Development of a sensitive high-throughput enzymatic assay capable of measuring sub-nanomolar inhibitors of SARS-CoV2 Mpro
Kovar, Peter, Richardson, Paul L, Korepanova, Alla, Afanador, Gustavo A, Stojkovic, Vladimir, Li, Tao, Schrimpf, Michael R, Ng, Teresa I, Degoey, David A, Gopalakrishnan, Sujatha M, Chen, Jun
Published in SLAS discovery (01.09.2024)
Published in SLAS discovery (01.09.2024)
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Journal Article
Novel N-Benzoyl-2-Hydroxybenzamide Disrupts Unique Parasite Secretory Pathway
Fomovska, Alina, Huang, Qingqing, El Bissati, Kamal, Mui, Ernest J, Witola, William H, Cheng, Gang, Zhou, Ying, Sommerville, Caroline, Roberts, Craig W, Bettis, Sam, Prigge, Sean T, Afanador, Gustavo A, Hickman, Mark R, Lee, Patty J, Leed, Susan E, Auschwitz, Jennifer M, Pieroni, Marco, Stec, Jozef, Muench, Stephen P, Rice, David W, Kozikowski, Alan P, McLeod, Rima
Published in Antimicrobial Agents and Chemotherapy (01.05.2012)
Published in Antimicrobial Agents and Chemotherapy (01.05.2012)
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Journal Article
A novel lipoate attachment enzyme is shared by Plasmodium and Chlamydia species
Afanador, Gustavo A., Guerra, Alfredo J., Swift, Russell P., Rodriguez, Ryan E., Bartee, David, Matthews, Krista A., Schön, Arne, Freire, Ernesto, Freel Meyers, Caren L., Prigge, Sean T.
Published in Molecular microbiology (01.11.2017)
Published in Molecular microbiology (01.11.2017)
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Journal Article
Identification and Mechanistic Understanding of Dihydroorotate Dehydrogenase Point Mutations in Plasmodium falciparum that Confer in Vitro Resistance to the Clinical Candidate DSM265
White, John, Dhingra, Satish K, Deng, Xiaoyi, El Mazouni, Farah, Lee, Marcus C. S, Afanador, Gustavo A, Lawong, Aloysus, Tomchick, Diana R, Ng, Caroline L, Bath, Jade, Rathod, Pradipsinh K, Fidock, David A, Phillips, Margaret A
Published in ACS infectious diseases (11.01.2019)
Published in ACS infectious diseases (11.01.2019)
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Journal Article
Design, synthesis, and biological activity of diaryl ether inhibitors of Toxoplasma gondii enoyl reductase
Cheng, Gang, Muench, Stephen P., Zhou, Ying, Afanador, Gustavo A., Mui, Ernest J., Fomovska, Alina, Lai, Bo Shiun, Prigge, Sean T., Woods, Stuart, Roberts, Craig W., Hickman, Mark R., Lee, Patty J., Leed, Susan E., Auschwitz, Jennifer M., Rice, David W., McLeod, Rima
Published in Bioorganic & medicinal chemistry letters (01.04.2013)
Published in Bioorganic & medicinal chemistry letters (01.04.2013)
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Journal Article
Development of a triclosan scaffold which allows for adaptations on both the A- and B-ring for transport peptides
Muench, Stephen P., Stec, Jozef, Zhou, Ying, Afanador, Gustavo A., McPhillie, Martin J., Hickman, Mark R., Lee, Patty J., Leed, Susan E., Auschwitz, Jennifer M., Prigge, Sean T., Rice, David W., McLeod, Rima
Published in Bioorganic & medicinal chemistry letters (15.06.2013)
Published in Bioorganic & medicinal chemistry letters (15.06.2013)
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Journal Article
Discrimination of Potent Inhibitors of Toxoplasma gondii Enoyl-Acyl Carrier Protein Reductase by a Thermal Shift Assay
Afanador, Gustavo A, Muench, Stephen P, McPhillie, Martin, Fomovska, Alina, Schön, Arne, Zhou, Ying, Cheng, Gang, Stec, Jozef, Freundlich, Joel S, Shieh, Hong-Ming, Anderson, John W, Jacobus, David P, Fidock, David A, Kozikowski, Alan P, Fishwick, Colin W, Rice, David W, Freire, Ernesto, McLeod, Rima, Prigge, Sean T
Published in Biochemistry (Easton) (23.12.2013)
Published in Biochemistry (Easton) (23.12.2013)
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Journal Article
Novel TypeII Fatty Acid Biosynthesis (FAS II) Inhibitors as Multistage Antimalarial Agents
Schrader, Florian C., Glinca, Serghei, Sattler, Julia M., Dahse, Hans-Martin, Afanador, Gustavo A., Prigge, Sean T., Lanzer, Michael, Mueller, Ann-Kristin, Klebe, Gerhard, Schlitzer, Martin
Published in ChemMedChem (01.03.2013)
Published in ChemMedChem (01.03.2013)
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Journal Article
The benzimidazole based drugs show good activity against T. gondii but poor activity against its proposed enoyl reductase enzyme target
Wilkinson, Craig, McPhillie, Martin J., Zhou, Ying, Woods, Stuart, Afanador, Gustavo A., Rawson, Shaun, Khaliq, Farzana, Prigge, Sean T., Roberts, Craig W., Rice, David W., McLeod, Rima, Fishwick, Colin W., Muench, Stephen P.
Published in Bioorganic & medicinal chemistry letters (01.02.2014)
Published in Bioorganic & medicinal chemistry letters (01.02.2014)
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Journal Article
Modification of Triclosan Scaffold in Search of Improved Inhibitors for Enoyl-Acyl Carrier Protein (ACP) Reductase in Toxoplasma gondii
Stec, Jozef, Fomovska, Alina, Afanador, Gustavo A., Muench, Stephen P., Zhou, Ying, Lai, Bo-Shiun, El Bissati, Kamal, Hickman, Mark R., Lee, Patty J., Leed, Susan E., Auschwitz, Jennifer M., Sommervile, Caroline, Woods, Stuart, Roberts, Craig W., Rice, David, Prigge, Sean T., McLeod, Rima, Kozikowski, Alan P.
Published in ChemMedChem (01.07.2013)
Published in ChemMedChem (01.07.2013)
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Journal Article
Novel Type II Fatty Acid Biosynthesis (FAS II) Inhibitors as Multistage Antimalarial Agents
Schrader, Florian C., Glinca, Serghei, Sattler, Julia M., Dahse, Hans-Martin, Afanador, Gustavo A., Prigge, Sean T., Lanzer, Michael, Mueller, Ann-Kristin, Klebe, Gerhard, Schlitzer, Martin
Published in ChemMedChem (01.03.2013)
Published in ChemMedChem (01.03.2013)
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Journal Article
Cover Image, Volume 85, Issue 9: Malaria Parasite Lipoate Ligase Structure
Guerra, Alfredo J., Afanador, Gustavo A., Prigge, Sean T.
Published in Proteins, structure, function, and bioinformatics (01.09.2017)
Published in Proteins, structure, function, and bioinformatics (01.09.2017)
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Journal Article
Cover Image, Volume 85, Issue 9
Guerra, Alfredo J, Afanador, Gustavo A, Prigge, Sean T
Published in Proteins, structure, function, and bioinformatics (01.09.2017)
Published in Proteins, structure, function, and bioinformatics (01.09.2017)
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