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Bari, Ahmed, Grenier, Daniel, Azelmat, Jabrane, Syed, Saeed Ali, Al‐Obaid, Abdulrahman M., Hosten, Eric C.
Published in Chemical biology & drug design (01.10.2019)
Published in Chemical biology & drug design (01.10.2019)
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Synthesis, potential antitumor activity, cell cycle analysis, and multitarget mechanisms of novel hydrazones incorporating a 4-methylsulfonylbenzene scaffold: a molecular docking study
Abdel-Aziz, Alaa A.-M., El-Azab, Adel S., AlSaif, Nawaf A., Obaidullah, Ahmad J., Al-Obaid, Abdulrahman M., Al-Suwaidan, Ibrahim A.
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2021)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2021)
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Synthesis, anticancer and apoptosis-inducing activities of quinazoline-isatin conjugates: epidermal growth factor receptor-tyrosine kinase assay and molecular docking studies
El-Azab, Adel S., Al-Dhfyan, Abdullah, Abdel-Aziz, Alaa A.-M., Abou-Zeid, Laila A., Alkahtani, Hamad M., Al-Obaid, Abdulrahman M., Al-Gendy, Manal A.
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2017)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2017)
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Molecular design, synthesis and biological evaluation of cyclic imides bearing benzenesulfonamide fragment as potential COX-2 inhibitors. Part 2
Al-Suwaidan, Ibrahim A., Alanazi, Amer M., El-Azab, Adel S., Al-Obaid, Abdulrahman M., ElTahir, Kamal E.H., Maarouf, Azza R., Abu El-Enin, Mohamed A., Abdel-Aziz, Alaa A.-M.
Published in Bioorganic & medicinal chemistry letters (01.05.2013)
Published in Bioorganic & medicinal chemistry letters (01.05.2013)
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LC–MS/MS method for the quantitation of decitabine and venetoclax in rat plasma after SPE: Application to pharmacokinetic study
Alnasser, Abdulaziz I., Hefnawy, Mohamed M., Al-Hossaini, Abdullah M., Bin Jardan, Yousef A., El-Azab, Adel S., Abdel-Aziz, Alaa M., Al-Obaid, Abdulrahman M., Al-Suwaidan, Ibrahim A., Attwa, Mohamed W., El-Gendy, Manal A.
Published in Saudi pharmaceutical journal (01.09.2023)
Published in Saudi pharmaceutical journal (01.09.2023)
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Synthesis, dihydrofolate reductase inhibition, antitumor testing, and molecular modeling study of some new 4(3 H)-quinazolinone analogs
Al-Rashood, Sarah T., Aboldahab, Ihsan A., Nagi, Mahmoud N., Abouzeid, Laila A., Abdel-Aziz, Alaa A.M., Abdel-hamide, Sami G., Youssef, Khairia M., Al-Obaid, Abdulrahman M., El-Subbagh, Hussein I.
Published in Bioorganic & medicinal chemistry (15.12.2006)
Published in Bioorganic & medicinal chemistry (15.12.2006)
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Synthesis and biological evaluation of some novel cyclic-imides as hypoglycaemic, anti-hyperlipidemic agents
Abdel-Aziz, Alaa A.-M., El-Azab, Adel S., Attia, Sabry M., Al-Obaid, Abdulrahman M., Al-Omar, Mohamed A., El-Subbagh, Hussein I.
Published in European journal of medicinal chemistry (01.09.2011)
Published in European journal of medicinal chemistry (01.09.2011)
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Synthesis of Bivalent Ni(II), Cu(II) and Zn(II) Complexes of Azodicarbonamide in Mixture of Methanol and Aqueous Solvents: Spectral Characterizations and Anti-Microbial Studies
Younes, Ayman A. O., Adam, Abdel Majid A., Refat, Moamen S., Al-Wasidi, Asma S., Almehizia, Abdulrahman A., Al-Omar, Mohamed A., Naglah, Ahmed M., Al-Obaid, Abdulrahman M., Alkahtani, Hamad M., Obaidullah, Ahmad J., El-Sayed, Mohamed Y., Asla, Kareem A.
Published in Crystals (Basel) (01.03.2023)
Published in Crystals (Basel) (01.03.2023)
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Non-classical antifolates. Part 2: Synthesis, biological evaluation, and molecular modeling study of some new 2,6-substituted-quinazolin-4-ones
Al-Omary, Fatmah A.M., Abou-zeid, Laila A., Nagi, Mahmoud N., Habib, El-Sayed E., Abdel-Aziz, Alaa A.-M., El-Azab, Adel S., Abdel-Hamide, Sami G., Al-Omar, Mohamed A., Al-Obaid, Abdulrahman M., El-Subbagh, Hussein I.
Published in Bioorganic & medicinal chemistry (15.04.2010)
Published in Bioorganic & medicinal chemistry (15.04.2010)
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Synthesis of orotic acid derivatives and their effects on stem cell proliferation
Syed, Saeed Ali, Mahmood, Amer, Alfayez, Musaad, Hosten, Eric C., Betz, Richard, Al-Obaid, Abdulrahman M., Ghadeer, Abdulrahman, Bari, Ahmed
Published in Open Chemistry (01.01.2020)
Published in Open Chemistry (01.01.2020)
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Synthesis, enzyme inhibition assay, and molecular modeling study of novel pyrazolines linked to 4-methylsulfonylphenyl scaffold: antitumor activity and cell cycle analysis
Abdel-Aziz, Alaa A.-M, El-Azab, Adel S, Brogi, Simone, Ayyad, Rezk R, Alkahtani, Hamad M, Abuelizz, Hatem A, Al-Suwaidan, Ibrahim A, Al-Obaid, Abdulrahman M
Published in RSC advances (12.07.2024)
Published in RSC advances (12.07.2024)
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Synthesis, anti-inflammatory, analgesic and COX-1/2 inhibition activities of anilides based on 5,5-diphenylimidazolidine-2,4-dione scaffold: Molecular docking studies
Abdel-Aziz, Alaa A.-M., El-Azab, Adel S., Abou-Zeid, Laila A., ElTahir, Kamal Eldin H., Abdel-Aziz, Naglaa I., Ayyad, Rezk R., Al-Obaid, Abdulrahman M.
Published in European journal of medicinal chemistry (10.06.2016)
Published in European journal of medicinal chemistry (10.06.2016)
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Synthesis of new peptide-based macrocycles: Evaluation of their in vitro anti-proliferative activity and molecular dynamic simulation studies
O. Moustafa, Gaber, A. Almehizia, Abdulrahman, A. Al-Omar, Mohamed, M. Al-Obaid, Abdulrahman, M. Naglah, Ahmed, A. Zen, Amer
Published in Bulletin of the Chemical Society of Ethiopia (01.01.2024)
Published in Bulletin of the Chemical Society of Ethiopia (01.01.2024)
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Synthesis, anticonvulsant activity and molecular modeling study of some new hydrazinecarbothioamide, benzenesulfonohydrazide, and phenacylacetohydrazide analogues of 4(3H)-quinazolinone
Al-Salem, Huda S.A., Hegazy, Gehan H., El-Taher, Kamal E.H., El-Messery, Shahenda M., Al-Obaid, Abdulrahman M., El-Subbagh, Hussein I.
Published in Bioorganic & medicinal chemistry letters (01.04.2015)
Published in Bioorganic & medicinal chemistry letters (01.04.2015)
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Synthesis, antitumor and antimicrobial activity of some new 6-methyl-3-phenyl-4(3H)-quinazolinone analogues: in silico studies
Alanazi, Amer M., Abdel-Aziz, Alaa A.-M., Shawer, Taghreed Z., Ayyad, Rezk R., Al-Obaid, Abdulrahman M., Al-Agamy, Mohamed H. M., Maarouf, Azza R., El-Azab, Adel S.
Published in Journal of enzyme inhibition and medicinal chemistry (02.09.2016)
Published in Journal of enzyme inhibition and medicinal chemistry (02.09.2016)
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Substituted Quinazolines, Part 2. Synthesis and In-Vitro Anticancer Evaluation of New 2-Substituted Mercapto-3H-quinazoline Analogs
Khalil, Ashraf A., Hamide, Sami G. Abdel, Al-Obaid, Abdulrahman M., El-Subbagh, Hussein I.
Published in Archiv der Pharmazie (Weinheim) (01.04.2003)
Published in Archiv der Pharmazie (Weinheim) (01.04.2003)
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Design, synthesis, single-crystal and preliminary antitumor activity of novel arenesulfonylimidazolidin-2-ones
Abdel-Aziz, Alaa A.-M., El-Azab, Adel S., El-Subbagh, Hussein I., Al-Obaid, Abdulrahman M., Alanazi, Amer M., Al-Omar, Mohamed A.
Published in Bioorganic & medicinal chemistry letters (01.03.2012)
Published in Bioorganic & medicinal chemistry letters (01.03.2012)
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Synthesis and anticonvulsant activity of some new thiazolo[3,2-a][1,3]diazepine, benzo[d]thiazolo[5,2-a][12,6]diazepine and benzo[d]oxazolo[5,2-a][12,6]diazepine analogues
El-Subbagh, Hussein I., Hassan, Ghada S., El-Azab, Adel S., Abdel-Aziz, Alaa A.-M., Kadi, Adnan A., Al-Obaid, Abdulrahman M., Al-Shabanah, Othman A., Sayed-Ahmed, Mohamed M.
Published in European journal of medicinal chemistry (01.11.2011)
Published in European journal of medicinal chemistry (01.11.2011)
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