Metallo-β-lactamase inhibitors by bioisosteric replacement: Preparation, activity and binding
Skagseth, Susann, Akhter, Sundus, Paulsen, Marianne H., Muhammad, Zeeshan, Lauksund, Silje, Samuelsen, Ørjan, Leiros, Hanna-Kirsti S., Bayer, Annette
Published in European journal of medicinal chemistry (28.07.2017)
Published in European journal of medicinal chemistry (28.07.2017)
Get full text
Journal Article
Structural studies of triazole inhibitors with promising inhibitor effects against antibiotic resistance metallo-β-lactamases
Muhammad, Zeeshan, Skagseth, Susann, Boomgaren, Marc, Akhter, Sundus, Fröhlich, Christopher, Ismael, Aya, Christopeit, Tony, Bayer, Annette, Leiros, Hanna-Kirsti S.
Published in Bioorganic & medicinal chemistry (01.08.2020)
Published in Bioorganic & medicinal chemistry (01.08.2020)
Get full text
Journal Article
A focused fragment library targeting the antibiotic resistance enzyme - Oxacillinase-48: Synthesis, structural evaluation and inhibitor design
Akhter, Sundus, Lund, Bjarte Aarmo, Ismael, Aya, Langer, Manuel, Isaksson, Johan, Christopeit, Tony, Leiros, Hanna-Kirsti S., Bayer, Annette
Published in European journal of medicinal chemistry (10.02.2018)
Published in European journal of medicinal chemistry (10.02.2018)
Get full text
Journal Article
Structural Insights into TMB-1 and the Role of Residues 119 and 228 in Substrate and Inhibitor Binding
Skagseth, Susann, Christopeit, Tony, Akhter, Sundus, Bayer, Annette, Samuelsen, Ørjan, Leiros, Hanna-Kirsti S
Published in Antimicrobial agents and chemotherapy (01.08.2017)
Published in Antimicrobial agents and chemotherapy (01.08.2017)
Get full text
Journal Article