Discovery of a Clinical Stage Multi-Kinase Inhibitor Sodium (E)-2-{2-Methoxy-5-[(2′,4′,6′-trimethoxystyrylsulfonyl)methyl]phenylamino}acetate (ON 01910.Na): Synthesis, Structure–Activity Relationship, and Biological Activity
Reddy, M. V. Ramana, Venkatapuram, Padmavathi, Mallireddigari, Muralidhar R, Pallela, Venkat R, Cosenza, Stephen C, Robell, Kimberly A, Akula, Balaiah, Hoffman, Benjamin S, Reddy, E. Premkumar
Published in Journal of medicinal chemistry (22.09.2011)
Published in Journal of medicinal chemistry (22.09.2011)
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Glycogen Synthase Kinase-3 (GSK-3) Inhibitory Activity and Structure–Activity Relationship (SAR) Studies of the Manzamine Alkaloids. Potential for Alzheimer’s Disease
Hamann, Mark, Alonso, Diana, Martín-Aparicio, Ester, Fuertes, Ana, Pérez-Puerto, M. José, Castro, Ana, Morales, Susana, Navarro, María Luisa, del Monte-Millán, María, Medina, Miguel, Pennaka, Hari, Balaiah, Akula, Peng, Jiangnan, Cook, Jennifer, Wahyuono, Subagus, Martínez, Ana
Published in Journal of natural products (Washington, D.C.) (01.09.2007)
Published in Journal of natural products (Washington, D.C.) (01.09.2007)
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Modulation of Physical Properties of Ter(9,9-ditolylfluorene) by Backbone-Embedded Heteroarenes
Wong, Ken-Tsung, Hwu, Tsyr-Yuan, Balaiah, Akula, Chao, Teng-Chih, Fang, Fu-Chuan, Lee, Ching-Tien, Peng, Ying-Chu
Published in Organic letters (30.03.2006)
Published in Organic letters (30.03.2006)
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Synthesis of Some Fused Pyrazoles and Isoxazoles
Padmavathi, Venkatapuram, Reddy, Boggu Jagan Mohan, Balaiah, Akula, Reddy, Katta Venugopal, Reddy, Dandu Bhaskar
Published in MolBank (01.12.2000)
Published in MolBank (01.12.2000)
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Syntheses and Structures of Novel Heteroarene-Fused Coplanar π-Conjugated Chromophores
Wong, Ken-Tsung, Chao, Teng-Chih, Chi, Liang-Chen, Chu, Ying-Ying, Balaiah, Akula, Chiu, Shih-Feng, Liu, Yi-Hung, Wang, Yu
Published in Organic letters (26.10.2006)
Published in Organic letters (26.10.2006)
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(Z)-1-Aryl-3-arylamino-2-propen-1-ones, Highly Active Stimulators of Tubulin Polymerization: Synthesis, Structure–Activity Relationship (SAR), Tubulin Polymerization, and Cell Growth Inhibition Studies
Reddy, M. V. Ramana, Akula, Balaiah, Cosenza, Stephen C, Lee, Clement M, Mallireddigari, Muralidhar R, Pallela, Venkat R, Subbaiah, D. R. C. Venkata, Udofa, Andrew, Reddy, E. Premkumar
Published in Journal of medicinal chemistry (14.06.2012)
Published in Journal of medicinal chemistry (14.06.2012)
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Abstract 4519: Targeting of cyclin D/Rb/E2F and PI3K/AKT/MTOR pathways with ON 123300 as a therapeutic strategy for mantle cell lymphoma
Reddy, E. Premkumar, Divakar, Saikrishna A., Reddy, M.V. Ramana, Cosenza, Stephen C., Baker, Stacey J., Akula, Balaiah, Parekh, Samir
Published in Cancer research (Chicago, Ill.) (01.10.2014)
Published in Cancer research (Chicago, Ill.) (01.10.2014)
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Dual inhibition of CDK4/Rb and PI3K/AKT/mTOR pathways by ON123300 induces synthetic lethality in mantle cell lymphomas
Divakar, S K A, Ramana Reddy, M V, Cosenza, S C, Baker, S J, Perumal, D, Antonelli, A C, Brody, J, Akula, B, Parekh, S, Reddy, E Premkumar
Published in Leukemia (01.01.2016)
Published in Leukemia (01.01.2016)
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Hydrothiolation of benzyl mercaptan to arylacetylene: application to the synthesis of (E) and (Z)-isomers of ON 01910 center dot Na (Rigosertib (R)), a phase III clinical stage anti-cancer agent
Pallela, Venkat R., Mallireddigari, Muralidhar R., Cosenza, Stephen C., Akula, Balaiah, Subbaiah, D. R. C. Venkata, Reddy, E. Premkumar, Reddy, M. V. Ramana
Published in Organic & biomolecular chemistry (01.01.2013)
Published in Organic & biomolecular chemistry (01.01.2013)
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Journal Article
Design, Synthesis, and Biological Evaluation of (E)‑N‑Aryl-2-arylethenesulfonamide Analogues as Potent and Orally Bioavailable Microtubule-Targeted Anticancer Agents
Reddy, M. V. Ramana, Mallireddigari, Muralidhar R, Pallela, Venkat R, Cosenza, Stephen C, Billa, Vinay K, Akula, Balaiah, Subbaiah, D. R. C. Venkata, Bharathi, E. Vijaya, Padgaonkar, Amol, Lv, Hua, Gallo, James M, Reddy, E. Premkumar
Published in Journal of medicinal chemistry (11.07.2013)
Published in Journal of medicinal chemistry (11.07.2013)
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Hydrothiolation of benzyl mercaptan to arylacetylene: application to the synthesis of (E) and (Z)-isomers of ON 01910·Na (Rigosertib®), a phase III clinical stage anti-cancer agent
Pallela, Venkat R, Mallireddigari, Muralidhar R, Cosenza, Stephen C, Akula, Balaiah, Subbaiah, D R C Venkata, Reddy, E Premkumar, Reddy, M V Ramana
Published in Organic & biomolecular chemistry (28.03.2013)
Published in Organic & biomolecular chemistry (28.03.2013)
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Design, Synthesis and Biological Evaluation of (E)-N-Aryl-2-arylethene-sulfonamide Analogues as Potent and Orally Bioavailable Microtubule-targeted Anticancer Agents
Ramana Reddy, M. V., Mallireddigari, Muralidhar R., Pallela, Venkat R., Cosenza, Stephen C., Billa, Vinay K., Akula, Balaiah, Venkata Subbaiah, D. R. C., Bharathi, E. Vijaya, Padgaonkar, Amol, Lv, Hua, Gallo, James M., Reddy, E. Premkumar
Published in Journal of medicinal chemistry (25.06.2013)
Published in Journal of medicinal chemistry (25.06.2013)
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Hydrothiolation of benzyl mercaptan to arylacetylene: application to the synthesis of (E) and (Z)-isomers of ON 01910·Na (Rigosertib®), a phase III clinical stage anti-cancer agentElectronic supplementary information (ESI) available: 1H and 13C NMR spectra of all new compounds. See DOI: 10.1039/c3ob27220f
Pallela, Venkat R, Mallireddigari, Muralidhar R, Cosenza, Stephen C, Akula, Balaiah, Subbaiah, D. R. C. Venkata, Reddy, E. Premkumar, Reddy, M. V. Ramana
Year of Publication 27.02.2013
Year of Publication 27.02.2013
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Design, synthesis and evaluation of ( E)-α-benzylthio chalcones as novel inhibitors of BCR-ABL kinase
Reddy, M.V. Ramana, Pallela, Venkat R., Cosenza, Stephen C., Mallireddigari, Muralidhar R., Patti, Revathi, Bonagura, Marie, Truongcao, May, Akula, Balaiah, Jatiani, Shashidhar S., Reddy, E. Premkumar
Published in Bioorganic & medicinal chemistry (15.03.2010)
Published in Bioorganic & medicinal chemistry (15.03.2010)
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Syntheses and Structures of Novel Heteroarene-Fused Coplanar π-Conjugated Chromophores
Wong, Ken-Tsung, Chao, Teng-Chih, Chi, Liang-Chen, Chu, Ying-Ying, Balaiah, Akula, Chiu, Shih-Feng, Liu, Yi-Hung, Wang, Yu
Published in ChemInform (20.02.2007)
Published in ChemInform (20.02.2007)
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Journal Article
Fluorine derivatives with thiophene moiety and method for forming the same
FANG, FU CHUAN, CHU, YING YING, CHAO, TENG CHIH, LEE, CHING TIEN, WONG, KEN TSUNG, AKULA BALAIAH, CHIU, SHIH FENG
Year of Publication 11.09.2009
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Year of Publication 11.09.2009
Patent
Fluorene derivatives with thiophene moiety and method for forming the same
CHU, YING YING, FANG, FUUAN, LEE, CHING-TIEN, BALAIAH, AKULA, CHAO, TENGIH, WONG, KEN-TSUNG, CHIU, SHIH FENG
Year of Publication 01.12.2007
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Year of Publication 01.12.2007
Patent