Novel Dual-Target Kinase Inhibitors of EGFR and ALK Were Designed, Synthesized, and Induced Cell Apoptosis in Non-Small Cell Lung Cancer
Fan, Yangyang, Li, Wei, Nie, Wenyan, Yao, Han, Ren, Yuanyuan, Wang, Mengxuan, Nie, Haoran, Gu, Chenxi, Liu, Jiadai, An, Baijiao
Published in Molecules (Basel, Switzerland) (21.02.2023)
Published in Molecules (Basel, Switzerland) (21.02.2023)
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Journal Article
A novel c-Met/TRK inhibitor 1D228 efficiently inhibits tumor growth by targeting angiogenesis and tumor cell proliferation
An, Baijiao, Nie, Wenyan, Hu, Jinhui, Fan, Yangyang, Nie, Haoran, Wang, Mengxuan, Zhao, Yaxuan, Yao, Han, Ren, Yuanyuan, Zhang, Chuanchuan, Wei, Mengna, Li, Wei, Liu, Jiadai, Yang, Chunhua, Zhang, Yin, Li, Xingshu, Tian, Geng
Published in Cell death & disease (09.11.2023)
Published in Cell death & disease (09.11.2023)
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Journal Article
Synthesis and evaluation of selenium-containing indole chalcone and diarylketone derivatives as tubulin polymerization inhibition agents
Zhang, Shun, An, Baijiao, Li, Jiayan, Hu, Jinhui, Huang, Ling, Li, Xingshu, Chan, Albert S. C.
Published in Organic & biomolecular chemistry (2017)
Published in Organic & biomolecular chemistry (2017)
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Journal Article
Synthesis and evaluation of new 2-chloro-4-aminopyrimidine and 2,6-dimethyl-4-aminopyrimidine derivatives as tubulin polymerization inhibitors
Xu, Shaoyu, An, Baijiao, Li, Yuxin, Luo, Xunbang, Li, Xingshu, Jia, Xian
Published in Bioorganic & medicinal chemistry letters (01.06.2018)
Published in Bioorganic & medicinal chemistry letters (01.06.2018)
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Journal Article
Glucagon Enhances Chemotherapy Efficacy By Inhibition of Tumor Vessels in Colorectal Cancer
Xu, Yuxue, Ni, Feixue, Sun, Daxi, Peng, Yue, Zhao, Yaxuan, Wu, Xiaojun, Li, Shasha, Qi, Xiangyu, He, Xinkang, Li, Min, Zhou, Yizi, Zhang, Chao, Yan, Miao, Yao, Cuifang, Zhu, Shuaishuai, Yang, Yang, An, Baijiao, Yang, Chunhua, Zhang, Guilong, Jiang, Wenguo, Mi, Jia, Chen, Xinju, Wei, Pengfei, Tian, Geng, Zhang, Yin
Published in Advanced science (01.02.2024)
Published in Advanced science (01.02.2024)
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Journal Article
Design, Synthesis, and Biological Evaluation of Novel Selenium-Containing Isocombretastatins and Phenstatins as Antitumor Agents
Pang, Yanqing, An, Baijiao, Lou, Lanlan, Zhang, Junsheng, Yan, Jun, Huang, Ling, Li, Xingshu, Yin, Sheng
Published in Journal of medicinal chemistry (14.09.2017)
Published in Journal of medicinal chemistry (14.09.2017)
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Journal Article
Synthesis and evaluation of clioquinol-rolipram/roflumilast hybrids as multitarget-directed ligands for the treatment of Alzheimer's disease
Hu, Jinhui, Pan, Tingting, An, Baijiao, Li, Zhengcunxiao, Li, Xingshu, Huang, Ling
Published in European journal of medicinal chemistry (01.02.2019)
Published in European journal of medicinal chemistry (01.02.2019)
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Journal Article
Design, synthesis, and biological evaluation of novel benzodiazepine derivatives as anticancer agents through inhibition of tubulin polymerization in vitro and in vivo
Pang, Yanqing, Lin, Haibiao, Ou, Caiwen, Cao, Yingying, An, Baijiao, Yan, Jun, Li, Xingshu
Published in European journal of medicinal chemistry (15.11.2019)
Published in European journal of medicinal chemistry (15.11.2019)
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Journal Article
Evaluation of 4-phenylamino-substituted naphthalene-1,2-diones as tubulin polymerization inhibitors
Yang, Honghao, An, Baijiao, Li, Xingshu, Zeng, Wei
Published in Bioorganic & medicinal chemistry letters (01.10.2018)
Published in Bioorganic & medicinal chemistry letters (01.10.2018)
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Journal Article
Design, synthesis and biological evaluation of novel 2,4-diaryl pyrimidine derivatives as selective EGFRL858R/T790M inhibitors
Li, Jianheng, An, Baijiao, Song, Xianheng, Zhang, Qianzhong, Chen, Chun, Wei, Shuxian, Fan, Runzhu, Li, Xingshu, Zou, Yong
Published in European journal of medicinal chemistry (15.02.2021)
Published in European journal of medicinal chemistry (15.02.2021)
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Journal Article
A Multifunctional Vanadium-Iron-Oxide Nanoparticle Eradicates Hepatocellular Carcinoma via Targeting Tumor and Endothelial Cells
Yang, Xiaoming, Xiao, Jianmin, Jiang, Lingyu, Ran, Lang, Fan, Yangyang, Zhang, Minghui, Xu, Yuxue, Yao, Cuifang, An, Baijiao, Yang, Yang, Yang, Chunhua, Tian, Geng, Zhang, Guilong, Zhang, Yin
Published in ACS applied materials & interfaces (29.06.2022)
Published in ACS applied materials & interfaces (29.06.2022)
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Journal Article
The synthesis and evaluation of new butadiene derivatives as tubulin polymerization inhibitors
Pang, Yanqing, Yan, Jun, An, Baijiao, Huang, Ling, Li, Xingshu
Published in Bioorganic & medicinal chemistry (15.06.2017)
Published in Bioorganic & medicinal chemistry (15.06.2017)
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Journal Article
Design, synthesis, and biological evaluation of histone deacetylase inhibitors possessing glutathione peroxidase-like and antioxidant activities against Alzheimer’s disease
Hu, Jinhui, An, Baijiao, Pan, Tingting, Li, Zhengcunxiao, Huang, Ling, Li, Xingshu
Published in Bioorganic & medicinal chemistry (15.11.2018)
Published in Bioorganic & medicinal chemistry (15.11.2018)
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Journal Article
Inhibition of TGF-β1/Smad3 signaling by compound 5aa: A potential treatment for idiopathic pulmonary fibrosis
An, Baijiao, Fang, Yanhua, Wang, Lihan, Nie, Wenyan, Wang, Mengxuan, Nie, Haoran, Wu, Chengjun, Wang, Ruoyu
Published in Bioorganic chemistry (01.06.2024)
Published in Bioorganic chemistry (01.06.2024)
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Journal Article
Synthesis and evaluation of new pirfenidone derivatives as anti-fibrosis agents
Gu, Chenxi, Li, Wei, Ju, Qing, Yao, Han, Yang, Lisheng, An, Baijiao, Hu, Wenhao, Li, Xingshu
Published in RSC advances (12.05.2022)
Published in RSC advances (12.05.2022)
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Journal Article
Novel third-generation pyrimidines-based EGFR tyrosine kinase inhibitors targeting EGFR T790M mutation in advanced non-small cell lung cancer
An, Baijiao, Liu, Jian, Fan, Yangyang, Nie, Wenyan, Yang, Chunhua, Yao, Han, Li, Wei, Zhang, Yin, Li, Xingshu, Tian, Geng
Published in Bioorganic chemistry (01.05.2022)
Published in Bioorganic chemistry (01.05.2022)
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Journal Article
The discovery of a potent and selective third-generation EGFR kinase inhibitor as a therapy for EGFR L858R/T790M double mutant non-small cell lung cancer
An, Baijiao, Pan, Tingting, Hu, Jinhui, Pang, Yanqing, Huang, Ling, Chan, Albert S.C., Li, Xingshu, Yan, Jun
Published in European journal of medicinal chemistry (01.12.2019)
Published in European journal of medicinal chemistry (01.12.2019)
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