The discovery of quinoline based single-ligand human H-1 and H-3 receptor antagonists
Procopiou, Panayiotis A., Ancliff, Rachael A., Gore, Paul M., Hancock, Ashley P., Hodgson, Simon T., Holmes, Duncan S., Keeling, Steven P., Looker, Brian E., Parr, Nigel A., Rowedder, James E., Slack, Robert J.
Published in Bioorganic & medicinal chemistry letters (15.12.2016)
Published in Bioorganic & medicinal chemistry letters (15.12.2016)
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Journal Article
The discovery of quinoline based single-ligand human H1 and H3 receptor antagonists
Procopiou, Panayiotis A., Ancliff, Rachael A., Gore, Paul M., Hancock, Ashley P., Hodgson, Simon T., Holmes, Duncan S., Keeling, Steven P., Looker, Brian E., Parr, Nigel A., Rowedder, James E., Slack, Robert J.
Published in Bioorganic & medicinal chemistry letters (15.12.2016)
Published in Bioorganic & medicinal chemistry letters (15.12.2016)
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4-Acyl-1-(4-aminoalkoxyphenyl)-2-ketopiperazines as a Novel Class of Non-Brain-Penetrant Histamine H3 Receptor Antagonists
Procopiou, Panayiotis A, Ancliff, Rachael A, Bamford, Mark J, Browning, Christopher, Connor, Helen, Davies, Susannah, Fogden, Yvonne C, Hodgson, Simon T, Holmes, Duncan S, Looker, Brian E, Morriss, Karen M. L, Parr, Christopher A, Pickup, Elizabeth A, Sehmi, Sanjeet S, White, Gemma V, Watts, Clarissa J, Wilson, David M, Woodrow, Michael D
Published in Journal of medicinal chemistry (27.12.2007)
Published in Journal of medicinal chemistry (27.12.2007)
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Journal Article
4-acyl-1-(4-aminoalkoxyphenyl)-2-ketopiperazines as a novel class of non-brain-penetrant histamine H-3 receptor antagonists
Procopiou, Panayiotis A., Ancliff, Rachael A., Bamford, Mark J., Browning, Christopher, Connor, Helen, Davies, Susannah, Fogden, Yvonne C., Hodgson, Simon T., Holmes, Duncan S., Looker, Brian E., Morriss, Karen M. L., Parr, Christopher A., Pickup, Elizabeth A., Sehmi, Sanjeet S., White, Gemma V., Watts, Clarissa J., Wilson, David M., Woodrow, Michael D.
Published in Journal of medicinal chemistry (27.12.2007)
Published in Journal of medicinal chemistry (27.12.2007)
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Resolution of a citric acid derivative: synthesis of ( R)-(−)-homocitric acid-γ-lactone
Ancliff, Rachael A., Russell, Andrew T., Sanderson, Adam J.
Published in Tetrahedron: asymmetry (23.10.1997)
Published in Tetrahedron: asymmetry (23.10.1997)
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Morpholin-acetamide derivatives for the treatment of inflammatory diseases
HODGSON SIMON T, COOK CAROLINE M, ELDRED COLIN D, JUDD DUNCAN B, ROBERTSON GRAEME M, ANCLIFF RACHAEL A, LEWELL XIAO Q, GORE PAUL M, KEELING SUZANNE E, HARRISON LEE A, SWANSON STEPHEN
Year of Publication 13.04.2006
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Year of Publication 13.04.2006
Patent
Novel compounds
HODGSON SIMON T, MILLS GAIL, ANCLIFF RACHAEL A, HARRISON LEE A, COOK CAROLINE M, ELDRED COLIN D, JUDD DUNCAN B, LEWELL XIAO O, ROBERTSON GRAEME M, GORE PAUL M, KEELING SUZANNE E, WILKINSON MARK, WALKER ANDREW J, HAYES MARTIN A, SWANSON STEPHEN
Year of Publication 23.03.2006
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Year of Publication 23.03.2006
Patent
N-2s-4-3,4-difluorobenzyl morpholin-2yl methyl -2-(3-methylsulphonyl amino!phenyl acetamide as ccr3 antagonist for the treatment of inflammatory conditions
HODGSON SIMON T, MILLS GAIL, ANCLIFF RACHAEL A, LEWELL XIAO Q, HARRISON LEE A, COOK CAROLINE M, ELDRED COLIN D, JUDD DUNCAN B, ROBERTSON GRAEME M, GORE PAUL M, KEELING SUZANNE E, WILKINSON MARK, WALKER ANDREW J, HAYES MARTIN A, SWANSON STEPHEN
Year of Publication 16.03.2006
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Year of Publication 16.03.2006
Patent
Novel compounds
DUNCAN BRUCE JUDD, GORE, PAUL MARTIN, SIMON TEANBY HODGSON, GAIL MILLS, ELDRED, COLIN DAVID, HARRISON, LEE ANDREW, ANCLIFF, RACHAEL ANN, COOK, CAROLINE MARY, XIAO QING LEWELL, MARK WILKINSON, STEPHEN SWANSON, MARTIN ALISTAIR HAYES, GRAEME MICHAEL ROBERTSON, ANDREW JOHN WALKER, SUZANNE ELAINE KEELING
Year of Publication 16.03.2004
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Year of Publication 16.03.2004
Patent
Novel compounds
DUNCAN BRUCE JUDD, GORE, PAUL MARTIN, SIMON TEANBY HODGSON, GAIL MILLS, ELDRED, COLIN DAVID, HARRISON, LEE ANDREW, ANCLIFF, RACHAEL ANN, COOK, CAROLINE MARY, XIAO QING LEWELL, MARK WILKINSON, STEPHEN SWANSON, MARTIN ALISTAIR HAYES, GRAEME MICHAEL ROBERTSON, ANDREW JOHN WALKER, SUZANNE ELAINE KEELING
Year of Publication 01.03.2004
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Year of Publication 01.03.2004
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Novel compounds
DUNCAN BRUCE JUDD, GORE, PAUL MARTIN, SIMON TEANBY HODGSON, GAIL MILLS, ELDRED, COLIN DAVID, HARRISON, LEE ANDREW, ANCLIFF, RACHAEL ANN, COOK, CAROLINE MARY, XIAO QING LEWELL, MARK WILKINSON, STEPHEN SWANSON, MARTIN ALISTAIR HAYES, GRAEME MICHAEL ROBERTSON, ANDREW JOHN WALKER, SUZANNE ELAINE KEELING
Year of Publication 01.03.2004
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Year of Publication 01.03.2004
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Novel compounds
DUNCAN BRUCE JUDD, GORE, PAUL MARTIN, PAUL MARTIN GORE, SIMON TEANBY HODGSON, ELDRED, COLIN DAVID, HARRISON, LEE ANDREW, ANCLIFF, RACHAEL ANN, COOK, CAROLINE MARY, MARK WILKINSON, STEPHEN SWANSON, MARTIN ALISTAIR HAYES, GRAEME MICHAEL ROBERTSON, ANDREW JOHN WALKER, SUZANNE ELAINE KEELING, LEE ANDREW HARRISON
Year of Publication 16.02.2004
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Year of Publication 16.02.2004
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Novel compound
DUNCAN BRUCE JUDD, GORE, PAUL MARTIN, SIMON TEANBY HODGSON, GAIL MILLS, ELDRED, COLIN DAVID, HARRISON, LEE ANDREW, ANCLIFF, RACHAEL ANN, COOK, CAROLINE MARY, XIAO QING LEWELL, MARK WILKINSON, STEPHEN SWANSON, MARTIN ALISTAIR HAYES, GRAEME MICHAEL ROBERTSON, ANDREW JOHN WALKER, SUZANNE ELAINE KEELING
Year of Publication 01.02.2004
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Year of Publication 01.02.2004
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Novel compounds
DUNCAN BRUCE JUDD, GORE, PAUL MARTIN, SIMON TEANBY HODGSON, GAIL MILLS, ELDRED, COLIN DAVID, HARRISON, LEE ANDREW, ANCLIFF, RACHAEL ANN, COOK, CAROLINE MARY, XIAO QING LEWELL, MARK WILKINSON, STEPHEN SWANSON, MARTIN ALISTAIR HAYES, GRAEME MICHAEL ROBERTSON, ANDREW JOHN WALKER, SUZANNE ELAINE KEELING
Year of Publication 16.01.2004
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Year of Publication 16.01.2004
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Novel compounds
DUNCAN BRUCE JUDD, GORE, PAUL MARTIN, SIMON TEANBY HODGSON, GAIL MILLS, ELDRED, COLIN DAVID, HARRISON, LEE ANDREW, ANCLIFF, RACHAEL ANN, COOK, CAROLINE MARY, XIAO QING LEWELL, MARK WILKINSON, STEPHEN SWANSON, MARTIN ALISTAIR HAYES, GRAEME MICHAEL ROBERTSON, ANDREW JOHN WALKER, SUZANNE ELAINE KEELING
Year of Publication 16.01.2004
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Year of Publication 16.01.2004
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Novel compounds
DUNCAN BRUCE JUDD, GORE, PAUL MARTIN, SIMON TEANBY HODGSON, GAIL MILLS, ELDRED, COLIN DAVID, HARRISON, LEE ANDREW, ANCLIFF, RACHAEL ANN, COOK, CAROLINE MARY, XIAO QING LEWELL, MARK WILKINSON, STEPHEN SWANSON, MARTIN ALISTAIR HAYES, GRAEME MICHAEL ROBERTSON, ANDREW JOHN WALKER, SUZANNE ELAINE KEELING
Year of Publication 01.01.2004
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Year of Publication 01.01.2004
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