2-Butyl-4-chloroimidazole based substituted piperazine-thiosemicarbazone hybrids as potent inhibitors of Mycobacterium tuberculosis
Jallapally, Anvesh, Addla, Dinesh, Yogeeswari, Perumal, Sriram, Dharmarajan, Kantevari, Srinivas
Published in Bioorganic & medicinal chemistry letters (01.12.2014)
Published in Bioorganic & medicinal chemistry letters (01.12.2014)
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Journal Article
Design, synthesis and antimicrobial evaluation of novel 1-benzyl 2-butyl-4-chloroimidazole embodied 4-azafluorenones via molecular hybridization approach
Addla, Dinesh, Bhima, Sridhar, Balasubramanian, Devi, Anjana, Kantevari, Srinivas
Published in Bioorganic & medicinal chemistry letters (15.12.2012)
Published in Bioorganic & medicinal chemistry letters (15.12.2012)
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Journal Article
Multi-targeting exploration of new 2-aminothiazolyl quinolones: Synthesis, antimicrobial evaluation, interaction with DNA, combination with topoisomerase IV and penetrability into cells
Cheng, Yu, Avula, Srinivasa Rao, Gao, Wei-Wei, Addla, Dinesh, Tangadanchu, Vijai Kumar Reddy, Zhang, Ling, Lin, Jian-Mei, Zhou, Cheng-He
Published in European journal of medicinal chemistry (29.11.2016)
Published in European journal of medicinal chemistry (29.11.2016)
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Journal Article
Rational design, synthesis and antitubercular evaluation of novel 2-(trifluoromethyl)phenothiazine-[1,2,3]triazole hybrids
Addla, Dinesh, Jallapally, Anvesh, Gurram, Divya, Yogeeswari, Perumal, Sriram, Dharmarajan, Kantevari, Srinivas
Published in Bioorganic & medicinal chemistry letters (01.01.2014)
Published in Bioorganic & medicinal chemistry letters (01.01.2014)
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Journal Article
Discovery of membrane active benzimidazole quinolones-based topoisomerase inhibitors as potential DNA-binding antimicrobial agents
Zhang, Ling, Addla, Dinesh, Ponmani, Jeyakkumar, Wang, Ao, Xie, Dan, Wang, Ya-Nan, Zhang, Shao-Lin, Geng, Rong-Xia, Cai, Gui-Xin, Li, Shuo, Zhou, Cheng-He
Published in European journal of medicinal chemistry (23.03.2016)
Published in European journal of medicinal chemistry (23.03.2016)
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Journal Article
Design, synthesis and evaluation of 1,2,3-triazole-adamantylacetamide hybrids as potent inhibitors of Mycobacterium tuberculosis
Addla, Dinesh, Jallapally, Anvesh, Gurram, Divya, Yogeeswari, Perumal, Sriram, Dharmarajan, Kantevari, Srinivas
Published in Bioorganic & medicinal chemistry letters (15.04.2014)
Published in Bioorganic & medicinal chemistry letters (15.04.2014)
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Journal Article
Influence of temperature for the azide displacement in benzodiazepine derivatives: Experimental and DFT study of competing S(N)1, S(N)2 and double S(N)2 reaction pathways
Santos Evangelista, Tereza Cristina, Delarmelina, Maicon, Addla, Dinesh, Allao, Rafael A., Kaiser, Carlos Roland, Carneiro, Jose Walkimar de M., Silva-Jr, Floriano Paes, Ferreira, Sabrina Baptista
Published in Tetrahedron letters (30.03.2021)
Published in Tetrahedron letters (30.03.2021)
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Journal Article
Influence of temperature for the azide displacement in benzodiazepine derivatives: Experimental and DFT study of competing SN1, SN2 and double SN2 reaction pathways
Evangelista, Tereza Cristina Santos, Delarmelina, Maicon, Addla, Dinesh, Allão, Rafael A., Kaiser, Carlos Roland, Carneiro, José Walkimar de M., Silva-Jr, Floriano Paes, Ferreira, Sabrina Baptista
Published in Tetrahedron letters (30.03.2021)
Published in Tetrahedron letters (30.03.2021)
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Journal Article
Facile Diversity-Oriented Synthesis and Antitubercular Evaluation of Novel Aryl and Heteroaryl Tethered Pyridines and Dihydro-6H-quinolin-5-ones Derived via Variants of the Bohlmann–Rahtz Reaction
Kantevari, Srinivas, Patpi, Santhosh Reddy, Addla, Dinesh, Putapatri, Siddamal Reddy, Sridhar, Balasubramanian, Yogeeswari, Perumal, Sriram, Dharmarajan
Published in ACS combinatorial science (11.07.2011)
Published in ACS combinatorial science (11.07.2011)
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Journal Article
Design, synthesis and evaluation of novel 2-butyl-4-chloroimidazole derived peptidomimetics as Angiotensin Converting Enzyme (ACE) inhibitors
Jallapally, Anvesh, Addla, Dinesh, Bagul, Pankaj, Sridhar, Balasubramanian, Banerjee, Sanjay K., Kantevari, Srinivas
Published in Bioorganic & medicinal chemistry (01.07.2015)
Published in Bioorganic & medicinal chemistry (01.07.2015)
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Journal Article
Synthesis and evaluation of novel 2-butyl-4-chloro-1-methylimidazole embedded chalcones and pyrazoles as angiotensin converting enzyme (ACE) inhibitors
Kantevari, Srinivas, Addla, Dinesh, Bagul, Pankaj K., Sridhar, Balasubramanian, Banerjee, Sanjay K.
Published in Bioorganic & medicinal chemistry (15.08.2011)
Published in Bioorganic & medicinal chemistry (15.08.2011)
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Journal Article
Design, synthesis and evaluation of novel 2-hydroxypyrrolobenzodiazepine-5,11-dione analogues as potent angiotensin converting enzyme (ACE) inhibitors
Addla, Dinesh, Jallapally, Anvesh, Kanwal, Abhinav, Sridhar, Balasubramanian, Banerjee, Sanjay K., Kantevari, Srinivas
Published in Bioorganic & medicinal chemistry (01.08.2013)
Published in Bioorganic & medicinal chemistry (01.08.2013)
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