Controlling opioid receptor functional selectivity by targeting distinct subpockets of the orthosteric site
Uprety, Rajendra, Che, Tao, Zaidi, Saheem A, Grinnell, Steven G, Varga, Balázs R, Faouzi, Abdelfattah, Slocum, Samuel T, Allaoa, Abdullah, Varadi, András, Nelson, Melissa, Bernhard, Sarah M, Kulko, Elizaveta, Le Rouzic, Valerie, Eans, Shainnel O, Simons, Chloe A, Hunkele, Amanda, Subrath, Joan, Pan, Ying Xian, Javitch, Jonathan A, McLaughlin, Jay P, Roth, Bryan L, Pasternak, Gavril W, Katritch, Vsevolod, Majumdar, Susruta
Published in eLife (08.02.2021)
Published in eLife (08.02.2021)
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Journal Article
Oxidative Metabolism as a Modulator of Kratom’s Biological Actions
Chakraborty, Soumen, Uprety, Rajendra, Slocum, Samuel T, Irie, Takeshi, Le Rouzic, Valerie, Li, Xiaohai, Wilson, Lisa L, Scouller, Brittany, Alder, Amy F, Kruegel, Andrew C, Ansonoff, Michael, Varadi, Andras, Eans, Shainnel O, Hunkele, Amanda, Allaoa, Abdullah, Kalra, Sanjay, Xu, Jin, Pan, Ying Xian, Pintar, John, Kivell, Bronwyn M, Pasternak, Gavril W, Cameron, Michael D, McLaughlin, Jay P, Sames, Dalibor, Majumdar, Susruta
Published in Journal of medicinal chemistry (25.11.2021)
Published in Journal of medicinal chemistry (25.11.2021)
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Journal Article
Synthesis and Pharmacology of a Novel μ–δ Opioid Receptor Heteromer-Selective Agonist Based on the Carfentanyl Template
Faouzi, Abdelfattah, Uprety, Rajendra, Gomes, Ivone, Massaly, Nicolas, Keresztes, Attila I, Le Rouzic, Valerie, Gupta, Achla, Zhang, Tiffany, Yoon, Hye Jean, Ansonoff, Michael, Allaoa, Abdullah, Pan, Ying Xian, Pintar, John, Morón, Jose A, Streicher, John M, Devi, Lakshmi A, Majumdar, Susruta
Published in Journal of medicinal chemistry (25.11.2020)
Published in Journal of medicinal chemistry (25.11.2020)
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Journal Article
Synthesis of spiro-2,6-dioxopiperazine and spiro-2,6-dioxopyrazine scaffolds using amino acids in a three-component reaction to generate potential Sigma-1 (σ1) receptor selective ligands
Uprety, Rajendra, Váradi, András, Allaoa, Abdullah, Redel-Traub, Gabriel N., Palmer, Travis C., Feinberg, Evan N., Ferris, Alex C., Pande, Vijay S., Pasternak, Gavril W., Majumdar, Susruta
Published in European journal of medicinal chemistry (15.02.2019)
Published in European journal of medicinal chemistry (15.02.2019)
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Journal Article