The discovery of quinoline based single-ligand human H-1 and H-3 receptor antagonists
Procopiou, Panayiotis A., Ancliff, Rachael A., Gore, Paul M., Hancock, Ashley P., Hodgson, Simon T., Holmes, Duncan S., Keeling, Steven P., Looker, Brian E., Parr, Nigel A., Rowedder, James E., Slack, Robert J.
Published in Bioorganic & medicinal chemistry letters (15.12.2016)
Published in Bioorganic & medicinal chemistry letters (15.12.2016)
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The discovery of quinoline based single-ligand human H1 and H3 receptor antagonists
Procopiou, Panayiotis A., Ancliff, Rachael A., Gore, Paul M., Hancock, Ashley P., Hodgson, Simon T., Holmes, Duncan S., Keeling, Steven P., Looker, Brian E., Parr, Nigel A., Rowedder, James E., Slack, Robert J.
Published in Bioorganic & medicinal chemistry letters (15.12.2016)
Published in Bioorganic & medicinal chemistry letters (15.12.2016)
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4-Acyl-1-(4-aminoalkoxyphenyl)-2-ketopiperazines as a Novel Class of Non-Brain-Penetrant Histamine H3 Receptor Antagonists
Procopiou, Panayiotis A, Ancliff, Rachael A, Bamford, Mark J, Browning, Christopher, Connor, Helen, Davies, Susannah, Fogden, Yvonne C, Hodgson, Simon T, Holmes, Duncan S, Looker, Brian E, Morriss, Karen M. L, Parr, Christopher A, Pickup, Elizabeth A, Sehmi, Sanjeet S, White, Gemma V, Watts, Clarissa J, Wilson, David M, Woodrow, Michael D
Published in Journal of medicinal chemistry (27.12.2007)
Published in Journal of medicinal chemistry (27.12.2007)
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4-acyl-1-(4-aminoalkoxyphenyl)-2-ketopiperazines as a novel class of non-brain-penetrant histamine H-3 receptor antagonists
Procopiou, Panayiotis A., Ancliff, Rachael A., Bamford, Mark J., Browning, Christopher, Connor, Helen, Davies, Susannah, Fogden, Yvonne C., Hodgson, Simon T., Holmes, Duncan S., Looker, Brian E., Morriss, Karen M. L., Parr, Christopher A., Pickup, Elizabeth A., Sehmi, Sanjeet S., White, Gemma V., Watts, Clarissa J., Wilson, David M., Woodrow, Michael D.
Published in Journal of medicinal chemistry (27.12.2007)
Published in Journal of medicinal chemistry (27.12.2007)
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Resolution of a citric acid derivative: synthesis of ( R)-(−)-homocitric acid-γ-lactone
Ancliff, Rachael A., Russell, Andrew T., Sanderson, Adam J.
Published in Tetrahedron: asymmetry (23.10.1997)
Published in Tetrahedron: asymmetry (23.10.1997)
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MORPHOLIN-ACETAMIDE DERIVATIVES FOR THE TREATMENT OF INFLAMMATORY DISEASES
COOK, CAROLINE MARY, HODGSON, SIMON TEANBY, LEWELL, XIAO QING, ROBERTSON, GRAEME MICHAEL, GORE, PAUL MARTIN, SWANSON, STEPHEN, KEELING, SUZANNE ELAINE, ANCLIFF, RACHAEL ANNE, JUDD, DUNCAN BRUCE, ELDRED, COLIN DAVID, HARRISON, LEE ANDREW
Year of Publication 29.10.2014
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Year of Publication 29.10.2014
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EINEN AZEPIN-KERN ENTHALTENDE ANTAGONISTEN DES HISTAMINREZEPTORS
ANCLIFF, RACHAEL ANN, HANCOCK, ASHLEY PAUL, KRANZ, MICHAEL JOACHIM, PARR, NIGEL
Year of Publication 15.01.2010
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Year of Publication 15.01.2010
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HISTAMINE RECEPTOR ANTAGONISTS COMPRISING AN AZEPIN CORE
ANCLIFF, RACHAEL ANN, PARR, NIGEL, JAMES, HANCOCK, ASHLEY PAUL, KRANZ, MICHAEL JOACHIM
Year of Publication 13.01.2010
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Year of Publication 13.01.2010
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VERBINDUNGEN
HODGSON, SIMON, PARR, CHRISTOPHER, BAMFORD, MARK, ANCLIFF, RACHAEL, PROCOPIOU, PANAYIOTIS, WILSON, DAVID, WOODROW, MICHAEL
Year of Publication 15.09.2009
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Year of Publication 15.09.2009
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A Catalytic Asymmetric Bioorganic Route to Enantioenriched Tetrahydro- and Dihydropyranones
Baker-Glenn, Charles, Hodnett, Neil, Reiter, Maud, Ropp, Sandrine, Ancliff, Rachael, Gouverneur, Veronique
Published in ChemInform (21.06.2005)
Published in ChemInform (21.06.2005)
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Histamine Receptor Antagonists Comprising an Azepin Core
KRANZ MICHAEL JOACHIM, PARR NIGEL JAMES, ANCLIFF RACHAEL ANN, HANCOCK ASHLEY PAUL
Year of Publication 16.07.2009
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Year of Publication 16.07.2009
Patent
Morpholin-acetamide derivatives for the treatment of inflammatory diseases
Ancliff, Rachael Anne, Hodgson, Simon Teanby, Lewell, Xiao Qing, Robertson, Graeme Michael
Year of Publication 14.07.2009
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Year of Publication 14.07.2009
Patent
Morpholin-acetamide derivatives for the treatment of inflammatory diseases
ANCLIFF RACHAEL ANNE, HODGSON SIMON TEANBY, LEWELL XIAO QING, ROBERTSON GRAEME MICHAEL
Year of Publication 14.07.2009
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Year of Publication 14.07.2009
Patent
HISTAMINE RECEPTOR ANTAGONISTS COMPRISING AN AZEPIN CORE
ANCLIFF, RACHAEL ANN, PARR, NIGEL, JAMES, HANCOCK, ASHLEY PAUL, KRANZ, MICHAEL JOACHIM
Year of Publication 25.02.2009
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Year of Publication 25.02.2009
Patent
SUBSTITUTED PIPERAZINES, (1,4) DIAZEPINES, AND 2,5-DIAZABICYCLO (2.2.1) HEPTANES AS HISTAMINE H1 AND/OR H3 ANTAGONISTS OR HISTAMINE H3 REVERSE ANTAGONISTS
HEIGHTMAN THOMAS DANIEL, WILSON DAVID MATTHEW, HODGSON SIMON TEANBY, ANCLIFF RACHAEL, ELDRED COLIN DAVID, HOBBS HEATHER, HANCOCK ASHLEY PAUL
Year of Publication 25.03.2010
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Year of Publication 25.03.2010
Patent
COMPOUNDS
HODGSON, SIMON, TEANBY, PARR, CHRISTOPHER, ALLAN, BAMFORD, MARK, JAMES, PROCOPIOU, PANAYIOTIS, ALEXANDROU, WILSON, DAVID, MATTHEW, ANCLIFF, RACHAEL, ANN, WOODROW, MICHAEL
Year of Publication 26.08.2009
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Year of Publication 26.08.2009
Patent