CYP46A1 inhibition and activation: an in vitro high throughput screening assay to assess possible drug interactions using FDA approved chemical library
Adusumalli, Sravani, Metallides, Megan, Pham, Jennifer, Strock, Sarah, Strock, Christopher
Published in Drug metabolism and pharmacokinetics (01.04.2024)
Published in Drug metabolism and pharmacokinetics (01.04.2024)
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Journal Article
Use of SWATH-MS to relatively quantify the expression of hepatic drug metabolizing enzymes in human liver microsomes using a label-free approach
Jamwal, Rohitash, Barlock, Benjamin J., Adusumalli, Sravani, Ogasawara, Ken, Simons, Brigitte L., Akhlaghi, Fatemeh
Published in Drug metabolism and pharmacokinetics (01.01.2018)
Published in Drug metabolism and pharmacokinetics (01.01.2018)
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Journal Article
Decreased CYP3A4 activity and protein in nonalcoholic fatty liver (NAFL) and nonalcoholic steatohepatitis (NASH)
Jamwal, Rohitash, Barlock, Benjamin J., Adusumalli, Sravani, Ogasawara, Ken, La Monte, Suzanne M De, Akhlaghi, Fatemeh
Published in Drug metabolism and pharmacokinetics (01.01.2018)
Published in Drug metabolism and pharmacokinetics (01.01.2018)
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Journal Article
Characterization of Byproducts from Chemical Syntheses of Oligonucleotides Containing 1‑Methyladenine and 3‑Methylcytosine
Tang, Qi, Cai, Ang, Bian, Ke, Chen, Fangyi, Delaney, James C, Adusumalli, Sravani, Bach, Alvin C, Akhlaghi, Fatemeh, Cho, Bongsup P, Li, Deyu
Published in ACS omega (30.11.2017)
Published in ACS omega (30.11.2017)
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Journal Article
Nonalcoholic Fatty Liver Disease and Diabetes Are Associated with Decreased CYP3A4 Protein Expression and Activity in Human Liver
Jamwal, Rohitash, de la Monte, Suzanne M, Ogasawara, Ken, Adusumalli, Sravani, Barlock, Benjamin B, Akhlaghi, Fatemeh
Published in Molecular pharmaceutics (02.07.2018)
Published in Molecular pharmaceutics (02.07.2018)
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Journal Article
Development and validation of an assay for a novel ghrelin receptor inverse agonist PF-5190457 and its major hydroxy metabolite (PF-6870961) by LC-MS/MS in human plasma
Adusumalli, Sravani, Jamwal, Rohitash, Leggio, Lorenzo, Akhlaghi, Fatemeh
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (01.11.2019)
Published in Journal of chromatography. B, Analytical technologies in the biomedical and life sciences (01.11.2019)
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Journal Article
Multiplex and Label-Free Relative Quantification Approach for Studying Protein Abundance of Drug Metabolizing Enzymes in Human Liver Microsomes Using SWATH-MS
Jamwal, Rohitash, Barlock, Benjamin J, Adusumalli, Sravani, Ogasawara, Ken, Simons, Brigitte L, Akhlaghi, Fatemeh
Published in Journal of proteome research (03.11.2017)
Published in Journal of proteome research (03.11.2017)
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Journal Article
Role of Molybdenum-Containing Enzymes in the Biotransformation of the Novel Ghrelin Receptor Inverse Agonist PF-5190457: A Reverse Translational Bed-to-Bench Approach
Adusumalli, Sravani, Jamwal, Rohitash, Obach, R Scott, Ryder, Tim F, Leggio, Lorenzo, Akhlaghi, Fatemeh
Published in Drug metabolism and disposition (01.08.2019)
Published in Drug metabolism and disposition (01.08.2019)
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Journal Article
Initial Pharmacological Characterization of a Major Hydroxy Metabolite of PF-5190457: Inverse Agonist Activity of PF-6870961 at the Ghrelin Receptor
Deschaine, Sara L, Hedegaard, Morten A, Pince, Claire L, Farokhnia, Mehdi, Moose, Jacob E, Stock, Ingrid A, Adusumalli, Sravani, Akhlaghi, Fatemeh, Hougland, James L, Sulima, Agnieszka, Rice, Kenner C, Koob, George F, Vendruscolo, Leandro F, Holst, Birgitte, Leggio, Lorenzo
Published in The Journal of pharmacology and experimental therapeutics (01.08.2023)
Published in The Journal of pharmacology and experimental therapeutics (01.08.2023)
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Journal Article