian L, Andersen, Birgitte, Murphy, Douglas, Teng, Min, Truesdale, Larry, Kiel, Dan, May, John, Kuki, Atsuo, Shi, Shenghua, Johnson, Michael D, Teston, Kimberly Ann, Feng, Jun, Lakis, James, Anderes, Kenna, Gregor, Vlad, Lau, Jesper
Published in Journal of medicinal chemistry (19.12.2002)
Published in Journal of medicinal chemistry (19.12.2002)
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Positron-emission tomography reveals early flare in uptake of FLT in tumors following chemotherapy with gemcitabine
McArthur, G. A., Hicks, R. M., Shalinsky, D. R., Binns, D., O’Kane, C., Hogg, A., Fisher, R., McCarthy, T. J., Anderes, K. A.
Published in Journal of clinical oncology (20.06.2007)
Published in Journal of clinical oncology (20.06.2007)
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Imaging with FLT-PET demonstrates that PF-477736, an inhibitor of CHK1 kinase, overcomes a cell cycle checkpoint induced by gemcitabine in PC-3 xenografts
McArthur, G. A., Raleigh, J., Blasina, A., Cullinane, C., Dorow, D., Conus, N., Hicks, R. J., Kornmann, J., Chen, E., McCarthy, T. J., Anderes, K.
Published in Journal of clinical oncology (20.06.2006)
Published in Journal of clinical oncology (20.06.2006)
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Human glucagon receptor antagonists based on alkylidene hydrazides
Ling, Anthony, Plewe, Michael, Gonzalez, Javier, Madsen, Peter, Sams, Christian K., Lau, Jesper, Gregor, Vlad, Murphy, Doug, Teston, Kimberly, Kuki, Atsuo, Shi, Shenghua, Truesdale, Larry, Kiel, Dan, May, John, Lakis, James, Anderes, Kenna, Iatsimirskaia, Eugenia, Sidelmann, Ulla G., Knudsen, Lotte B., Brand, Christian L., Polinsky, Alex
Published in Bioorganic & medicinal chemistry letters (25.02.2002)
Published in Bioorganic & medicinal chemistry letters (25.02.2002)
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