5,6,7,8-Tetrahydro-1,6-naphthyridine Derivatives as Potent HIV-1-Integrase-Allosteric-Site Inhibitors
Peese, Kevin M, Allard, Christopher W, Connolly, Timothy, Johnson, Barry L, Li, Chen, Patel, Manoj, Sorensen, Margaret E, Walker, Michael A, Meanwell, Nicholas A, McAuliffe, Brian, Minassian, Beatrice, Krystal, Mark, Parker, Dawn D, Lewis, Hal A, Kish, Kevin, Zhang, Ping, Nolte, Robert T, Simmermacher, Jean, Jenkins, Susan, Cianci, Christopher, Naidu, B. Narasimhulu
Published in Journal of medicinal chemistry (14.02.2019)
Published in Journal of medicinal chemistry (14.02.2019)
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Design, synthesis and SAR study of novel C2-pyrazolopyrimidine amides and amide isosteres as allosteric integrase inhibitors
Patel, Manoj, Cianci, Christopher, Allard, Christopher W., Parker, Dawn D., Simmermacher, Jean, Jenkins, Susan, Mcauliffe, Brian, Minassian, Beatrice, Discotto, Linda, Krystal, Mark, Meanwell, Nicholas A., Naidu, B. Narasimhulu
Published in Bioorganic & medicinal chemistry letters (01.11.2020)
Published in Bioorganic & medicinal chemistry letters (01.11.2020)
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Discovery of Orally Active Isofuranones as Potent, Selective Inhibitors of Hematopoetic Progenitor Kinase 1
Degnan, Andrew P, Kumi, Godwin K, Allard, Christopher W, Araujo, Erika V, Johnson, Walter L, Zimmermann, Kurt, Pearce, Bradley C, Sheriff, Steven, Futran, Alan, Li, Xin, Locke, Gregory A, You, Dan, Morrison, John, Parrish, Karen E, Stromko, Caitlyn, Murtaza, Anwar, Liu, Jinqi, Johnson, Benjamin M, Vite, Gregory D, Wittman, Mark D
Published in ACS medicinal chemistry letters (11.03.2021)
Published in ACS medicinal chemistry letters (11.03.2021)
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