Chirality determination of unusual amino acids using precolumn derivatization and liquid chromatography–electrospray ionization mass spectrometry
Hess, Sonja, Gustafson, Kirk R, Milanowski, Dennis J, Alvira, Edgardo, Lipton, Mark A, Pannell, Lewis K
Published in Journal of Chromatography A (07.05.2004)
Published in Journal of Chromatography A (07.05.2004)
Get full text
Journal Article
Synthesis and spectroscopic correlation of the diastereoisomers of 2,3-dihydroxy-2,6,8-trimethyldeca-(4 Z,6 E)-dienoic acid: implications for the structures of papuamides A–D and mirabamides A–D
Ramamoorthy, Gurusankar, Acevedo, Cristina M., Alvira, Edgardo, Lipton, Mark A.
Published in Tetrahedron: asymmetry (17.11.2008)
Published in Tetrahedron: asymmetry (17.11.2008)
Get full text
Journal Article
Discovery of N-substituted pyridinones as potent and selective inhibitors of p38 kinase
Selness, Shaun R., Devraj, Rajesh V., Monahan, Joseph B., Boehm, Terri L., Walker, John K., Devadas, Balekudru, Durley, Richard C., Kurumbail, Ravi, Shieh, Huey, Xing, Li, Hepperle, Michael, Rucker, Paul V., Jerome, Kevin D., Benson, Alan G., Marrufo, Laura D., Madsen, Heather M., Hitchcock, Jeff, Owen, Tom J., Christie, Lance, Promo, Michele A., Hickory, Brian S., Alvira, Edgardo, Naing, Win, Blevis-Bal, Radhika
Published in Bioorganic & medicinal chemistry letters (15.10.2009)
Published in Bioorganic & medicinal chemistry letters (15.10.2009)
Get full text
Journal Article
Discovery of PH-797804, a highly selective and potent inhibitor of p38 MAP kinase
Selness, Shaun R, Devraj, Rajesh V, Devadas, Balekudru, Walker, John K, Boehm, Terri L, Durley, Richard C, Shieh, Huey, Xing, Li, Rucker, Paul V, Jerome, Kevin D, Benson, Alan G, Marrufo, Laura D, Madsen, Heather M, Hitchcock, Jeff, Owen, Tom J, Christie, Lance, Promo, Michele A, Hickory, Brian S, Alvira, Edgardo, Naing, Win, Blevis-Bal, Radhika, Messing, Dean, Yang, Jerry, Mao, Michael K, Yalamanchili, Gopi, Vonder Embse, Richard, Hirsch, Jeffrey, Saabye, Matthew, Bonar, Sheri, Webb, Elizabeth, Anderson, Gary, Monahan, Joseph B
Published in Bioorganic & medicinal chemistry letters (01.07.2011)
Published in Bioorganic & medicinal chemistry letters (01.07.2011)
Get full text
Journal Article
Design, synthesis and activity of a potent, selective series of N-aryl pyridinone inhibitors of p38 kinase
Selness, Shaun R, Boehm, Terri L, Walker, John K, Devadas, Balekudru, Durley, Richard C, Kurumbail, Ravi, Shieh, Huey, Xing, Li, Hepperle, Michael, Rucker, Paul V, Jerome, Kevin D, Benson, Alan G, Marrufo, Laura D, Madsen, Heather M, Hitchcock, Jeff, Owen, Tom J, Christie, Lance, Promo, Michele A, Hickory, Brian S, Alvira, Edgardo, Naing, Win, Blevis-Bal, Radhika, Devraj, Rajesh V, Messing, Dean, Schindler, John F, Hirsch, Jeffrey, Saabye, Matthew, Bonar, Sheri, Webb, Elizabeth, Anderson, Gary, Monahan, Joseph B
Published in Bioorganic & medicinal chemistry letters (01.07.2011)
Published in Bioorganic & medicinal chemistry letters (01.07.2011)
Get full text
Journal Article
Enzyme activation in organic solvents: Co-lyophilization of subtilisin Carlsberg with methyl-β-cyclodextrin renders an enzyme catalyst more active than the cross-linked enzyme crystals
Montañez-Clemente, Ileana, Alvira, Edgardo, Macias, Minedys, Ferrer, Amaris, Fonceca, Maricely, Rodriguez, Jessica, Gonzalez, Anicele, Barletta, Gabriel
Published in Biotechnology and bioengineering (05.04.2002)
Published in Biotechnology and bioengineering (05.04.2002)
Get full text
Journal Article
PYRAZOLE DERIVATIVES AS 5-LO INHIBITORS
SCHMIDT MICHELLE ANN, WAGNER GRACE MARY, GRANETO MATTHEW J, SELBO JON GORDON, TOLLEFSON MICHAEL BRENT, MASSA MARK ALAN, WOODARD SCOTT SANTFORD, ALVIRA EDGARDO, IYANAR KALIAPPAN, SAMPLE KIRBY RAY, VONDER EMBSE RICHARD ALAN, MAHONEY MATTHEW WILLIAM, GRAPPERHAUS MARGARET LANAHAN, SEIDEL RONALD EDWARD, MADDUX TODD MICHAEL
Year of Publication 29.06.2010
Get full text
Year of Publication 29.06.2010
Patent
High Initial Activity but Low Storage Stability Observed for Several Preparations of Subtilisin Carslberg Suspended in Organic Solvents
Martínez, Susimar González, Alvira, Edgardo, Cordero, Liz Vergara, Ferrer, Amaris, Montañés-Clemente, Ileana, Barletta, Gabriel
Published in Biotechnology progress (2002)
Published in Biotechnology progress (2002)
Get full text
Journal Article
Pyrazole derivatives as 5-LO inhibitors
MAHONEY MATTHEW WILLIAM, GRAPPERHAUS MARGARET LANAHAN, ALVIRA EDGARDO
Year of Publication 30.06.2010
Get full text
Year of Publication 30.06.2010
Patent
Pyrazole derivatives as 5-LO inhibitors
MAHONEY MATTHEW WILLIAM, GRAPPERHAUS MARGARET LANAHAN, ALVIRA EDGARDO
Year of Publication 30.06.2010
Get full text
Year of Publication 30.06.2010
Patent
SUBSTITUTED PYRIDINONES AS MODULATORS OF P38 MAP KINASE
MADSEN HEATHER M, NAING WIN, WALKER JOHN, DEVRAJ RAJESH, PROMO MICHELE A, MCGEE KEVIN F, DURLEY RICHARD C, BLEVIS-BAL RADHIKA M, OWEN THOMAS, SELNESS SHAUN R, ALVIRA EDGARDO, SHIEH HUEY S, JEROME KEVIN D, BOEHM TERRI L, LIU SHUANG, HITCHCOCK JEFF, SAMBANDAM ARUNA, DEVADAS BALEKUDRU, HICKORY BRIAN S, SCOTT IAN L, MARRUFO LAURA D, RUCKER PAUL V, XING LI
Year of Publication 30.01.2015
Get full text
Year of Publication 30.01.2015
Patent
ΥΠΟΚΑΤΕΣΤΗΜΕΝΕΣ ΠΥΡΙΔΙΝΟΝΕΣ ΩΣ ΡΥΘΜΙΣΤΕΣ ΤΗΣ Ρ38 ΜΑΡ ΚΙΝΑΣΗΣ
MADSEN HEATHER M, NAING WIN, WALKER JOHN, DEVRAJ RAJESH, PROMO MICHELE A, MCGEE KEVIN F, DURLEY RICHARD C, BLEVIS-BAL RADHIKA M, OWEN THOMAS, SELNESS SHAUN R, ALVIRA EDGARDO, SHIEH HUEY S, JEROME KEVIN D, BOEHM TERRI L, LIU SHUANG, HITCHCOCK JEFF, SAMBANDAM ARUNA, DEVADAS BALEKUDRU, HICKORY BRIAN S, SCOTT IAN L, MARRUFO LAURA D, RUCKER PAUL V, XING LI
Year of Publication 13.08.2014
Get full text
Year of Publication 13.08.2014
Patent
derivados de pirazol como inibidores de 5-lo
Kirby Ray Sample, Mark Alan Massa, Michael Brent Tollefson, Jon Gordon Selbo, Richard Alan Vonder Embse, Kaliappan Iyanar, Michelle Ann Schimdt, Todd Michael Maddux, Grace Mary Wagner, Matthew William Mahoney, Ronald Edward Seidel, Edgardo Alvira, Matthew J. Graneto, Scott Santford Woodard, Margaret Lanahan Grapperhaus
Year of Publication 24.09.2019
Get full text
Year of Publication 24.09.2019
Patent
SUBSTITUTED PYRIDINONES AS MODULATORS OF P38 MAP KINASE
SELNESS, SHAUN R, NAING, WIN, DURLEY, RICHARD C, WALKER, JOHN, HITCHCOCK, JEFF, SCOTT, IAN L, PROMO, MICHELE A, MCGEE, KEVIN F, MARRUFO, LAURA D, SAMBANDAM, ARUNA, LIU, SHUANG, XING, LI, SHIEH, HUEY S, BLEVIS-BAL, RADHIKA M, BOEHM, TERRI L, DEVRAJ, RAJESH, DEVADAS, BALEKUDRU, RUCKER, PAUL V, MADSEN, HEATHER M, OWEN, THOMAS, JEROME, KEVIN D, ALVIRA, EDGARDO, HICKORY, BRIAN S
Year of Publication 28.02.2013
Get full text
Year of Publication 28.02.2013
Patent
SUPSTITUTED PYRIDINONES AS MODULATORS OF P38 MAP KINASE
SELNESS, SHAUN R, NAING, WIN, WALKER, JOHN, SCOTT, IAN L, DURLEY, RICHARD, JEROME, KEVIN, D, BOEHM, TERRI, L, PROMO, MICHELE A, MCGEE, KEVIN F, MARRUFO, LAURA D, SAMBANDAM, ARUNA, LIU, SHUANG, XING, LI, SHIEH, HUEY S, BLEVIS-BAL, RADHIKA M, HITCHOCK, JEFF, DEVRAJ, RAJESH, DEVADAS, BALEKUDRU, RUCKER, PAUL V, MADSEN, HEATHER M, OWEN, THOMAS, ALVIRA, EDGARDO, HICKORY, BRIAN S
Year of Publication 31.12.2012
Get full text
Year of Publication 31.12.2012
Patent
PYRAZOLE DERIVATIVES AS 5-LO INHIBITORS
SEIDEL, RONALD EDWARD, TOLLEFSON, MICHAEL BRENT, VONDER EMBSE, RICHARD ALAN, MASSA, MARK ALAN, WOODARD, SCOTT SANTFORD, IYANAR, KALIAPPAN, GRAPPERHAUS, MARGARET LANAHAN, SAMPLE, KIRBY RAY, SELBO, JON GORDON, WAGNER, GRACE MARY, MADDUX, TODD MICHAEL, MAHONEY, MATTHEW WILLIAM, SCHMIDT, MICHELLE ANN, GRANETO, MATTHEW JAMES, ALVIRA, EDGARDO
Year of Publication 18.09.2012
Get full text
Year of Publication 18.09.2012
Patent
Pyrazole derivatives as 5-LO-inhibitors
SCHMIDT MICHELLE ANN, WAGNER GRACE MARY, GRANETO MATTHEW J, SELBO JON GORDON, TOLLEFSON MICHAEL BRENT, MASSA MARK ALAN, WOODARD SCOTT SANTFORD, ALVIRA EDGARDO, IYANAR KALIAPPAN, SAMPLE KIRBY RAY, VONDER EMBSE RICHARD ALAN, MAHONEY MATTHEW WILLIAM, GRAPPERHAUS MARGARET LANAHAN, SEIDEL RONALD EDWARD, MADDUX TODD MICHAEL
Year of Publication 17.01.2012
Get full text
Year of Publication 17.01.2012
Patent
Pyrazole derivatives as 5-LO-inhibitors
Alvira, Edgardo, Graneto, Matthew J, Grapperhaus, Margaret Lanahan, Iyanar, Kaliappan, Maddux, Todd Michael, Mahoney, Matthew William, Massa, Mark Alan, Sample, Kirby Ray, Schmidt, Michelle Ann, Seidel, Ronald Edward, Selbo, Jon Gordon, Tollefson, Michael Brent, Vonder Embse, Richard Alan, Wagner, Grace Mary, Woodard, Scott Santford
Year of Publication 17.01.2012
Get full text
Year of Publication 17.01.2012
Patent
PYRAZOLE DERIVATIVES AS 5-LO INHIBITORS
SCHMIDT MICHELLE ANN, WAGNER GRACE MARY, GRANETO MATTHEW J, TOLLEFSON MICHAEL BRENT, MASSA MARK ALAN, SELBO JON, WOODARD SCOTT SANTFORD, ALVIRA EDGARDO, IYANAR KALIAPPAN, SAMPLE RAY KIRBY, VONDER EMBSE RICHARD ALAN, MAHONEY MATTHEW WILLIAM, GRAPPERHAUS MARGARET LANAHAN, SEIDEL RONALD EDWARD, MADDUX TODD MICHAEL
Year of Publication 29.06.2011
Get full text
Year of Publication 29.06.2011
Patent