Rotational-Echo Double-Resonance NMR Distance Measurements for the Tubulin-Bound Paclitaxel Conformation
Paik, Younkee, Yang, Chao, Metaferia, Belhu, Tang, Shoubin, Bane, Susan, Ravindra, Rudravajhala, Shanker, Natasha, Alcaraz, Ana A, Johnson, Scott A, Schaefer, Jacob, O'Connor, Robert D, Cegelski, Lynette, Snyder, James P, Kingston, David G. I
Published in Journal of the American Chemical Society (17.01.2007)
Published in Journal of the American Chemical Society (17.01.2007)
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Journal Article
Anti-HIV Small-Molecule Binding in the Peptide Subpocket of the CXCR4:CVX15 Crystal Structure
Cox, Bryan D., Prosser, Anthony R., Katzman, Brooke M., Alcaraz, Ana A., Liotta, Dennis C., Wilson, Lawrence J., Snyder, James P.
Published in Chembiochem : a European journal of chemical biology (21.07.2014)
Published in Chembiochem : a European journal of chemical biology (21.07.2014)
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Journal Article
Tetrahydroisoquinoline CXCR4 Antagonists Adopt a Hybrid Binding Mode within the Peptide Subpocket of the CXCR4 Receptor
Katzman, Brooke M, Cox, Bryan D, Prosser, Anthony R, Alcaraz, Ana A, Murat, Brigitte, Héroux, Madeleine, Tebben, Andrew, Zhang, Yong, Schroeder, Gretchen M, Snyder, James P, Wilson, Lawrence J, Liotta, Dennis C
Published in ACS medicinal chemistry letters (10.01.2019)
Published in ACS medicinal chemistry letters (10.01.2019)
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Journal Article
Discovery of Tetrahydroisoquinoline-Based CXCR4 Antagonists
Truax, Valarie M, Zhao, Huanyu, Katzman, Brooke M, Prosser, Anthony R, Alcaraz, Ana A, Saindane, Manohar T, Howard, Randy B, Culver, Deborah, Arrendale, Richard F, Gruddanti, Prahbakar R, Evers, Taylor J, Natchus, Michael G, Snyder, James P, Liotta, Dennis C, Wilson, Lawrence J
Published in ACS medicinal chemistry letters (14.11.2013)
Published in ACS medicinal chemistry letters (14.11.2013)
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Journal Article
The Tubulin-Bound Conformation of Paclitaxel: T-Taxol vs “PTX-NY”
Yang, Yutao, Alcaraz, Ana A, Snyder, James P
Published in Journal of natural products (Washington, D.C.) (27.03.2009)
Published in Journal of natural products (Washington, D.C.) (27.03.2009)
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Journal Article
Dictyostatin Flexibility Bridges Conformations in Solution and in the β-Tubulin Taxane Binding Site
Jogalekar, Ashutosh S, Damodaran, Krishnan, Kriel, Frederik H, Jung, Won-Hyuk, Alcaraz, Ana A, Zhong, Shi, Curran, Dennis P, Snyder, James P
Published in Journal of the American Chemical Society (02.03.2011)
Published in Journal of the American Chemical Society (02.03.2011)
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Journal Article
Evaluation of the Tubulin-Bound Paclitaxel Conformation: Synthesis, Biology, and SAR Studies of C-4 to C-3‘ Bridged Paclitaxel Analogues
Ganesh, Thota, Yang, Chao, Norris, Andrew, Glass, Tom, Bane, Susan, Ravindra, Rudravajhala, Banerjee, Abhijit, Metaferia, Belhu, Thomas, Shala L, Giannakakou, Paraskevi, Alcaraz, Ana A, Lakdawala, Ami S, Snyder, James P, Kingston, David G. I
Published in Journal of medicinal chemistry (22.02.2007)
Published in Journal of medicinal chemistry (22.02.2007)
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Journal Article
The T-Taxol Conformation
Alcaraz, Ana A., Mehta, Anil K., Johnson, Scott A., Snyder, James P.
Published in Journal of medicinal chemistry (20.04.2006)
Published in Journal of medicinal chemistry (20.04.2006)
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Journal Article
Design, synthesis, and bioactivity of simplified paclitaxel analogs based on the T-Taxol bioactive conformation
Ganesh, Thota, Norris, Andrew, Sharma, Shubhada, Bane, Susan, Alcaraz, Ana A., Snyder, James P., Kingston, David G.I.
Published in Bioorganic & medicinal chemistry (15.05.2006)
Published in Bioorganic & medicinal chemistry (15.05.2006)
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Journal Article
The hematopoietic-specific β1-tubulin is naturally resistant to 2-Methoxyestradiol and protects patients from drug-induced myelosuppression
Escuin, Daniel, Burke, Patricia A., McMahon-Tobin, Grainne, Hembrough, Todd, Wang, Yuefang, Alcaraz, Ana A., Leandro-García, Luis Javier, Rodríguez-Rieiro, Cristina, Snyder, James P., LaVallee, Theresa M., Giannakakou, Paraskevi
Published in Cell cycle (Georgetown, Tex.) (01.12.2009)
Published in Cell cycle (Georgetown, Tex.) (01.12.2009)
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Journal Article
Synthesis and bioactivity of a side chain bridged paclitaxel: A test of the T-Taxol conformation
Hodge, Mathis, Chen, Qiao-Hong, Bane, Susan, Sharma, Shubhada, Loew, Maura, Banerjee, Abhijit, Alcaraz, Ana A., Snyder, James P., Kingston, David G.I.
Published in Bioorganic & medicinal chemistry letters (15.05.2009)
Published in Bioorganic & medicinal chemistry letters (15.05.2009)
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Journal Article
Enhanced Microtubule Binding and Tubulin Assembly Properties of Conformationally Constrained Paclitaxel Derivatives
Shanker, Natasha, Kingston, David G. I, Ganesh, Thota, Yang, Chao, Alcaraz, Ana A, Geballe, Matthew T, Banerjee, Abhijit, McGee, Dennis, Snyder, James P, Bane, Susan
Published in Biochemistry (Easton) (16.10.2007)
Published in Biochemistry (Easton) (16.10.2007)
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Journal Article
Synthesis, biological evaluations, and tubulin binding poses of C-2α sulfur linked taxol analogues
Wang, Lei, Alcaraz, Ana A., Matesanz, Ruth, Yang, Chun-Gang, Barasoain, Isabel, Díaz, J. Fernando, Li, Ye-Zhi, Snyder, James P., Fang, Wei-Shuo
Published in Bioorganic & medicinal chemistry letters (01.06.2007)
Published in Bioorganic & medicinal chemistry letters (01.06.2007)
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Journal Article
Synthesis, biological evaluations, and tubulin binding poses of C-2alpha sulfur linked taxol analogues
Wang, Lei, Alcaraz, Ana A, Matesanz, Ruth, Yang, Chun-Gang, Barasoain, Isabel, Díaz, J Fernando, Li, Ye-Zhi, Snyder, James P, Fang, Wei-Shuo
Published in Bioorganic & medicinal chemistry letters (01.06.2007)
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Published in Bioorganic & medicinal chemistry letters (01.06.2007)
Journal Article
REDOR NMR Distance Measurements for the Tubulin-Bound Paclitaxel Conformation
Paik, Younkee, Yang, Chao, Metaferia, Belhu, Tang, Shoubin, Bane, Susan, Ravindra, Rudravajhala, Shanker, Natasha, Alcaraz, Ana A, Johnson, Scott A., Schaefer, Jacob, O'Connor, Robert D., Cegelski, Lynette, Snyder, James P., Kingston, David G. I.
Published in Journal of the American Chemical Society (17.01.2007)
Published in Journal of the American Chemical Society (17.01.2007)
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Journal Article
The hematopoietic-specific beta1-tubulin is naturally resistant to 2-methoxyestradiol and protects patients from drug-induced myelosuppression
Escuin, Daniel, Burke, Patricia A, McMahon-Tobin, Grainne, Hembrough, Todd, Wang, Yuefang, Alcaraz, Ana A, Leandro-García, Luis Javier, Rodríguez-Antona, Cristina, Snyder, James P, Lavallee, Theresa M, Giannakakou, Paraskevi
Published in Cell cycle (Georgetown, Tex.) (01.12.2009)
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Published in Cell cycle (Georgetown, Tex.) (01.12.2009)
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