Targeting the PI3-kinase/Akt/mTOR signaling pathway
Hassan, Burhan, Akcakanat, Argun, Holder, Ashley M, Meric-Bernstam, Funda
Published in Surgical oncology clinics of North America (01.10.2013)
Published in Surgical oncology clinics of North America (01.10.2013)
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Journal Article
Phase II trial of AKT inhibitor MK-2206 in patients with advanced breast cancer who have tumors with PIK3CA or AKT mutations, and/or PTEN loss/PTEN mutation
Xing, Yan, Lin, Nancy U, Maurer, Matthew A, Chen, Huiqin, Mahvash, Armeen, Sahin, Aysegul, Akcakanat, Argun, Li, Yisheng, Abramson, Vandana, Litton, Jennifer, Chavez-MacGregor, Mariana, Valero, Vicente, Piha-Paul, Sarina A, Hong, David, Do, Kim-Anh, Tarco, Emily, Riall, Dianna, Eterovic, Agda Karina, Wulf, Gerburg M, Cantley, Lewis C, Mills, Gordon B, Doyle, L Austin, Winer, Eric, Hortobagyi, Gabriel N, Gonzalez-Angulo, Ana Maria, Meric-Bernstam, Funda
Published in Breast cancer research : BCR (05.07.2019)
Published in Breast cancer research : BCR (05.07.2019)
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Journal Article
PD-L1 expression in triple-negative breast cancer
Mittendorf, Elizabeth A, Philips, Anne V, Meric-Bernstam, Funda, Qiao, Na, Wu, Yun, Harrington, Susan, Su, Xiaoping, Wang, Ying, Gonzalez-Angulo, Ana M, Akcakanat, Argun, Chawla, Akhil, Curran, Michael, Hwu, Patrick, Sharma, Padmanee, Litton, Jennifer K, Molldrem, Jeffrey J, Alatrash, Gheath
Published in Cancer immunology research (01.04.2014)
Published in Cancer immunology research (01.04.2014)
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Journal Article
A Population of Heterogeneous Breast Cancer Patient-Derived Xenografts Demonstrate Broad Activity of PARP Inhibitor in BRCA1/2 Wild-Type Tumors
Evans, Kurt W, Yuca, Erkan, Akcakanat, Argun, Scott, Stephen M, Arango, Natalia Paez, Zheng, Xiaofeng, Chen, Ken, Tapia, Coya, Tarco, Emily, Eterovic, Agda K, Black, Dalliah M, Litton, Jennifer K, Yap, Timothy A, Tripathy, Debu, Mills, Gordon B, Meric-Bernstam, Funda
Published in Clinical cancer research (01.11.2017)
Published in Clinical cancer research (01.11.2017)
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Journal Article
Biomarkers of Response to Akt Inhibitor MK-2206 in Breast Cancer
SANGAI, Takafumi, AKCAKANAT, Argun, MERIC-BERNSTAM, Funda, HUIQIN CHEN, TARCO, Emily, YUN WU, DO, Kim-Anh, MILLER, Todd W, ARTEAGA, Carlos L, MILLS, Gordon B, GONZALEZ-ANGULO, Ana Maria
Published in Clinical cancer research (15.10.2012)
Published in Clinical cancer research (15.10.2012)
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Journal Article
Combined MEK/MDM2 inhibition demonstrates antitumor efficacy in TP53 wild-type thyroid and colorectal cancers with MAPK alterations
Pairawan, Seyed, Akcakanat, Argun, Kopetz, Scott, Tapia, Coya, Zheng, Xiaofeng, Chen, Huiqin, Ha, Min Jin, Rizvi, Yasmeen, Holla, Vijaykumar, Wang, Jing, Evans, Kurt W, Zhao, Ming, Busaidy, Naifa, Fang, Bingliang, Roth, Jack A, Dumbrava, Ecaterina Ileana, Meric-Bernstam, Funda
Published in Scientific reports (24.01.2022)
Published in Scientific reports (24.01.2022)
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First in class dual MDM2/MDMX inhibitor ALRN-6924 enhances antitumor efficacy of chemotherapy in TP53 wild-type hormone receptor-positive breast cancer models
Pairawan, Seyed, Zhao, Ming, Yuca, Erkan, Annis, Allen, Evans, Kurt, Sutton, David, Carvajal, Luis, Ren, Jian-Guo, Santiago, Solimar, Guerlavais, Vincent, Akcakanat, Argun, Tapia, Coya, Yang, Fei, Bose, Priya Subash Chandra, Zheng, Xiaofeng, Dumbrava, Ecaterina Ileana, Aivado, Manuel, Meric-Bernstam, Funda
Published in Breast cancer research : BCR (04.03.2021)
Published in Breast cancer research : BCR (04.03.2021)
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Journal Article
PIK3CA/PTEN Mutations and Akt Activation As Markers of Sensitivity to Allosteric mTOR Inhibitors
MERIC-BERNSTAM, Funda, AKCAKANAT, Argun, PHAN, Alexandria T, WOLFF, Robert A, GUPTA, Sanjay, MILLS, Gordon B, YAO, James, HUIQIN CHEN, DO, Kim-Anh, SANGAI, Takafumi, ADKINS, Farrell, GONZALEZ-ANGULO, Ana Maria, RASHID, Asif, CROSBY, Katherine, MEI DONG
Published in Clinical cancer research (15.03.2012)
Published in Clinical cancer research (15.03.2012)
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Journal Article
Selinexor (KPT-330) demonstrates anti-tumor efficacy in preclinical models of triple-negative breast cancer
Arango, Natalia Paez, Yuca, Erkan, Zhao, Ming, Evans, Kurt W, Scott, Stephen, Kim, Charissa, Gonzalez-Angulo, Ana Maria, Janku, Filip, Ueno, Naoto T, Tripathy, Debu, Akcakanat, Argun, Naing, Aung, Meric-Bernstam, Funda
Published in Breast cancer research : BCR (15.08.2017)
Published in Breast cancer research : BCR (15.08.2017)
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Journal Article
Efficacy of futibatinib, an irreversible fibroblast growth factor receptor inhibitor, in FGFR-altered breast cancer
Saridogan, Turcin, Akcakanat, Argun, Zhao, Ming, Evans, Kurt W, Yuca, Erkan, Scott, Stephen, Kirby, Bryce P, Zheng, Xiaofeng, Ha, Min Jin, Chen, Huiqin, Ng, Patrick K S, DiPeri, Timothy P, Mills, Gordon B, Rodon Ahnert, Jordi, Damodaran, Senthil, Meric-Bernstam, Funda
Published in Scientific reports (18.11.2023)
Published in Scientific reports (18.11.2023)
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Journal Article
Heterogeneous Profile of ROR1 Protein Expression across Tumor Types
Raso, Maria Gabriela, Barrientos Toro, Elizve, Evans, Kurt, Rizvi, Yasmeen, Lazcano, Rossana, Akcakanat, Argun, Sini, Patrizia, Trapani, Francesca, Madlener, Eva Johanna, Waldmeier, Lorenz, Lazar, Alexander, Meric-Bernstam, Funda
Published in Cancers (01.05.2024)
Published in Cancers (01.05.2024)
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Journal Article
Ability to Generate Patient-Derived Breast Cancer Xenografts Is Enhanced in Chemoresistant Disease and Predicts Poor Patient Outcomes
McAuliffe, Priscilla F, Evans, Kurt W, Akcakanat, Argun, Chen, Ken, Zheng, Xiaofeng, Zhao, Hao, Eterovic, Agda Karina, Sangai, Takafumi, Holder, Ashley M, Sharma, Chandeshwar, Chen, Huiqin, Do, Kim-Anh, Tarco, Emily, Gagea, Mihai, Naff, Katherine A, Sahin, Aysegul, Multani, Asha S, Black, Dalliah M, Mittendorf, Elizabeth A, Bedrosian, Isabelle, Mills, Gordon B, Gonzalez-Angulo, Ana Maria, Meric-Bernstam, Funda
Published in PloS one (01.09.2015)
Published in PloS one (01.09.2015)
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Journal Article
eIF4E knockdown decreases breast cancer cell growth without activating Akt signaling
Soni, Alpana, Akcakanat, Argun, Singh, Gopal, Luyimbazi, David, Zheng, Yuhuan, Kim, Doyil, Gonzalez-Angulo, Ana, Meric-Bernstam, Funda
Published in Molecular cancer therapeutics (01.07.2008)
Published in Molecular cancer therapeutics (01.07.2008)
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Journal Article
RAC1 Alterations Induce Acquired Dabrafenib Resistance in Association with Anaplastic Transformation in a Papillary Thyroid Cancer Patient
Bagheri-Yarmand, Rozita, Busaidy, Naifa L, McBeath, Elena, Danysh, Brian P, Evans, Kurt W, Moss, Tyler J, Akcakanat, Argun, Ng, Patrick K S, Knippler, Christina M, Golden, Jalyn A, Williams, Michelle D, Multani, Asha S, Cabanillas, Maria E, Shaw, Kenna R, Meric-Bernstam, Funda, Shah, Manisha H, Ringel, Matthew D, Hofmann, Marie Claude
Published in Cancers (30.09.2021)
Published in Cancers (30.09.2021)
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Journal Article
Rapamycin regulates stearoyl CoA desaturase 1 expression in breast cancer
Luyimbazi, David, Akcakanat, Argun, McAuliffe, Priscilla F, Zhang, Li, Singh, Gopal, Gonzalez-Angulo, Ana Maria, Chen, Huiqin, Do, Kim-Anh, Zheng, Yuhuan, Hung, Mien-Chie, Mills, Gordon B, Meric-Bernstam, Funda
Published in Molecular cancer therapeutics (01.10.2010)
Published in Molecular cancer therapeutics (01.10.2010)
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Journal Article
Epigenetically upregulating TROP2 and SLFN11 enhances therapeutic efficacy of TROP2 antibody drug conjugate sacitizumab govitecan
Zhao, Ming, DiPeri, Timothy P, Raso, Maria Gabriela, Zheng, Xiaofeng, Rizvi, Yasmeen Qamar, Evans, Kurt W, Yang, Fei, Akcakanat, Argun, Roberto Estecio, Marco, Tripathy, Debu, Dumbrava, Ecaterina E, Damodaran, Senthil, Meric-Bernstam, Funda
Published in NPJ breast cancer (11.08.2023)
Published in NPJ breast cancer (11.08.2023)
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Journal Article
The rapamycin-regulated gene expression signature determines prognosis for breast cancer
Akcakanat, Argun, Zhang, Li, Tsavachidis, Spiridon, Meric-Bernstam, Funda
Published in Molecular cancer (24.09.2009)
Published in Molecular cancer (24.09.2009)
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Journal Article
Correction: Ability to Generate Patient-Derived Breast Cancer Xenografts Is Enhanced in Chemoresistant Disease and Predicts Poor Patient Outcomes
McAuliffe, Priscilla F, Evans, Kurt W, Akcakanat, Argun, Chen, Ken, Zheng, Xiaofeng, Zhao, Hao, Eterovic, Agda Karina, Sangai, Takafumi, Holder, Ashley M, Sharma, Chandeshwar, Chen, Huiqin, Do, Kim-Anh, Tarco, Emily, Gagea, Mihai, Naff, Katherine A, Sahin, Aysegul, Multani, Asha S, Black, Dalliah M, Mittendorf, Elizabeth A, Bedrosian, Isabelle, Mills, Gordon B, Gonzalez-Angulo, Ana Maria, Meric-Bernstam, Funda
Published in PloS one (08.03.2016)
Published in PloS one (08.03.2016)
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Journal Article
RNA-binding specificity of Y-box protein 1
Dong, Jinjiang, Akcakanat, Argun, Stivers, David N., Zhang, Jiexin, Kim, Doyil, Meric-Bernstam, Funda
Published in RNA biology (01.01.2009)
Published in RNA biology (01.01.2009)
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