Discovery of GLPG2737, a Potent Type 2 Corrector of CFTR for the Treatment of Cystic Fibrosis in Combination with a Potentiator and a Type 1 Co-corrector
Pizzonero, Mathieu, Akkari, Rhalid, Bock, Xavier, Gosmini, Romain, De Lemos, Elsa, Duthion, Béranger, Newsome, Gregory, Mai, Thi-Thu-Trang, Roques, Virginie, Jary, Hélène, Lefrancois, Jean-Michel, Cherel, Laetitia, Quenehen, Vanessa, Babel, Marielle, Merayo, Nuria, Bienvenu, Natacha, Mammoliti, Oscar, Coti, Ghjuvanni, Palisse, Adeline, Cowart, Marlon, Shrestha, Anurupa, Greszler, Stephen, Van Der Plas, Steven, Jansen, Koen, Claes, Pieter, Jans, Mia, Gees, Maarten, Borgonovi, Monica, De Wilde, Gert, Conrath, Katja
Published in Journal of medicinal chemistry (11.04.2024)
Published in Journal of medicinal chemistry (11.04.2024)
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Decoding signaling and function of the orphan G protein-coupled receptor GPR17 with a small-molecule agonist
Hennen, Stephanie, Wang, Haibo, Peters, Lucas, Merten, Nicole, Simon, Katharina, Spinrath, Andreas, Blättermann, Stefanie, Akkari, Rhalid, Schrage, Ramona, Schröder, Ralf, Schulz, Daniel, Vermeiren, Celine, Zimmermann, Katrin, Kehraus, Stefan, Drewke, Christel, Pfeifer, Alexander, König, Gabriele M, Mohr, Klaus, Gillard, Michel, Müller, Christa E, Lu, Q Richard, Gomeza, Jesus, Kostenis, Evi
Published in Science signaling (22.10.2013)
Published in Science signaling (22.10.2013)
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3-(2-Carboxyethyl)indole-2-carboxylic Acid Derivatives: Structural Requirements and Properties of Potent Agonists of the Orphan G Protein-Coupled Receptor GPR17
Baqi, Younis, Pillaiyar, Thanigaimalai, Abdelrahman, Aliaa, Kaufmann, Olesja, Alshaibani, Samer, Rafehi, Muhammad, Ghasimi, Saman, Akkari, Rhalid, Ritter, Kirsten, Simon, Katharina, Spinrath, Andreas, Kostenis, Evi, Zhao, Qiang, Köse, Meryem, Namasivayam, Vigneshwaran, Müller, Christa E
Published in Journal of medicinal chemistry (27.09.2018)
Published in Journal of medicinal chemistry (27.09.2018)
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염증성 질환의 치료를 위한 신규 화합물 및 그의 약학 조성물
JARY HELENE MARIE, AKKARI RHALID, BRYS REGINALD CHRISTOPHE XAVIER, KOMAC MARIJANA, ORSULIC MISLAV, MAMMOLITI OSCAR, VRBAN DENANA
Year of Publication 01.12.2021
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Year of Publication 01.12.2021
Patent
1,3-Dialkyl-substituted tetrahydropyrimido[1,2-f]purine-2,4-diones as multiple target drugs for the potential treatment of neurodegenerative diseases
Koch, Pierre, Akkari, Rhalid, Brunschweiger, Andreas, Borrmann, Thomas, Schlenk, Miriam, Küppers, Petra, Köse, Meryem, Radjainia, Hamid, Hockemeyer, Jörg, Drabczyńska, Anna, Kieć-Kononowicz, Katarzyna, Müller, Christa E.
Published in Bioorganic & medicinal chemistry (01.12.2013)
Published in Bioorganic & medicinal chemistry (01.12.2013)
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Abstract 4748: Discovery of JNJ-42756493, a potent fibroblast growth factor receptor (FGFR) inhibitor using a fragment based approach
Angibaud, Patrick R., Mevellec, Laurence, Saxty, Gordon, Adelinet, Christophe, Akkari, Rhalid, Berdini, Valerio, Bonnet, Pascal, Bourgeois, Marine, Bourdrez, Xavier, Cleasby, Anne, Colombel, Helene, Csoka, Imre, Embrechts, Werner, Freyne, Eddy, Gilissen, Ronaldus, Jovcheva, Eleonora, King, Peter, Lacrampe, Jean, Lardeau, Delphine, Ligny, Yannick, Mcclue, Steve, Meerpoel, Lieven, Newell, David R., Page, Martin, Papanikos, Alexandra, Pasquier, Elisabeth, Pilatte, Isabelle, Poncelet, Virginie, Querolle, Olivier, Rees, David C., Rich, Sharna, Roux, Bruno, Sement, Elodie, Simonnet, Yvan, Squires, Matthew, Tronel, Virginie, Verhulst, Tinne, Vialard, Jorge, Willems, Marc, Woodhead, Steven J., Wroblowski, Berthold, Murray, Christopher W., Perera, Timothy
Published in Cancer research (Chicago, Ill.) (01.10.2014)
Published in Cancer research (Chicago, Ill.) (01.10.2014)
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PYRAZOLYL QUINOXALINE KINASE INHIBITORS
FREYNE EDDY JEAN EDGARD, PAPANIKOS ALEXANDRA, AKKARI RHALID, MEERPOEL LIEVEN, ANGIBAUD PATRICK RENE, EMBRECHTS WERNER CONSTANT JOHAN, LACRAMPE JEAN FERNAND ARMAND, BERDINI VALERIO, WROBLOWSKI BERTHOLD, SAXTY GORDON, WOODHEAD STEVEN JOHN, HAMLETT CHRISTOPHER CHARLES FREDERICK, MEVELLEC LAURENCE ANNE, BESONG GILBERT EBAI, WEERTS JOHAN ERWIN EDMOND, QUEROLLE OLIVIER ALEXIS GEORGES, JOHNSON CHRISTOPHER NORBERT, PASQUIER ELISABETH THERESE JEANNE, GOVAERTS TOM CORNELIS HORTENSE, REES DAVID CHARLES, BONNET PASCAL GHISLAIN ANDRE, PILATTE ISABELLE NOELLE CONSTANCE, PERERA TIMOTHY PIETRO SUREN, READER MICHAEL, URRAY CHRISTOPHER WILLIAM, GILISSEN RONALDUS ARNODUS HENDRIKA JOSEPH
Year of Publication 20.08.2018
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Year of Publication 20.08.2018
Patent
N-설포닐화 피라졸로[3,4-b]피리딘-6-카복스아미드 및 사용 방법
AKKARI RHALID, BROWN BRIAN S, BOCK XAVIER MARIE, HOUSSEMAN CHRISTOPHER GAETAN, PATEL SACHIN V, JI JIANGUO, DE BLIECK ANN, KYM PHILIP R, SHRESTHA ANURUPA, WANG XUEQING, GFESSER GREGORY A, SWIFT ELIZABETH C, ALVEY LUKE JONATHAN, PALISSE ADELINE MARIE ELISE, NEWSOME GREGORY JOHN ROBERT, PIZZONERO MATHIEU RAFAEL, DESROY NICOLAS, MERAYO NURIA MERAYO, CLAES PIETER ISABELLE ROGER, GOSMINI ROMAIN LUC MARIE, DUTHION BERANGER, MENET CHRISTEL JEANNE MARIE, DE LEMOS ELSA, LEFRANCOIS JEAN MICHEL, MAMMOLITI OSCAR, VAN DER PLAS STEVEN EMIEL, JANSEN KOEN KAREL, COWART MARLON D
Year of Publication 20.07.2018
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Year of Publication 20.07.2018
Patent
Asymmetric Baylis–Hillman reactions using ( R)-4-(3-hydroxy-4,4-dimethyl-2-oxopyrrolidin-1-yl) benzoic acid acrylate derivatives in solution and on solid support
Calmès, Monique, Akkari, Rhalid, Barthes, Nicolas, Escale, Françoise, Martinez, Jean
Published in Tetrahedron: asymmetry (20.06.2005)
Published in Tetrahedron: asymmetry (20.06.2005)
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( R)- or ( S)-4-(3-hydroxy-4,4-dimethyl-2-oxopyrrolidin-1-yl)benzoic acid as a new chiral auxiliary for solid phase asymmetric Diels–Alder reactions
Akkari, Rhalid, Calmès, Monique, Escale, Françoise, Iapichella, Julien, Rolland, Marc, Martinez, Jean
Published in Tetrahedron: asymmetry (23.08.2004)
Published in Tetrahedron: asymmetry (23.08.2004)
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Journal Article
PYRAZOLYL QUINAZOLINE KINASE INHIBITORS
FREYNE EDDY JEAN EDGARD, PAPANIKOS ALEXANDRA, AKKARI RHALID, MEERPOEL LIEVEN, ANGIBAUD PATRICK RENE, EMBRECHTS WERNER CONSTANT JOHAN, LACRAMPE JEAN FERNAND ARMAND, MURRAY CHRISTOPHER WILLIAM, BERDINI VALERIO, WROBLOWSKI BERTHOLD, SAXTY GORDON, WOODHEAD STEVEN JOHN, HAMLETT CHRISTOPHER CHARLES FREDERICK, MEVELLEC LAURENCE ANNE, BESONG GILBERT EBAI, WEERTS JOHAN ERWIN EDMOND, QUEROLLE OLIVER ALEXIS GEORGES, JOHNSON CHRISTOPHER NORBERT, PASQUIER ELISABETH THERESE JEANNE, GOVAERTS TOM CORNELIS HORTENSE, REES DAVID CHARLES, BONNET PASCAL GHISLAIN ANDRE, PILATTE ISABELLE NOELLE CONSTANCE, PERERA TIMOTHY PIETRO SUREN, READER MICHAEL, GILISSEN RONALDUS ARNODUS HENDRIKA JOSEPH
Year of Publication 02.10.2013
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Year of Publication 02.10.2013
Patent
(S)-(3-Hydroxy-4,4-dimethyl-2-oxopyrrolidin-1-yl) acetic acid as a solid supported chiral auxiliary in the asymmetric synthesis of β2-homoarylglycines
Akkari, Rhalid, Calmès, Monique, Di Malta, Delphine, Escale, Françoise, Martinez, Jean
Published in Tetrahedron: asymmetry (01.05.2003)
Published in Tetrahedron: asymmetry (01.05.2003)
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Journal Article
( S)-(3-Hydroxy-4,4-dimethyl-2-oxopyrrolidin-1-yl) acetic acid as a solid supported chiral auxiliary in the asymmetric synthesis of β 2-homoarylglycines
Akkari, Rhalid, Calmès, Monique, Di Malta, Delphine, Escale, Françoise, Martinez, Jean
Published in Tetrahedron: asymmetry (2003)
Published in Tetrahedron: asymmetry (2003)
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