GABA transporters and GABA-transaminase as drug targets
Sarup, Alan, Larsson, Orla Miller, Schousboe, Arne
Published in Current drug targets. CNS & neurological disorders (01.08.2003)
Published in Current drug targets. CNS & neurological disorders (01.08.2003)
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Journal Article
Role of the betaine/GABA transporter (BGT-1/GAT2) for the control of epilepsy
Schousboe, Arne, Larsson, Orla M., Sarup, Alan, White, H. Steve
Published in European journal of pharmacology (01.10.2004)
Published in European journal of pharmacology (01.10.2004)
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Journal Article
Effects of 3-hydroxy-4-amino-4,5,6,7-tetrahydro-1,2-benzisoxazol (exo-THPO) and its N-substituted analogs on GABA transport in cultured neurons and astrocytes and by the four cloned mouse GABA transporters
Sarup, Alan, Larsson, Orla Miller, Bolvig, Tina, Frølund, Bente, Krogsgaard-Larsen, Povl, Schousboe, Arne
Published in Neurochemistry international (01.09.2003)
Published in Neurochemistry international (01.09.2003)
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Conference Proceeding
GABA transporters as drug targets for modulation of GABAergic activity
Schousboe, Arne, Sarup, Alan, Larsson, Orla M., White, H. Steve
Published in Biochemical pharmacology (15.10.2004)
Published in Biochemical pharmacology (15.10.2004)
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Journal Article
Conference Proceeding
First Demonstration of a Functional Role for Central Nervous System Betaine/γ-Aminobutyric Acid Transporter (mGAT2) Based on Synergistic Anticonvulsant Action among Inhibitors of mGAT1 and mGAT2
White, H. Steve, Watson, William P., Hansen, Suzanne L., Slough, Scott, Perregaard, Jens, Sarup, Alan, Bolvig, Tina, Petersen, Gitte, Larsson, Orla M., Clausen, Rasmus P., Frølund, Bente, Falch, Erik, Krogsgaard-Larsen, Povl, Schousboe, Arne
Published in The Journal of pharmacology and experimental therapeutics (01.02.2005)
Published in The Journal of pharmacology and experimental therapeutics (01.02.2005)
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Journal Article
Selective inhibitors of GABA uptake: synthesis and molecular pharmacology of 4- N-methylamino-4,5,6,7-tetrahydrobenzo[ d]isoxazol-3-ol analogues
Clausen, Rasmus P., Moltzen, Ejner K., Perregaard, Jens, Lenz, Sibylle M., Sanchez, Connie, Falch, Erik, Frølund, Bente, Bolvig, Tina, Sarup, Alan, Larsson, Orla M., Schousboe, Arne, Krogsgaard-Larsen, Povl
Published in Bioorganic & medicinal chemistry (01.02.2005)
Published in Bioorganic & medicinal chemistry (01.02.2005)
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Correlation between anticonvulsant activity and inhibitory action on glial gamma-aminobutyric acid uptake of the highly selective mouse gamma-aminobutyric acid transporter 1 inhibitor 3-hydroxy-4-amino-4,5,6,7-tetrahydro-1,2-benzisoxazole and its N-alkylated analogs
White, H Steve, Sarup, Alan, Bolvig, Tina, Kristensen, Anders S, Petersen, Gitte, Nelson, Nathan, Pickering, Darryl S, Larsson, Orla M, Frølund, Bente, Krogsgaard-Larsen, Povl, Schousboe, Arne
Published in The Journal of pharmacology and experimental therapeutics (01.08.2002)
Published in The Journal of pharmacology and experimental therapeutics (01.08.2002)
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Journal Article
First Demonstration of a Functional Role for Central Nervous System Betaine/γ-Aminobutyric Acid Transporter (mGAT2) Based on Synergistic Anticonvulsant Action among Inhibitors of mGAT1 and mGAT2
H. Steve White, William P. Watson, Suzanne L. Hansen, Scott Slough, Jens Perregaard, Alan Sarup, Tina Bolvig, Gitte Petersen, Orla M. Larsson, Rasmus P. Clausen, Bente Frølund, Erik Falch, Povl Krogsgaard-Larsen, Arne Schousboe
Published in The Journal of pharmacology and experimental therapeutics (01.02.2005)
Published in The Journal of pharmacology and experimental therapeutics (01.02.2005)
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Journal Article
First demonstration of a functional role for central nervous system betaine/{gamma}-aminobutyric acid transporter (mGAT2) based on synergistic anticonvulsant action among inhibitors of mGAT1 and mGAT2
White, H Steve, Watson, William P, Hansen, Suzanne L, Slough, Scott, Perregaard, Jens, Sarup, Alan, Bolvig, Tina, Petersen, Gitte, Larsson, Orla M, Clausen, Rasmus P, Frølund, Bente, Falch, Erik, Krogsgaard-Larsen, Povl, Schousboe, Arne
Published in The Journal of pharmacology and experimental therapeutics (01.02.2005)
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Published in The Journal of pharmacology and experimental therapeutics (01.02.2005)
Journal Article
Correlation between Anticonvulsant Activity and Inhibitory Action on Glial γ-Aminobutyric Acid Uptake of the Highly Selective Mouse γ-Aminobutyric Acid Transporter 1 Inhibitor 3-Hydroxy-4-amino-4,5,6,7-tetrahydro-1,2-benzisoxazole and ItsN-Alkylated Analogs
H. Steve White, Alan Sarup, Tina Bolvig, Anders S. Kristensen, Gitte Petersen, Nathan Nelson, Darryl S. Pickering, Orla M. Larsson, Bente Frølund, Povl Krogsgaard-Larsen, Arne Schousboe
Published in The Journal of pharmacology and experimental therapeutics (01.08.2002)
Published in The Journal of pharmacology and experimental therapeutics (01.08.2002)
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Journal Article