Antituberculosis drugs: reducing efflux=increasing activity
Rodrigues, Liliana, Parish, Tanya, Balganesh, Meenakshi, Ainsa, José A.
Published in Drug discovery today (01.03.2017)
Published in Drug discovery today (01.03.2017)
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Spectinamides: a new class of semisynthetic antituberculosis agents that overcome native drug efflux
Lee, Richard E, Hurdle, Julian G, Liu, Jiuyu, Bruhn, David F, Matt, Tanja, Scherman, Michael S, Vaddady, Pavan K, Zheng, Zhong, Qi, Jianjun, Akbergenov, Rashid, Das, Sourav, Madhura, Dora B, Rathi, Chetan, Trivedi, Ashit, Villellas, Cristina, Lee, Robin B, Rakesh, Waidyarachchi, Samanthi L, Sun, Dianqing, McNeil, Michael R, Ainsa, Jose A, Boshoff, Helena I, Gonzalez-Juarrero, Mercedes, Meibohm, Bernd, Böttger, Erik C, Lenaerts, Anne J
Published in Nature medicine (01.02.2014)
Published in Nature medicine (01.02.2014)
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Identification of aminopyrimidine‐sulfonamides as potent modulators of Wag31‐mediated cell elongation in mycobacteria
Singh, Vinayak, Dhar, Neeraj, Pató, János, Kolly, Gaëlle S., Korduláková, Jana, Forbak, Martin, Evans, Joanna C., Székely, Rita, Rybniker, Jan, Palčeková, Zuzana, Zemanová, Júlia, Santi, Isabella, Signorino‐Gelo, François, Rodrigues, Liliana, Vocat, Anthony, Covarrubias, Adrian S., Rengifo, Monica G., Johnsson, Kai, Mowbray, Sherry, Buechler, Joseph, Delorme, Vincent, Brodin, Priscille, Knott, Graham W., Aínsa, José A., Warner, Digby F., Kéri, György, Mikušová, Katarína, McKinney, John D., Cole, Stewart T., Mizrahi, Valerie, Hartkoorn, Ruben C.
Published in Molecular microbiology (01.01.2017)
Published in Molecular microbiology (01.01.2017)
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Boldine-Derived Alkaloids Inhibit the Activity of DNA Topoisomerase I and Growth of Mycobacterium tuberculosis
García, María T, Carreño, David, Tirado-Vélez, José M, Ferrándiz, María J, Rodrigues, Liliana, Gracia, Begoña, Amblar, Mónica, Ainsa, José A, de la Campa, Adela G
Published in Frontiers in microbiology (24.07.2018)
Published in Frontiers in microbiology (24.07.2018)
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A Prodrug Approach for Improving Antituberculosis Activity of Potent Mycobacterium tuberculosis Type II Dehydroquinase Inhibitors
Tizón, Lorena, Otero, José M, Prazeres, Verónica F. V, Llamas-Saiz, Antonio L, Fox, Gavin C, van Raaij, Mark J, Lamb, Heather, Hawkins, Alastair R, Ainsa, José A, Castedo, Luis, González-Bello, Concepción
Published in Journal of medicinal chemistry (08.09.2011)
Published in Journal of medicinal chemistry (08.09.2011)
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Role of the Mmr Efflux Pump in Drug Resistance in Mycobacterium tuberculosis
RODRIGUES, Liliana, VILLELLAS, Cristina, BAILO, Rebeca, VIVEIROS, Miguel, AINSA, Jose A
Published in Antimicrobial Agents and Chemotherapy (01.02.2013)
Published in Antimicrobial Agents and Chemotherapy (01.02.2013)
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How can nanoparticles contribute to antituberculosis therapy?
Costa-Gouveia, Joana, Aínsa, José A., Brodin, Priscille, Lucía, Ainhoa
Published in Drug discovery today (01.03.2017)
Published in Drug discovery today (01.03.2017)
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Role of mycobacterial efflux transporters in drug resistance: an unresolved question
Rossi, Edda De, Aínsa, José A., Riccardi, Giovanna
Published in FEMS microbiology reviews (01.01.2006)
Published in FEMS microbiology reviews (01.01.2006)
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Co-delivery of free vancomycin and transcription factor decoy-nanostructured lipid carriers can enhance inhibition of methicillin resistant Staphylococcus aureus (MRSA)
Hibbitts, Alan, Lucía, Ainhoa, Serrano-Sevilla, Inés, De Matteis, Laura, McArthur, Michael, de la Fuente, Jesús M, Aínsa, José A, Navarro, Fabrice
Published in PloS one (03.09.2019)
Published in PloS one (03.09.2019)
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Functional and Genetic Characterization of the Tap Efflux Pump in Mycobacterium bovis BCG
Ramón-García, Santiago, Mick, Virginie, Dainese, Elisa, Martín, Carlos, Thompson, Charles J, De Rossi, Edda, Manganelli, Riccardo, Aínsa, José A
Published in Antimicrobial Agents and Chemotherapy (01.04.2012)
Published in Antimicrobial Agents and Chemotherapy (01.04.2012)
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Synergy between Circular Bacteriocin AS-48 and Ethambutol against Mycobacterium tuberculosis
Aguilar-Pérez, Clara, Gracia, Begoña, Rodrigues, Liliana, Vitoria, Asunción, Cebrián, Rubén, Deboosère, Nathalie, Song, Ok-Ryul, Brodin, Priscille, Maqueda, Mercedes, Aínsa, José A
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Published in Antimicrobial agents and chemotherapy (01.09.2018)
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Zanthoxylum capense constituents with antimycobacterial activity against Mycobacterium tuberculosis in vitro and ex vivo within human macrophages
Luo, Xuan, Pires, David, Aínsa, José A., Gracia, Begoña, Duarte, Noélia, Mulhovo, Silva, Anes, Elsa, Ferreira, Maria-José U.
Published in Journal of ethnopharmacology (07.03.2013)
Published in Journal of ethnopharmacology (07.03.2013)
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Mycobacterial Aminoglycoside Acetyltransferases: A Little of Drug Resistance, and a Lot of Other Roles
Sanz-García, Fernando, Anoz-Carbonell, Ernesto, Pérez-Herrán, Esther, Martín, Carlos, Lucía, Ainhoa, Rodrigues, Liliana, Aínsa, José A
Published in Frontiers in microbiology (2019)
Published in Frontiers in microbiology (2019)
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Structure-aided optimization of non-nucleoside M. tuberculosis thymidylate kinase inhibitors
Song, Lijun, Merceron, Romain, Hulpia, Fabian, Lucía, Ainhoa, Gracia, Begoña, Jian, Yanlin, Risseeuw, Martijn D.P., Verstraelen, Toon, Cos, Paul, Aínsa, José A., Boshoff, Helena I., Munier-Lehmann, Hélène, Savvides, Savvas N., Van Calenbergh, Serge
Published in European journal of medicinal chemistry (05.12.2021)
Published in European journal of medicinal chemistry (05.12.2021)
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Structure Guided Lead Generation toward Nonchiral M. tuberculosis Thymidylate Kinase Inhibitors
Song, Lijun, Merceron, Romain, Gracia, Begoña, Quintana, Ainhoa Lucía, Risseeuw, Martijn D. P, Hulpia, Fabian, Cos, Paul, Aínsa, José A, Munier-Lehmann, Hélène, Savvides, Savvas N, Van Calenbergh, Serge
Published in Journal of medicinal chemistry (12.04.2018)
Published in Journal of medicinal chemistry (12.04.2018)
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Analysis of Mutations in Streptomycin-Resistant Strains Reveals a Simple and Reliable Genetic Marker for Identification of the Mycobacterium tuberculosis Beijing Genotype
Villellas, Cristina, Aristimuño, Liselotte, Vitoria, María-Asunción, Prat, Cristina, Blanco, Silvia, García de Viedma, Darío, Domínguez, José, Samper, Sofía, Aínsa, José A
Published in Journal of Clinical Microbiology (01.07.2013)
Published in Journal of Clinical Microbiology (01.07.2013)
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