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Glucocorticoid Receptor Modulators Informed by Crystallography Lead to a New Rationale for Receptor Selectivity, Function, and Implications for Structure-Based Design
Carson, Matthew W, Luz, John G, Suen, Chen, Montrose, Chahrzad, Zink, Richard, Ruan, Xiaoping, Cheng, Christine, Cole, Harlan, Adrian, Mary D, Kohlman, Dan T, Mabry, Thomas, Snyder, Nancy, Condon, Brad, Maletic, Milan, Clawson, David, Pustilnik, Anna, Coghlan, Michael J
Published in Journal of medicinal chemistry (13.02.2014)
Published in Journal of medicinal chemistry (13.02.2014)
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Repurposing a novel parathyroid hormone analogue to treat hypoparathyroidism
Krishnan, Venkatesh, Ma, Yanfei L, Chen, Catherine Z, Thorne, Natasha, Bullock, Heather, Tawa, Gregory, Javella‐Cauley, Christy, Chu, Shaoyou, Li, Weiming, Kohn, Wayne, Adrian, Mary D, Benson, Charles, Liu, Lifei, Sato, Masahiko, Zheng, Wei, Pilon, Andre M, Yang, N. Nora, Bryant, Henry U
Published in British journal of pharmacology (01.01.2018)
Published in British journal of pharmacology (01.01.2018)
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Efficacy of a sclerostin antibody compared to a low dose of PTH on metaphyseal bone healing
Agholme, Fredrik, Macias, Brandon, Hamang, Matt, Lucchesi, Jonathan, Adrian, Mary D., Kuhstoss, Stuart, Harvey, Anita, Sato, Masahiko, Aspenberg, Per
Published in Journal of orthopaedic research (01.03.2014)
Published in Journal of orthopaedic research (01.03.2014)
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Time course of disassociation of bone formation signals with bone mass and bone strength in sclerostin antibody treated ovariectomized rats
Ma, Yanfei L, Hamang, Matthew, Lucchesi, Jonathan, Bivi, Nicoletta, Zeng, Qianqiang, Adrian, Mary D, Raines, Sarah E, Li, Jiliang, Kuhstoss, Stuart A, Obungu, Victor, Bryant, Henry U, Krishnan, Venkatesh
Published in Bone (New York, N.Y.) (01.04.2017)
Published in Bone (New York, N.Y.) (01.04.2017)
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A New Selective Estrogen Receptor Modulator with Potent Uterine Antagonist Activity, Agonist Activity in Bone, and Minimal Ovarian Stimulation
Geiser, Andrew G., Hummel, Conrad W., Draper, Michael W., Henck, Judith W., Cohen, Ilene R., Rudmann, Daniel G., Donnelly, Kevin B, Adrian, Mary D., Shepherd, Timothy A., Wallace, Owen B., McCann, Denis J., Oldham, Samuel W., Bryant, Henry U., Sato, Masahiko, Dodge, Jeffrey A.
Published in Endocrinology (Philadelphia) (01.10.2005)
Published in Endocrinology (Philadelphia) (01.10.2005)
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A Selective Estrogen Receptor Modulator for the Treatment of Hot Flushes
Wallace, Owen B, Lauwers, Kenneth S, Dodge, Jeffrey A, May, Scott A, Calvin, Joel R, Hinklin, Ronald, Bryant, Henry U, Shetler, Pamela K, Adrian, Mary D, Geiser, Andrew G, Sato, Masahiko, Burris, Thomas P
Published in Journal of medicinal chemistry (09.02.2006)
Published in Journal of medicinal chemistry (09.02.2006)
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Benzothiophene and naphthalene derived constrained SERMs
Wallace, Owen B., Bryant, Henry U., Shetler, Pamela K., Adrian, Mary D., Geiser, Andrew G.
Published in Bioorganic & medicinal chemistry letters (18.10.2004)
Published in Bioorganic & medicinal chemistry letters (18.10.2004)
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B-Ring unsaturated estrogens: biological evaluation of 17α-Dihydroequilein and novel B-Nor-6-thiaequilenins as tissue selective estrogens
Lugar, Charles W, Magee, David, Adrian, Mary D, Shetler, Pamela, Bryant, Henry U, Dodge, Jeffrey A
Published in Bioorganic & medicinal chemistry letters (15.12.2003)
Published in Bioorganic & medicinal chemistry letters (15.12.2003)
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Efficacy of a sclerostin antibody compared to a low dose of PTH on metaphyseal bone healing: SCLEROSTIN ANTIBODY VERSUS PTH
Agholme, Fredrik, Macias, Brandon, Hamang, Matt, Lucchesi, Jonathan, Adrian, Mary D., Kuhstoss, Stuart, Harvey, Anita, Sato, Masahiko, Aspenberg, Per
Published in Journal of orthopaedic research (01.03.2014)
Published in Journal of orthopaedic research (01.03.2014)
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B-ring unsaturated estrogens: biological evaluation of 17alpha-Dihydroequilein and novel B-Nor-6-thiaequilenins as tissue selective estrogens
Lugar, 3rd, Charles W, Magee, David, Adrian, Mary D, Shetler, Pamela, Bryant, Henry U, Dodge, Jeffrey A
Published in Bioorganic & medicinal chemistry letters (15.12.2003)
Published in Bioorganic & medicinal chemistry letters (15.12.2003)
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Benzothiophene and Naphthalene Derived Constrained SERMs
Wallace, Owen B., Bryant, Henry U., Shetler, Pamela K., Adrian, Mary D., Geiser, Andrew G.
Published in ChemInform (25.01.2005)
Published in ChemInform (25.01.2005)
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B-Ring Unsaturated Estrogens: Biological Evaluation of 17α-Dihydroequilein and Novel B-Nor-6-thiaequilenins as Tissue Selective Estrogens
Lugar, Charles W. III, Magee, David, Adrian, Mary D., Shetler, Pamela, Bryant, Henry U., Dodge, Jeffrey A.
Published in ChemInform (06.04.2004)
Published in ChemInform (06.04.2004)
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