Targeted inhibition of the COP9 signalosome for treatment of cancer
Schlierf, Anita, Altmann, Eva, Quancard, Jean, Jefferson, Anne B, Assenberg, René, Renatus, Martin, Jones, Matthew, Hassiepen, Ulrich, Schaefer, Michael, Kiffe, Michael, Weiss, Andreas, Wiesmann, Christian, Sedrani, Richard, Eder, Jörg, Martoglio, Bruno
Published in Nature communications (24.10.2016)
Published in Nature communications (24.10.2016)
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Journal Article
The Most Common Functional Groups in Bioactive Molecules and How Their Popularity Has Evolved over Time
Ertl, Peter, Altmann, Eva, McKenna, Jeffrey M
Published in Journal of medicinal chemistry (13.08.2020)
Published in Journal of medicinal chemistry (13.08.2020)
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Journal Article
The most common linkers in bioactive molecules and their bioisosteric replacement network
Ertl, Peter, Altmann, Eva, Racine, Sophie
Published in Bioorganic & medicinal chemistry (01.03.2023)
Published in Bioorganic & medicinal chemistry (01.03.2023)
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Journal Article
Which boronic acids are used most frequently for synthesis of bioactive molecules?
Ertl, Peter, Altmann, Eva, Racine, Sophie, Decoret, Odile
Published in Bioorganic & medicinal chemistry (15.08.2023)
Published in Bioorganic & medicinal chemistry (15.08.2023)
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Journal Article
Ring replacement recommender: Ring modifications for improving biological activity
Ertl, Peter, Altmann, Eva, Racine, Sophie, Lewis, Richard
Published in European journal of medicinal chemistry (05.08.2022)
Published in European journal of medicinal chemistry (05.08.2022)
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Journal Article
Design and Biochemical Characterization of Peptidic Inhibitors of the Myb/p300 Interaction
Jones, Matthew, Grosche, Philipp, Floersheimer, Andreas, André, Jérome, Gattlen, Raphael, Oser, Dieter, Tinchant, Juliette, Wille, Roman, Chie-Leon, Barbara, Gerspacher, Marc, Ertl, Peter, Ostermann, Nils, Altmann, Eva, Manchado, Eusebio, Vorherr, Thomas, Chène, Patrick
Published in Biochemistry (Easton) (04.04.2023)
Published in Biochemistry (Easton) (04.04.2023)
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Journal Article
Complementary use of ion trap/time-of-flight mass spectrometry in combination with capillary high-pressure liquid chromatography: early characterization of in vivo metabolites of the cathepsin K inhibitor NVP-AAV490 in rat
Blum, Wolfgang, Buhl, Thomas, Altmann, Eva, Kühnöl, Jürgen, Ramstein, Philippe, Aichholz, Reiner
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (25.04.2003)
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (25.04.2003)
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Journal Article
MicroCycle: An Integrated and Automated Platform to Accelerate Drug Discovery
Brocklehurst, Cara E., Altmann, Eva, Bon, Corentin, Davis, Holly, Dunstan, David, Ertl, Peter, Ginsburg-Moraff, Carol, Grob, Jonathan, Gosling, Daniel J., Lapointe, Guillaume, Marziale, Alexander N., Mues, Heinrich, Palmieri, Marco, Racine, Sophie, Robinson, Richard I., Springer, Clayton, Tan, Kian, Ulmer, William, Wyler, René
Published in Journal of medicinal chemistry (08.02.2024)
Published in Journal of medicinal chemistry (08.02.2024)
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Journal Article
Correction to “MicroCycle: An Integrated and Automated Platform to Accelerate Drug Discovery”
Brocklehurst, Cara E., Altmann, Eva, André, Jérôme, Bon, Corentin, Caya, Thomas, Davis, Holly, Decoret, Odile, Dunstan, David, Ertl, Peter, Ginsburg-Moraff, Carol, Grob, Jonathan, Gosling, Daniel J., Lapointe, Guillaume, Majumdar, Dyuti, Marziale, Alexander N., Mues, Heinrich, Palmieri, Marco, Racine, Sophie, Robinson, Richard I., Springer, Clayton, Tan, Kian, Ulmer, William, West, Laura, Wyler, René
Published in Journal of medicinal chemistry (28.03.2024)
Published in Journal of medicinal chemistry (28.03.2024)
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Journal Article
Discovery of Potent, Highly Selective, and In Vivo Efficacious, Allosteric MALT1 Inhibitors by Iterative Scaffold Morphing
Pissot Soldermann, Carole, Simic, Oliver, Renatus, Martin, Erbel, Paulus, Melkko, Samu, Wartmann, Markus, Bigaud, Marc, Weiss, Andreas, McSheehy, Paul, Endres, Ralf, Santos, Paulo, Blank, Jutta, Schuffenhauer, Ansgar, Bold, Guido, Buschmann, Nicole, Zoller, Thomas, Altmann, Eva, Manley, Paul W, Dix, Ina, Buchdunger, Elisabeth, Scesa, Julien, Quancard, Jean, Schlapbach, Achim, Bornancin, Frédéric, Radimerski, Thomas, Régnier, Catherine H
Published in Journal of medicinal chemistry (10.12.2020)
Published in Journal of medicinal chemistry (10.12.2020)
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Journal Article
Azaindoles as Zinc‐Binding Small‐Molecule Inhibitors of the JAMM Protease CSN5
Altmann, Eva, Erbel, Paul, Renatus, Martin, Schaefer, Michael, Schlierf, Anita, Druet, Adelaide, Kieffer, Laurence, Sorge, Mickael, Pfister, Keith, Hassiepen, Ulrich, Jones, Matthew, Ruedisser, Simon, Ostermeier, Daniela, Martoglio, Bruno, Jefferson, Anne B., Quancard, Jean
Published in Angewandte Chemie International Edition (24.01.2017)
Published in Angewandte Chemie International Edition (24.01.2017)
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Journal Article
Structure-Based Design and Preclinical Characterization of Selective and Orally Bioavailable Factor XIa Inhibitors: Demonstrating the Power of an Integrated S1 Protease Family Approach
Lorthiois, Edwige, Roache, James, Barnes-Seeman, David, Altmann, Eva, Hassiepen, Ulrich, Turner, Gordon, Duvadie, Rohit, Hornak, Viktor, Karki, Rajeshri G, Schiering, Nikolaus, Weihofen, Wilhelm A, Perruccio, Francesca, Calhoun, Amy, Fazal, Tanzina, Dedic, Darija, Durand, Corinne, Dussauge, Solene, Fettis, Kamal, Tritsch, Fabien, Dentel, Celine, Druet, Adelaide, Liu, Donglei, Kirman, Louise, Lachal, Julie, Namoto, Kenji, Bevan, Douglas, Mo, Rose, Monnet, Gabriela, Muller, Lionel, Zessis, Richard, Huang, Xueming, Lindsley, Loren, Currie, Treeve, Chiu, Yu-Hsin, Fridrich, Cary, Delgado, Peter, Wang, Shuangxi, Hollis-Symynkywicz, Micah, Berghausen, Joerg, Williams, Eric, Liu, Hong, Liang, Guiqing, Kim, Hyungchul, Hoffmann, Peter, Hein, Andreas, Ramage, Paul, D’Arcy, Allan, Harlfinger, Stefanie, Renatus, Martin, Ruedisser, Simon, Feldman, David, Elliott, Jason, Sedrani, Richard, Maibaum, Juergen, Adams, Christopher M
Published in Journal of medicinal chemistry (13.08.2020)
Published in Journal of medicinal chemistry (13.08.2020)
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Journal Article
Structural Basis of Substrate Recognition and Covalent Inhibition of Cdu1 from Chlamydia trachomatis
Ramirez, Yesid A., Adler, Thomas B., Altmann, Eva, Klemm, Theresa, Tiesmeyer, Christian, Sauer, Florian, Kathman, Stefan G., Statsyuk, Alexander V., Sotriffer, Christoph, Kisker, Caroline
Published in ChemMedChem (08.10.2018)
Published in ChemMedChem (08.10.2018)
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Journal Article
Front Cover: Structural Basis of Substrate Recognition and Covalent Inhibition of Cdu1 from Chlamydia trachomatis (ChemMedChem 19/2018)
Ramirez, Yesid A., Adler, Thomas B., Altmann, Eva, Klemm, Theresa, Tiesmeyer, Christian, Sauer, Florian, Kathman, Stefan G., Statsyuk, Alexander V., Sotriffer, Christoph, Kisker, Caroline
Published in ChemMedChem (08.10.2018)
Published in ChemMedChem (08.10.2018)
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Journal Article
Structure-based design and optimization of potent inhibitors of the adenoviral protease
Grosche, Philipp, Sirockin, Finton, Mac Sweeney, Aengus, Ramage, Paul, Erbel, Paul, Melkko, Samu, Bernardi, Anna, Hughes, Nicola, Ellis, David, Combrink, Keith D., Jarousse, Nadine, Altmann, Eva
Published in Bioorganic & medicinal chemistry letters (01.02.2015)
Published in Bioorganic & medicinal chemistry letters (01.02.2015)
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Journal Article
Discovery and Structure-Based Optimization of Adenain Inhibitors
Mac Sweeney, Aengus, Grosche, Philipp, Ellis, David, Combrink, Keith, Erbel, Paul, Hughes, Nicola, Sirockin, Finton, Melkko, Samu, Bernardi, Anna, Ramage, Paul, Jarousse, Nadine, Altmann, Eva
Published in ACS medicinal chemistry letters (14.08.2014)
Published in ACS medicinal chemistry letters (14.08.2014)
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Journal Article
1-Alkyl-4-phenyl-6-alkoxy-1H-quinazolin-2-ones: A Novel Series of Potent Calcium-Sensing Receptor Antagonists
Widler, Leo, Altmann, Eva, Beerli, René, Breitenstein, Werner, Bouhelal, Rochdi, Buhl, Thomas, Gamse, Rainer, Gerspacher, Marc, Halleux, Christine, John, Markus R, Lehmann, Hansjoerg, Kalb, Oskar, Kneissel, Michaela, Missbach, Martin, Müller, Irene R, Reidemeister, Sibylle, Renaud, Johanne, Taillardat, Agnes, Tommasi, Ruben, Weiler, Sven, Wolf, Romain M, Seuwen, Klaus
Published in Journal of medicinal chemistry (11.03.2010)
Published in Journal of medicinal chemistry (11.03.2010)
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Journal Article
2-Cyano-pyrimidines: A New Chemotype for Inhibitors of the Cysteine Protease Cathepsin K
Altmann, Eva, Aichholz, Reiner, Betschart, Claudia, Buhl, Thomas, Green, Jonathan, Irie, Osamu, Teno, Naoki, Lattmann, René, Tintelnot-Blomley, Marina, Missbach, Martin
Published in Journal of medicinal chemistry (22.02.2007)
Published in Journal of medicinal chemistry (22.02.2007)
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Journal Article