Synthesis and evaluation of hybrid sulfonamide‐chalcones with potential antileishmanial activity
Oliveira, Nathalia S., Souza, Luana G., Almeida, Vitor M., Barreto, Arielly R. R., Carvalho‐Gondim, Felipe, Schaeffer, Edgar, Santos‐Filho, Osvaldo A., Rossi‐Bergmann, Bartira, Silva, Alcides J. M.
Published in Archiv der Pharmazie (Weinheim) (01.03.2024)
Published in Archiv der Pharmazie (Weinheim) (01.03.2024)
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Differences in Gluco and Galacto Substrate-Binding Interactions in a Dual 6Pβ-Glucosidase/6Pβ-Galactosidase Glycoside Hydrolase 1 Enzyme from Bacillus licheniformis
Veldman, Wayde, Liberato, Marcelo Vizona, Souza, Valquiria P, Almeida, Vitor M, Marana, Sandro R, Tastan Bishop, Özlem, Polikarpov, Igor
Published in Journal of chemical information and modeling (27.09.2021)
Published in Journal of chemical information and modeling (27.09.2021)
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Journal Article
Rational Exploration of 2,4-Diaminopyrimidines as DHFR Inhibitors Active against Mycobacterium abscessus and Mycobacterium avium , Two Emerging Human Pathogens
Andrade Meirelles, Matheus, Almeida, Vitor M, Sullivan, Jaryd R, de Toledo, Ian, Dos Reis, Caio Vinicius, Cunha, Micael Rodrigues, Zigweid, Rachel, Shim, Abraham, Sankaran, Banumathi, Woodward, Elijah L, Seibold, Steve, Liu, Lijun, Mian, Mohammad Rasel, Battaile, Kevin P, Riley, Jennifer, Duncan, Christina, Simeons, Frederick R C, Ferguson, Liam, Joji, Halimatu, Read, Kevin D, Lovell, Scott, Staker, Bart L, Behr, Marcel A, Pilli, Ronaldo A, Couñago, Rafael M
Published in Journal of medicinal chemistry (28.10.2024)
Published in Journal of medicinal chemistry (28.10.2024)
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Journal Article
Aurones: A Promising Scaffold to Inhibit SARS-CoV‑2 Replication
Caleffi, Guilherme S., Rosa, Alice S., de Souza, Luana G., Avelar, João L. S., Nascimento, Sarah M. R., de Almeida, Vitor M., Tucci, Amanda R., Ferreira, Vivian N., da Silva, Alcides J. M., Santos-Filho, Osvaldo A., Miranda, Milene D., Costa, Paulo R. R.
Published in Journal of natural products (Washington, D.C.) (23.06.2023)
Published in Journal of natural products (Washington, D.C.) (23.06.2023)
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Discovery of pyrazolo[3,4-d]pyrimidines as novel mitogen-activated protein kinase kinase 3 (MKK3) inhibitors
Takarada, Jessica E., Cunha, Micael R., Almeida, Vitor M., Vasconcelos, Stanley N. S., Santiago, Andre S., Godoi, Paulo H., Salmazo, Anita, Ramos, Priscila Z., Fala, Angela M., De Souza, Lucas R., Da Silva, Italo E. P., Bengtson, Mario H., Massirer, Katlin B., Counago, Rafael M.
Published in Bioorganic & medicinal chemistry (15.01.2024)
Published in Bioorganic & medicinal chemistry (15.01.2024)
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Identification of potential inhibitors of casein kinase 2 alpha of Plasmodium falciparum with potent in vitro activity
Tomaz, Kaira C P, Tavella, Tatyana A, Borba, Joyce V B, Salazar-Alvarez, Luis C, Levandoski, João E, Mottin, Melina, Sousa, Bruna K P, Moreira-Filho, José T, Almeida, Vitor M, Clementino, Leandro C, Bourgard, Catarina, Massirer, Katlin B, Couñago, Rafael M, Andrade, Carolina H, Sunnerhagen, Per, Bilsland, Elizabeth, Cassiano, Gustavo C, Costa, Fabio T M
Published in Antimicrobial agents and chemotherapy (15.11.2023)
Published in Antimicrobial agents and chemotherapy (15.11.2023)
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X‑ray Structure, Bioinformatics Analysis, and Substrate Specificity of a 6‑Phospho-β-glucosidase Glycoside Hydrolase 1 Enzyme from Bacillus licheniformis
Veldman, Wayde, Liberato, Marcelo Vizona, Almeida, Vitor M, Souza, Valquiria P, Frutuoso, Maira A, Marana, Sandro R, Moses, Vuyani, Tastan Bishop, Özlem, Polikarpov, Igor
Published in Journal of chemical information and modeling (28.12.2020)
Published in Journal of chemical information and modeling (28.12.2020)
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Journal Article
Novel centratherin derivatives: Molecular docking design, asymmetric synthesis, and antitumoral activity
H. R. de Oliveira, Pedro, C. R. M. da Frota, Lívia, M. Borges, Ricardo, A. Q. Beraldini, Monah, M. de Almeida, Vitor, A. Santos-Filho, Osvaldo, P. G. A. Fontão, Ana, L. F. Sampaio, André, G. Finelli, Fernanda
Published in Tetrahedron (03.08.2024)
Published in Tetrahedron (03.08.2024)
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Novel Dihydropteridinone Derivatives As Potent Inhibitors of the Understudied Human Kinases Vaccinia-Related Kinase 1 and Casein Kinase 1δ/ε
de Souza Gama, Fernando H., Dutra, Luiz A., Hawgood, Michael, dos Reis, Caio Vinícius, Serafim, Ricardo A. M., Ferreira, Marcos A., Teodoro, Bruno V. M., Takarada, Jéssica Emi, Santiago, André S., Balourdas, Dimitrios-Ilias, Nilsson, Ann-Sofie, Urien, Bruno, Almeida, Vitor M., Gileadi, Carina, Ramos, Priscila Z., Salmazo, Anita, Vasconcelos, Stanley N. S., Cunha, Micael R., Mueller, Susanne, Knapp, Stefan, Massirer, Katlin B., Elkins, Jonathan M., Gileadi, Opher, Mascarello, Alessandra, Lemmens, Bennie B. L. G., Guimarães, Cristiano R. W., Azevedo, Hatylas, Couñago, Rafael M.
Published in Journal of medicinal chemistry (13.06.2024)
Published in Journal of medicinal chemistry (13.06.2024)
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