651 A phase 1, multicenter, open-label, dose-escalation, safety, pharmacodynamic, pharmacokinetic study of Q702 with a cohort expansion at the RP2D in patients with advanced solid tumors
Mahalingam, Devalingam, Alistar, Angela, Mita, Alain, Kim, Jeongjun, Ahn, Hyunji, Choi, Jinho, Ryu, Seung-Hee, Ahn, Jiye, Choi, Bae Jung, Kang, Hwankyu, Yang, Yeong-In, Lee, Seung-Joo, Jeon, Borami, Proniuk, Stefan, Nam, Kiyean, El-Khoueiry, Anthony
Published in Journal for immunotherapy of cancer (01.11.2023)
Published in Journal for immunotherapy of cancer (01.11.2023)
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Journal Article
645 A phase 1B/2, open-label study of Q702 in combination with intravenous pembrolizumab in patients with selected advanced solid tumors
Kim, Seung-Tae, Chon, Hong Jae, Oh, Do-Youn, Grewal, Jaspreet, Rha, Sun Young, El-Khoueiry, Anthony, Ryoo, Baek-Yeol, Kim, Jeongjun, Ahn, Hyunji, Ryu, Seung-Hee, Choi, Jinho, Choi, Bae Jung, Ahn, Jiye, Kang, Hwankyu, Yang, Yeong-In, Lee, Seung-Joo, Jeon, Borami, Proniuk, Stefan, Nam, Kiyean
Published in Journal for immunotherapy of cancer (01.11.2023)
Published in Journal for immunotherapy of cancer (01.11.2023)
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Journal Article
Potential of the Volatile-Producing Fungus Nodulisporium sp. CF016 for the Control of Postharvest Diseases of Apple
Park, M.S., Korea Research Institute of Chemical Technology, Daejeon, Republic of Korea, Ahn, J.Y., Korea Research Institute of Chemical Technology, Daejeon, Republic of Korea, Choi, G.J., Korea Research Institute of Chemical Technology, Daejeon, Republic of Korea, Choi, Y.H., Korea Research Institute of Chemical Technology, Daejeon, Republic of Korea, Jang, K.S., Korea Research Institute of Chemical Technology, Daejeon, Republic of Korea, Kim, J.C., Korea Research Institute of Chemical Technology, Daejeon, Republic of Korea
Published in The plant pathology journal (01.09.2010)
Published in The plant pathology journal (01.09.2010)
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Journal Article
Safety, Tolerability, and Pharmacokinetics of Telacebec (Q203), a New Antituberculosis Agent, in Healthy Subjects
Kim, Jeongjun, Choi, Jinho, Kang, Hwankyu, Ahn, Jiye, Hutchings, Jane, van Niekerk, Christo, Park, Dongsik, Kim, Jaeseung, Jeon, Yeejin, Nam, Kiyean, Shin, Soyoung, Shin, Beom Soo
Published in Antimicrobial agents and chemotherapy (18.01.2022)
Published in Antimicrobial agents and chemotherapy (18.01.2022)
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Journal Article
Safety, Tolerability, Pharmacokinetics, and Metabolism of Telacebec (Q203) for the Treatment of Tuberculosis: a Randomized, Placebo-Controlled, Multiple Ascending Dose Phase 1B Trial
Kim, Jeongjun, Choi, Jinho, Kang, Hwankyu, Ahn, Jiye, Hutchings, Jane, Niekerk, Christo van, Kim, Jaeseung, Jeon, Yeejin, Nam, Kiyean, Kim, Tae Hwan, Shin, Beom Soo, Shin, Soyoung
Published in Antimicrobial agents and chemotherapy (24.01.2023)
Published in Antimicrobial agents and chemotherapy (24.01.2023)
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Journal Article
GM-CSF and IL-4 produced by NKT cells inversely regulate IL-1β production by macrophages
Ahn, Sehee, Jeong, Dongjin, Oh, Sae Jin, Ahn, Jiye, Lee, Seung Hyo, Chung, Doo Hyun
Published in Immunology letters (01.02.2017)
Published in Immunology letters (01.02.2017)
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Journal Article
A phase 1, multicenter, open-label, dose-escalation, safety, pharmacodynamic, pharmacokinetic study of Q702 with a cohort expansion at the RP2D in patients with advanced solid tumors
Alistar, Angela Tatiana, El-Khoueiry, Anthony B., Mahalingam, Devalingam, Mita, Monica M., Kang, Hwankyu, Yang, Yeong-In, Ahn, Jiye, Kim, Jeongjun, Choi, Baejung, Jeon, Yeejin, Jung, Chunwon, Jeon, Borami, Kim, Jaeseung, Nam, Kiyean
Published in Journal of clinical oncology (20.05.2021)
Published in Journal of clinical oncology (20.05.2021)
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Journal Article
Abstract A205: Q701, a selective Axl and Mer inhibitor as an immune checkpoint inhibitor
Yang, Yeong-In, Kang, Hwankyu, Park, Dongsik, Ahn, Jiye, Choi, Jinho, Ahn, Seohyun, Kim, Jaeseung, Nam, Kiyean
Published in Molecular cancer therapeutics (01.01.2018)
Published in Molecular cancer therapeutics (01.01.2018)
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Journal Article
Abstract 5712: Functional dissection of CDK7 in transcription using a highly selective CDK7 inhibitor Q901
Jung, Hyerim, Um, Dahun, Lee, Yoonji, Yu, Donghoon, Lee, Dayoung, Ahn, Jiye, Kim, Jeongjun, Lee, Seung-Joo, Kim, Jaeseung, Nam, Kiyean, Kim, Tae-Kyung
Published in Cancer research (Chicago, Ill.) (22.03.2024)
Published in Cancer research (Chicago, Ill.) (22.03.2024)
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Abstract B162: Highly selective, orally available CDK7 inhibitor for cancer therapy
Jeon, Yeejin, Yu, Donghoon, Seo, Mooyoung, Kim, June, Shin, Jaehee, Kang, Hwankyu, Ahn, Jiye, Choi, Jinho, Ahn, Seohyun, Kim, Jaeseung, Nam, Kiyean
Published in Molecular cancer therapeutics (01.01.2018)
Published in Molecular cancer therapeutics (01.01.2018)
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Journal Article
Abstract 2255: Patient pharmacodynamic biomarker and pk evaluation results from an ongoing phase I dose-escalation study of q702, an axl, mer and csf1r kinase inhibitor in patients with advanced solid tumors
Choi, Bae Jung, Devalingam, Devalingam, Alistar, Angela, El-Khoueiry, Anthony, Mita, Alain, Kang, Hwankyu, Choi, Jinho, Ahn, Hyunji, Kim, Jeongjun, Lee, Seung-Joo, Yang, Yeong-In, Ahn, Jiye, Jeon, Borami, Kim, Jaeseung, Nam, Kiyean
Published in Cancer research (Chicago, Ill.) (04.04.2023)
Published in Cancer research (Chicago, Ill.) (04.04.2023)
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Journal Article
A novel 3,4-dihydropyrimidin-2(1H)-one: HIV-1 replication inhibitors with improved metabolic stability
Kim, Junwon, Ok, Taedong, Park, Changmin, So, Wonyoung, Jo, Mina, Kim, Youngmi, Seo, Minjung, Lee, Doohyun, Jo, Suyeon, Ko, Yoonae, Choi, Inhee, Park, Youngsam, Yoon, Jaewan, Ju, Moon Kyeong, Ahn, JiYe, Kim, Junghwan, Han, Sung-Jun, Kim, Tae-Hee, Cechetto, Jonathan, Nam, Jiyoun, Liuzzi, Michel, Sommer, Peter, No, Zaesung
Published in Bioorganic & medicinal chemistry letters (01.04.2012)
Published in Bioorganic & medicinal chemistry letters (01.04.2012)
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Journal Article
Serendipitous discovery of 2-((phenylsulfonyl)methyl)-thieno[3,2-d]pyrimidine derivatives as novel HIV-1 replication inhibitors
Kim, Junwon, Kwon, Jeongjin, Lee, Doohyun, Jo, Suyeon, Park, Dong-Sik, Choi, Jihyun, Park, Eunjung, Hwang, Jong Yeon, Ko, Yoonae, Choi, Inhee, Ju, Moon Kyeong, Ahn, JiYe, Kim, Junghwan, Han, Sung-Jun, Kim, Tae-Hee, Cechetto, Jonathan, Nam, Jiyoun, Ahn, Sujin, Sommer, Peter, Liuzzi, Michel, Lee, Jinhwa
Published in Bioorganic & medicinal chemistry letters (01.12.2014)
Published in Bioorganic & medicinal chemistry letters (01.12.2014)
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Journal Article
Synthesis and biological evaluation of triazolothienopyrimidine derivatives as novel HIV-1 replication inhibitors
Kim, Junwon, Kwon, Jeongjin, Lee, Doohyun, Jo, Suyeon, Park, Dong-Sik, Choi, Jihyun, Park, Eunjung, Hwang, Jong Yeon, Ko, Yoonae, Choi, Inhee, Ju, Moon Kyeong, Ahn, JiYe, Kim, Junghwan, Han, Sung-Jun, Kim, Tae-Hee, Cechetto, Jonathan, Nam, Jiyoun, Ahn, Sujin, Sommer, Peter, Liuzzi, Michel, No, Zaesung, Lee, Jinhwa
Published in Bioorganic & medicinal chemistry letters (01.01.2013)
Published in Bioorganic & medicinal chemistry letters (01.01.2013)
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Journal Article
QUINOLINE DERIVATIVES AS TAM RTK INHIBITORS
CARSTEN SCHULTZ-FADEMRECHT, JUNG CHUN-WON, LEE SAE YOUNG, YANG YOUNG-IN, AHN JIYE, JEON YEEJIN, LEE DOOHYUNG, KIM JEONG-JUN, KIM JAESUNG, AHN SEOHYUN, PARK DONG SIK, KIM HANA, NAM KIYEAN
Year of Publication 23.01.2020
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Year of Publication 23.01.2020
Patent
ANTI-INFECTIVE COMPOUND
SEO JEONGJEA, OH SOOHYUN, AHN JIYE, SEO MOOYOUNG, KANG SUNHEE, KIM JEONG-JUN, KIM RYANG YEO, LEE SAEYEON, KANG JUHEE, KEVIN PETHE, KIM JAESUNG, SEO MIN JUNG, PARK DONG SIK, LEE SUMI, NAM KIYEAN
Year of Publication 08.08.2019
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Year of Publication 08.08.2019
Patent
ANTI-INFECTIVE COMPOUND
SEO JEONGJEA, OH SOOHYUN, AHN JIYE, SEO MOOYOUNG, KANG SUNHEE, KIM JEONG-JUN, KIM RYANG YEO, LEE SAEYEON, KANG JUHEE, KEVIN PETHE, KIM JAESUNG, SEO MIN JUNG, PARK DONG SIK, LEE SUMI, NAM KIYEAN
Year of Publication 11.10.2018
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Year of Publication 11.10.2018
Patent
TAM RTK 억제제로서 퀴놀린 유도체들
PARK DONGSIK, AHN JIYE, KIM JAESEUNG, SCHULTZ FADEMRECHT CARSTEN, JEON YEEJIN, LEE DOOHYUNG, LEE SAEYEON, AHN SEOHYUN, KIM HANA, JUNG CHUN WON, NAM KIYEAN, YANG YEONG IN, KIM JEONGJUN
Year of Publication 08.12.2017
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Year of Publication 08.12.2017
Patent
2-- 5- / E 2-AMINO-BENZIMIDAZOLE DERIVATIVES AND THEIR USE AS 5-LIPOXYGENASE AND/OR PROSTAGLANDIN E SYNTHASE INHIBITORS
PARK DONGSIK, SEO JEONGJEA, AHN JIYE, KIM JUNG HWAN, LEE YUNMI, KIM JAESEUNG, SEO MOOYOUNG, JEON YEEJIN, KANG SUNHEE, LEE SANGCHUL, LEE DOOHYUNG, CHOI GAHEE, HAN SUNG JUN, LEE SAEYEON, AHN SEOHYUN, SEO MINJUNG, NAM KIYEAN, YANG YEONG IN, KIM JEONGJUN
Year of Publication 26.04.2017
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Year of Publication 26.04.2017
Patent
QUINOLINE DERIVATIVES AS TAM RTK INHIBITORS
JAESEUNG, Kim, YEEJIN, Jeon, KIYEAN, Nam, JIYE, Ahn, HANA, Kim, DOOHYUNG, Lee, YOUNG-IN, Yang, SAEYEON, Lee, DONGSIK, Park, JEONGJUN, Kim, SCHULTZ-FADEMRECHT, Carsten, SEOHYUN, Ahn, CHUN-WON, Jung
Year of Publication 13.03.2023
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Year of Publication 13.03.2023
Patent