Design, synthesis and antiproliferative evaluation of new acridine-thiosemicarbazone derivatives as topoisomerase IIα inhibitors
Leonel Silva Sousa, Gleyton, da Silva Honório, Thiago, de Souza Furtado, Priscila, Simon, Alice, Mendes Cabral, Lucio, Rodrigues Coutinho Pereira, Gabriel, Emanuel Ferreira Alves, Josival, Mônica Vitalino de Almeida, Sinara, Rodrigues Silva, Valdenizia, de Souza Santos, Luciano, Pereira Bezerra, Daniel, Nora Castro, Rosane, Olímpio de Moura, Ricardo, Eugen Kümmerle, Arthur
Published in Results in Chemistry (01.01.2024)
Published in Results in Chemistry (01.01.2024)
Get full text
Journal Article
Novel indole-thiazole and indole-thiazolidinone derivatives as DNA groove binders
Alves, Josival Emanuel Ferreira, de Oliveira, Jamerson Ferreira, de Lima Souza, Tulio Ricardo Couto, de Moura, Ricardo Olímpio, de Carvalho Júnior, Luiz Bezerra, Alves de Lima, Maria do Carmo, de Almeida, Sinara Mônica Vitalino
Published in International journal of biological macromolecules (15.02.2021)
Published in International journal of biological macromolecules (15.02.2021)
Get full text
Journal Article
COVID-19 therapy: What weapons do we bring into battle?
de Almeida, Sinara Mônica Vitalino, Santos Soares, José Cleberson, dos Santos, Keriolaine Lima, Alves, Josival Emanuel Ferreira, Ribeiro, Amélia Galdino, Jacob, Íris Trindade Tenório, da Silva Ferreira, Cindy Juliane, dos Santos, Jéssica Celerino, de Oliveira, Jamerson Ferreira, de Carvalho Junior, Luiz Bezerra, de Lima, Maria do Carmo Alves
Published in Bioorganic & medicinal chemistry (01.12.2020)
Published in Bioorganic & medicinal chemistry (01.12.2020)
Get full text
Journal Article
A simple method for obtaining human albumin and its use for in vitro interaction assays with indole-thiazole and indole-thiazolidinone derivatives
Alves, Josival Emanuel Ferreira, Lucena, Maria Luiza Cavalcanti, de Souza Lucena, Antônio Edson, das Merces, Aurenice Arruda Dutra, de Azevedo, Rafael David Souto, Sousa, Gleyton Leonel Silva, de Moura, Ricardo Olimpio, Alves de Lima, Maria do Carmo, de Carvalho Júnior, Luiz Bezerra, de Almeida, Sinara Mônica Vitalino
Published in International journal of biological macromolecules (01.12.2021)
Published in International journal of biological macromolecules (01.12.2021)
Get full text
Journal Article
Topoisomerase inhibition and albumin interaction studies of acridine-thiosemicarbazone derivatives
da Silva Filho, Francivaldo Araújo, de Freitas Souza, Thais, Ribeiro, Amélia Galdino, Alves, Josival Emanuel Ferreira, de Oliveira, Jamerson Ferreira, de Lima Souza, Túlio Ricardo Couto, de Moura, Ricardo Olímpio, do Carmo Alves de Lima, Maria, de Carvalho Junior, Luiz Bezerra, de Almeida, Sinara Mônica Vitalino
Published in International journal of biological macromolecules (01.10.2019)
Published in International journal of biological macromolecules (01.10.2019)
Get full text
Journal Article
Albumin roles in developing anticancer compounds
Ribeiro, Amélia Galdino, Alves, Josival Emanuel Ferreira, Soares, José Cleberson Santos, dos Santos, Keriolaine Lima, Jacob, Íris Trindade Tenório, da Silva Ferreira, Cindy Juliane, dos Santos, Jéssica Celerino, de Azevedo, Rafael David Souto, de Almeida, Sinara Mônica Vitalino, de Lima, Maria do Carmo Alves
Published in Medicinal chemistry research (01.08.2021)
Published in Medicinal chemistry research (01.08.2021)
Get full text
Journal Article
Study of nitrogen heterocycles as DNA/HSA binder, topoisomerase inhibitors and toxicological safety
Dos Santos, Jéssica Celerino, Alves, Josival Emanuel Ferreira, de Azevedo, Rafael David Souto, de Lima, Maksuelly Libanio, de Oliveira Silva, Maria Regina, da Silva, Josefa Gerlane, da Silva, Jamire Muriel, de Carvalho Correia, Ana Carolina, do Carmo Alves de Lima, Maria, de Oliveira, Jamerson Ferreira, de Moura, Ricardo Olímpio, de Almeida, Sinara Mônica Vitalino
Published in International journal of biological macromolecules (01.01.2024)
Published in International journal of biological macromolecules (01.01.2024)
Get full text
Journal Article
Interaction study with DNA/HSA, anti-topoisomerase IIα, cytotoxicity and in vitro antiproliferative evaluations and molecular docking of indole-thiosemicarbazone compounds
Jacob, Iris Trindade, da Cruz Filho, Iranildo José, Alves, Josival Emanuel Ferreira, de Melo Souza, Felipe, de Azevedo, Rafael David Souto, Marques, Diego Santa Clara, de Lima Souza, Túlio Ricardo Couto, dos Santos, Keriolaine Lima, da Rocha Pitta, Maira Galdino, de Melo Rêgo, Moacyr Jesus Barreto, Oliveira, Jamerson Ferreira, Almeida, Sinara Mônica Vitalino, do Carmo Alves de Lima, Maria
Published in International journal of biological macromolecules (15.04.2023)
Published in International journal of biological macromolecules (15.04.2023)
Get full text
Journal Article
DNA binding and Topoisomerase inhibition: How can these mechanisms be explored to design more specific anticancer agents?
de Almeida, Sinara Mônica Vitalino, Ribeiro, Amélia Galdino, de Lima Silva, Geilza Carla, Ferreira Alves, Josival Emanuel, Beltrão, Eduardo Isidoro Carneiro, de Oliveira, Jamerson Ferreira, de Carvalho, Luiz Bezerra, Alves de Lima, Maria do Carmo
Published in Biomedicine & pharmacotherapy (01.12.2017)
Published in Biomedicine & pharmacotherapy (01.12.2017)
Get full text
Journal Article