Synthesis of a New Dual Metalloprotease Inhibitor. II. Stereoselective Synthesis of Peptidomimetic [5.7]-Bicyclic Compounds
AKASAKA, Kozo, KOMATSU, Yuki, TAGAMI, Katsuya, SHIMIZU, Toshikazu, SHIMOMURA, Naoyuki, NAKA, Hiroshi, HAYASHI, Kenji, NEGI, Shigeto
Published in Chemical & pharmaceutical bulletin (1999)
Published in Chemical & pharmaceutical bulletin (1999)
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Synthesis of a New Dual Metalloprotease Inhibitor. I. Diastereoselective Alkylation of Protected 6-Oxopipecolic Acid Esters
AKASAKA, Kozo, AKAMATSU, Hiroshi, KIMOTO, Yuichi, KOMATSU, Yuki, SHIMIZU, Toshikazu, SHIMOMURA, Naoyuki, TAGAMI, Katsuya, NEGI, Shigeto
Published in Chemical & pharmaceutical bulletin (1999)
Published in Chemical & pharmaceutical bulletin (1999)
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Synthesis and biological evaluation of (−)-laulimalide analogues
Gallagher, Brian M., Fang, Francis G., Johannes, Charles W., Pesant, Marc, Tremblay, Martin R., Zhao, Hongjuan, Akasaka, Kozo, Li, Xiang-yi, Liu, Junke, Littlefield, Bruce A.
Published in Bioorganic & medicinal chemistry letters (09.02.2004)
Published in Bioorganic & medicinal chemistry letters (09.02.2004)
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E2011 a novel, selective and reversible inhibitor of monoamine oxidase type A
Kagaya, T, Kajiwara, A, Nagato, S, Akasaka, K, Kubota, A
Published in The Journal of pharmacology and experimental therapeutics (01.07.1996)
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Published in The Journal of pharmacology and experimental therapeutics (01.07.1996)
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OXAZOLIDONE DERIVATIVE
AKASAKA, KOZO, NAGATO, SATOSHI, KAJIWARA, AKIHARA, SASAKI, ATSUSHI, YOSHIDA, ICHIROU, IIMURA, YOUICHI, KAGAYA, TAKAKI, KOMATSU, MARIK, KUBOTA, ATSUHIKO, MIZUNO, MASANORI
Year of Publication 09.07.1997
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Year of Publication 09.07.1997
Patent
OXAZOLIDONE DERIVATIVE
KAJIWARA, AKIHARU, AKASAKA, KOZO, NAGATO, SATOSHI, SASAKI, ATSUSHI, YOSHIDA, ICHIROU, IIMURA, YOUICHI, KAGAYA, TAKAKI, KUBOTA, ATSUHIKO, MIZUNO, MASANORI
Year of Publication 29.04.1993
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Year of Publication 29.04.1993
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BIPHENYL DERIVATIVES
AKASAKA, KOZO, UENO, KOHSHI, KOMATSU, YUKI, KAJIWARA AKIHARU, SHIMIZU, TOSHIKAZU, MACHIDA, YOSHIMASA, YONAGA, MASAHIRO, KOMATSU, MAKOTO, UENO, MASATAKA, NAGAOKA, ATSUSHI, NAGATO, SATOSHI, HIGURASHI, KUNIZO, MINAMI, NORIO, YAMANISHI, YOSHIHARU, SHIMOMURA, NAOYUKI, KITAZAWA, NORITAKA
Year of Publication 15.06.1999
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Year of Publication 15.06.1999
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BENZO THIAZOLE DERIVATIVE
ABE SHINYA, YAMATSU ISAO, KATAYAMA SATOSHI, SAKUMA YOSHINORI, SUZUKI TAKESHI, HAYASHI KENJI, MIYAMOTO MITSUAKI, KAWAHARA TETSUYA, AKASAKA KOZO, TANAKA MASAYUKI
Year of Publication 02.08.1991
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Year of Publication 02.08.1991
Patent
Structure-activity relationship of N-[2-(dimethylamino)-6-[3-(5-methyl-4-phenyl-1H-imidazol-1-yl)propoxy]phenyl]-N'-pentylurea and analogs. Novel potent inhibitors of acyl-CoA:cholesterol O-acyltransferase with antiatherosclerotic activity
Kimura, Teiji, Takase, Yasutaka, Hayashi, Kenji, Tanaka, Hiroshi, Ohtsuka, Issei, Saeki, Takao, Kogushi, Motoji, Yamada, Toshie, Fujimori, Tohru
Published in Journal of medicinal chemistry (28.05.1993)
Published in Journal of medicinal chemistry (28.05.1993)
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Structure-activity relationship of a series of phenylureas linked to 4-phenylimidazole. Novel potent inhibitors of acyl-CoA:cholesterol O-acyltransferase with antiatherosclerotic activity. 2
Kimura, Teiji, Watanabe, Nobuhisa, Matsui, Makoto, Hayashi, Kenji, Tanaka, Hiroshi, Ohtsuka, Issei, Saeki, Takao, Kogushi, Motoji, Kabayashi, Hiroko
Published in Journal of medicinal chemistry (28.05.1993)
Published in Journal of medicinal chemistry (28.05.1993)
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Laulimalide Analogs and Uses Thereof
LI XIANG-YI, JOHANNES CHARLES, FANG FRANCIS G, ZHAO HONGJUAN, AKASAKA KOZO, PESANT MARC, GALLAGHER, JR. BRIAN M
Year of Publication 15.04.2010
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Year of Publication 15.04.2010
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LAULIMALIDE ANALOGS WITH ANTI-CANCER ACTIVITITY
AKASAKA, KOZO, FANG, FRANCIS, G, LI, XIANG-YI, PESANT, MARC, JOHANNES, CHARLES, ZHAO, HONGJUAN, GALLAGHER, BRIAN
Year of Publication 24.01.2008
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Year of Publication 24.01.2008
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