Identification of the First "Two Digit Nano-molar" Inhibitors of the Human Glyoxalase-I Enzyme as Potential Anticancer Agents
Al-Balas, Qosay A, Al-Sha'er, Mahmoud A, Hassan, Mohammad A, Al Zou'bi, Esra'a
Published in Medicinal chemistry (Shp-sariqah, United Arab Emirates) (01.01.2022)
Published in Medicinal chemistry (Shp-sariqah, United Arab Emirates) (01.01.2022)
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Journal Article
Computational and experimental exploration of the structure–activity relationships of flavonoids as potent glyoxalase‐I inhibitors
Al‐Balas, Qosay A., Hassan, Mohammad A., Al‐Shar'i, Nizar A., El‐Elimat, Tamam, Almaaytah, Ammar M.
Published in Drug development research (01.03.2018)
Published in Drug development research (01.03.2018)
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Journal Article
Computational fragment-based drug design of potential Glo-I inhibitors
Bibars, Roaa S, Al-Balas, Qosay A
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2024)
Published in Journal of enzyme inhibition and medicinal chemistry (01.12.2024)
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Journal Article
Design, synthesis and biological evaluation of novel glyoxalase I inhibitors possessing diazenylbenzenesulfonamide moiety as potential anticancer agents
Al-Oudat, Buthina A., Jaradat, Hana'a M., Al‑Balas, Qosay A., Al-Shar'i, Nizar A., Bryant-Friedrich, Amanda, Bedi, Mel F.
Published in Bioorganic & medicinal chemistry (15.08.2020)
Published in Bioorganic & medicinal chemistry (15.08.2020)
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Journal Article
Recent Advances in Glyoxalase-I Inhibition
Al-Balas, Qosay A, Hassan, Mohammad A, Al-Shar'i, Nizar A, Al Jabal, Ghazi A, Almaaytah, Ammar M
Published in Mini reviews in medicinal chemistry (01.01.2019)
Published in Mini reviews in medicinal chemistry (01.01.2019)
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Multi-Armed 1,2,3-Selenadiazole and 1,2,3-Thiadiazole Benzene Derivatives as Novel Glyoxalase-I Inhibitors
Al-Balas, Qosay A, Al-Smadi, Mousa L, Hassan, Mohammad A, Al Jabal, Ghazi A, Almaaytah, Ammar M, Alzoubi, Karem H
Published in Molecules (Basel, Switzerland) (04.09.2019)
Published in Molecules (Basel, Switzerland) (04.09.2019)
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Journal Article
Ellagic acid: A potent glyoxalase-I inhibitor with a unique scaffold
Al-Shar’i, Nizar A., Al-Balas, Qosay A., Hassan, Mohammad A., El-Elimat, Tamam M., Aljabal, Ghazi A., Almaaytah, Ammar M.
Published in Acta Pharmaceutica (01.03.2021)
Published in Acta Pharmaceutica (01.03.2021)
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Identification of Human Leukotriene A4 Hydrolase Inhibitors Using Structure-Based Pharmacophore Modeling and Molecular Docking
Audat, Suaad A, Al-Shar'i, Nizar A, Al-Oudat, Buthina A, Bryant-Friedrich, Amanda, Bedi, Mel F, Zayed, Aref L, Al-Balas, Qosay A
Published in Molecules (Basel, Switzerland) (22.06.2020)
Published in Molecules (Basel, Switzerland) (22.06.2020)
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Lead optimization and biological evaluation of diazenylbenzenesulfonamides inhibitors against glyoxalase-I enzyme as potential anticancer agents
Al-Oudat, Buthina A., Al-Shar'i, Nizar A., Al‑Balas, Qosay A., Audat, Suaad A., Alqudah, Mohammad A.Y., Hamzah, Ali H., Hallak, Ramez W., Bedi, Mel, Bryant-Friedrich, Amanda
Published in Bioorganic chemistry (01.03.2022)
Published in Bioorganic chemistry (01.03.2022)
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Journal Article
Virtual lead identification of farnesyltransferase inhibitors based on ligand and structure-based pharmacophore techniques
Al-Balas, Qosay A, Amawi, Haneen A, Hassan, Mohammad A, Qandil, Amjad M, Almaaytah, Ammar M, Mhaidat, Nizar M
Published in Pharmaceuticals (Basel, Switzerland) (27.05.2013)
Published in Pharmaceuticals (Basel, Switzerland) (27.05.2013)
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Synthesis, Antibacterial Evaluation and QSAR of α-Substituted-N₄-Acetamides of Ciprofloxacin and Norfloxacin
Qandil, Amjad M, Al-Zoubi, Lorca O, Al-Bakri, Amal G, Amawi, Haneen A, Al-Balas, Qosay A, Alkatheri, Abdulmalik M, Albekairy, Abdulkareem M
Published in Antibiotics (Basel) (25.06.2014)
Published in Antibiotics (Basel) (25.06.2014)
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