Noncovalent structure of SENP1 in complex with SUMO2
Ambaye, Nigus D.
Published in Acta crystallographica. Section F, Structural biology communications (01.05.2019)
Published in Acta crystallographica. Section F, Structural biology communications (01.05.2019)
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Journal Article
Identification of the first small-molecule inhibitor of the REV7 DNA repair protein interaction
Actis, Marcelo L., Ambaye, Nigus D., Evison, Benjamin J., Shao, Youming, Vanarotti, Murugendra, Inoue, Akira, McDonald, Ezelle T., Kikuchi, Sotaro, Heath, Richard, Hara, Kodai, Hashimoto, Hiroshi, Fujii, Naoaki
Published in Bioorganic & medicinal chemistry (15.09.2016)
Published in Bioorganic & medicinal chemistry (15.09.2016)
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Journal Article
RWD Domain as an E2 (Ubc9)-Interaction Module
Alontaga, Aileen Y., Ambaye, Nigus D., Li, Yi-Jia, Vega, Ramir, Chen, Chih-Hong, Bzymek, Krzysztof P., Williams, John C., Hu, Weidong, Chen, Yuan
Published in The Journal of biological chemistry (03.07.2015)
Published in The Journal of biological chemistry (03.07.2015)
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Journal Article
Unexpected involvement of staple leads to redesign of selective bicyclic peptide inhibitor of Grb7
Gunzburg, Menachem J, Kulkarni, Ketav, Watson, Gabrielle M, Ambaye, Nigus D, Del Borgo, Mark P, Brandt, Rebecca, Pero, Stephanie C, Perlmutter, Patrick, Wilce, Matthew C J, Wilce, Jacqueline A
Published in Scientific reports (03.06.2016)
Published in Scientific reports (03.06.2016)
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Journal Article
Cyclic Peptides Incorporating Phosphotyrosine Mimetics as Potent and Specific Inhibitors of the Grb7 Breast Cancer Target
Watson, Gabrielle M., Gunzburg, Menachem J., Ambaye, Nigus D., Lucas, William A. H., Traore, Daouda A., Kulkarni, Ketav, Cergol, Katie M., Payne, Richard J., Panjikar, Santosh, Pero, Stephanie C., Perlmutter, Patrick, Wilce, Matthew C. J., Wilce, Jacqueline A.
Published in Journal of medicinal chemistry (08.10.2015)
Published in Journal of medicinal chemistry (08.10.2015)
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Journal Article
Design and testing of bicyclic inhibitors of Grb7-are two cycles better than one?
Gunzburg, Menachem J., Ambaye, Nigus D., Del Borgo, Mark P., Perlmutter, Patrick, Wilce, Jacqueline A.
Published in Biopolymers (01.09.2013)
Published in Biopolymers (01.09.2013)
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Journal Article
Potent antitumor effects of cell-penetrating peptides targeting STAT3 axis
Aftabizadeh, Maryam, Li, Yi-Jia, Zhao, Qianqian, Zhang, Chunyan, Ambaye, Nigus, Song, Jieun, Nagao, Toshikage, Lahtz, Christoph, Fakih, Marwan, Ann, David K, Yu, Hua, Herrmann, Andreas
Published in JCI insight (25.01.2021)
Published in JCI insight (25.01.2021)
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Journal Article
Structural Basis of Binding by Cyclic Nonphosphorylated Peptide Antagonists of Grb7 Implicated in Breast Cancer Progression
Ambaye, Nigus D., Pero, Stephanie C., Gunzburg, Menachem J., Yap, MinYin, Clayton, Daniel J., Del Borgo, Mark P., Perlmutter, Patrick, Aguilar, Marie-Isabel, Shukla, Girja S., Peletskaya, Elena, Cookson, Michelle M., Krag, David N., Wilce, Matthew C.J., Wilce, Jacqueline A.
Published in Journal of molecular biology (23.09.2011)
Published in Journal of molecular biology (23.09.2011)
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Journal Article
The Discovery of Phenylbenzamide Derivatives as Grb7-Based Antitumor Agents
Ambaye, Nigus D., Gunzburg, Menachem J., Lim, Reece C. C., Price, John T., Wilce, Matthew C. J., Wilce, Jacqueline A.
Published in ChemMedChem (01.02.2013)
Published in ChemMedChem (01.02.2013)
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Journal Article
Observation of an E2 (Ubc9)-homodimer by crystallography
Alontaga, Aileen Y., Ambaye, Nigus D., Li, Yi-Jia, Vega, Ramir, Chen, Chih-Hong, Bzymek, Krzysztof P., Williams, John C., Hu, Weidong, Chen, Yuan
Published in Data in brief (01.06.2016)
Published in Data in brief (01.06.2016)
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Journal Article
Interaction of the non-phosphorylated peptide G7-18NATE with Grb7-SH2 domain requires phosphate for enhanced affinity and specificity
Gunzburg, Menachem J., Ambaye, Nigus D., Del Borgo, Mark P., Pero, Stephanie C., Krag, David N., Wilce, Matthew C.J., Wilce, Jacqueline A.
Published in Journal of molecular recognition (01.01.2012)
Published in Journal of molecular recognition (01.01.2012)
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Journal Article
Preparation of crystals for characterizing the Grb7 SH2 domain before and after complex formation with a bicyclic peptide antagonist
Ambaye, Nigus D., Gunzburg, Menachem J., Traore, Daouda A. K., Del Borgo, Mark P., Perlmutter, Patrick, Wilce, Matthew C. J., Wilce, Jacqueline A.
Published in Acta crystallographica. Section F, Structural biology communications (01.02.2014)
Published in Acta crystallographica. Section F, Structural biology communications (01.02.2014)
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Journal Article
Use of SPR to Study the Interaction of G7-18NATE Peptide with the Grb7-SH2 Domain
Gunzburg, Menachem J., Ambaye, Nigus D., Hertzog, Jack T., Del Borgo, Mark P., Pero, Stephanie C., Krag, David N., Wilce, Matthew C. J., Aguilar, Marie-Isabel, Perlmutter, Patrick, Wilce, Jacqueline A.
Published in International journal of peptide research and therapeutics (01.09.2010)
Published in International journal of peptide research and therapeutics (01.09.2010)
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Journal Article
Streptonigrin Inhibits SENP1 and Reduces the Protein Level of Hypoxia-Inducible Factor 1α (HIF1α) in Cells
Ambaye, Nigus, Chen, Chih-Hong, Khanna, Swati, Li, Yi-Jia, Chen, Yuan
Published in Biochemistry (Easton) (20.03.2018)
Published in Biochemistry (Easton) (20.03.2018)
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Journal Article
Streptonigrin inhibits SENP1 and reduces the protein level of hypoxia-inducible factor 1 (HIF1α) in cells
Ambaye, Nigus, Chen, Chih-Hong, Khanna, Swati, Li, Yi-Jia, Chen, Yuan
Published in Biochemistry (Easton) (01.03.2018)
Published in Biochemistry (Easton) (01.03.2018)
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Journal Article
Uptake of a cell permeable G7-18NATE construct into cells and binding with the Grb7-SH2 domain
Ambaye, Nigus D., Lim, Reece C. C., Clayton, Daniel J., Gunzburg, Menachem J., Price, John T., Pero, Stephanie C., Krag, David N., Wilce, Matthew C. J., Aguilar, Marie-Isabel, Perlmutter, Patrick, Wilce, Jacqueline A.
Published in Peptide Science (2011)
Published in Peptide Science (2011)
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Journal Article
Uptake of a cell permeable G7-18NATE contruct into cells and binding with the Grb-7-SH2 domain
Ambaye, Nigus D, Lim, Reece C C, Clayton, Daniel J, Gunzburg, Menachem J, Price, John T, Pero, Stephanie C, Krag, David N, Wilce, Matthew C J, Aguilar, Marie-Isabel, Perlmutter, Patrick, Wilce, Jacqueline A
Published in Biopolymers (2011)
Published in Biopolymers (2011)
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Journal Article