Pharmacological Profile and Molecular Modeling of Cyclic Opioid Analogues Incorporating Various Phenylalanine Derivatives
Adamska‐Bartłomiejczyk, Anna, Lipiński, Piotr F. J., Piekielna‐Ciesielska, Justyna, Kluczyk, Alicja, Janecka, Anna
Published in ChemMedChem (20.07.2020)
Published in ChemMedChem (20.07.2020)
Get full text
Journal Article
Synthesis, Biological Activity and Molecular Docking of Chimeric Peptides Targeting Opioid and NOP Receptors
Wtorek, Karol, Ghidini, Alessia, Gentilucci, Luca, Adamska-Bartłomiejczyk, Anna, Piekielna-Ciesielska, Justyna, Ruzza, Chiara, Sturaro, Chiara, Calò, Girolamo, Pieretti, Stefano, Kluczyk, Alicja, McDonald, John, Lambert, David G., Janecka, Anna
Published in International journal of molecular sciences (21.10.2022)
Published in International journal of molecular sciences (21.10.2022)
Get full text
Journal Article
Synthesis, Pharmacological Evaluation, and Computational Studies of Cyclic Opioid Peptidomimetics Containing β3-Lysine
Wtorek, Karol, Lipiński, Piotr F. J., Adamska-Bartłomiejczyk, Anna, Piekielna-Ciesielska, Justyna, Sukiennik, Jarosław, Kluczyk, Alicja, Janecka, Anna
Published in Molecules (Basel, Switzerland) (28.12.2021)
Published in Molecules (Basel, Switzerland) (28.12.2021)
Get full text
Journal Article
Synthesis, receptor binding studies, optical spectroscopic and in silico structural characterization of morphiceptin analogs with cis‐4‐amino‐L‐proline residues
Adamska‐Bartłomiejczyk, Anna, Borics, Attila, Tömböly, Csaba, Dvorácskó, Szabolcs, Lisowski, Marek, Kluczyk, Alicja, Wołczański, Grzegorz, Piekielna‐Ciesielska, Justyna, Janecka, Anna
Published in Journal of peptide science (01.12.2017)
Published in Journal of peptide science (01.12.2017)
Get full text
Journal Article
Analgesic Peptides: From Natural Diversity to Rational Design
Gach-Janczak, Katarzyna, Biernat, Monika, Kuczer, Mariola, Adamska-Bartłomiejczyk, Anna, Kluczyk, Alicja
Published in Molecules (Basel, Switzerland) (01.04.2024)
Published in Molecules (Basel, Switzerland) (01.04.2024)
Get full text
Journal Article
Neuroprotective and Anti-inflammatory Effects of Rubiscolin-6 Analogs with Proline Surrogates in Position 2
Perlikowska, Renata, Silva, Joana, Alves, Celso, Susano, Patricia, Zakłos-Szyda, Małgorzata, Skibska, Agnieszka, Adamska-Bartłomiejczyk, Anna, Wtorek, Karol, do Rego, Jean-Claude, do Rego, Jean-Luc, Kluczyk, Alicja, Pedrosa, Rui
Published in Neurochemical research (01.04.2024)
Published in Neurochemical research (01.04.2024)
Get full text
Journal Article
Synthesis and Pharmacological Evaluation of Hybrids Targeting Opioid and Neurokinin Receptors
Wtorek, Karol, Adamska-Bartłomiejczyk, Anna, Piekielna-Ciesielska, Justyna, Ferrari, Federica, Ruzza, Chiara, Kluczyk, Alicja, Piasecka-Zelga, Joanna, Calo', Girolamo, Janecka, Anna
Published in Molecules (Basel, Switzerland) (05.12.2019)
Published in Molecules (Basel, Switzerland) (05.12.2019)
Get full text
Journal Article
Synthesis and activity of opioid peptidomimetics with β2- and β3-amino acids
Gach-Janczak, Katarzyna, Piekielna-Ciesielska, Justyna, Adamska-Bartłomiejczyk, Anna, Perlikowska, Renata, Kruszyński, Rafał, Kluczyk, Alicja, Krzywik, Julia, Sukiennik, Jarosław, Cerlesi, Maria Camilla, Calo, Girolamo, Wasilewski, Andrzej, Zielińska, Marta, Janecka, Anna
Published in Peptides (New York, N.Y. : 1980) (01.09.2017)
Published in Peptides (New York, N.Y. : 1980) (01.09.2017)
Get full text
Journal Article
Design, Synthesis and Functional Analysis of Cyclic Opioid Peptides with Dmt-Tic Pharmacophore
Sarkar, Arijit, Adamska-Bartlomiejczyk, Anna, Piekielna-Ciesielska, Justyna, Wtorek, Karol, Kluczyk, Alicja, Borics, Attila, Janecka, Anna
Published in Molecules (Basel, Switzerland) (17.09.2020)
Published in Molecules (Basel, Switzerland) (17.09.2020)
Get full text
Journal Article
In vitro and in vivo activity of cyclopeptide Dmt-c[d-Lys-Phe-Asp]NH2, a mu opioid receptor agonist biased toward β-arrestin
Gach-Janczak, Katarzyna, Piekielna-Ciesielska, Justyna, Adamska-Bartłomiejczyk, Anna, Wtorek, Karol, Ferrari, Federica, Calo’, Girolamo, Szymaszkiewicz, Agata, Piasecka-Zelga, Joanna, Janecka, Anna
Published in Peptides (New York, N.Y. : 1980) (01.07.2018)
Published in Peptides (New York, N.Y. : 1980) (01.07.2018)
Get full text
Journal Article
Cyclic mu-opioid receptor ligands containing multiple N-methylated amino acid residues
Adamska-Bartłomiejczyk, Anna, Janecka, Anna, Szabó, Márton Richárd, Cerlesi, Maria Camilla, Calo, Girolamo, Kluczyk, Alicja, Tömböly, Csaba, Borics, Attila
Published in Bioorganic & medicinal chemistry letters (15.04.2017)
Published in Bioorganic & medicinal chemistry letters (15.04.2017)
Get full text
Journal Article
In vitro and in vivo activity of cyclopeptide Dmt-c[d-Lys-Phe-Asp]NH 2 , a mu opioid receptor agonist biased toward β-arrestin
Gach-Janczak, Katarzyna, Piekielna-Ciesielska, Justyna, Adamska-Bartłomiejczyk, Anna, Wtorek, Karol, Ferrari, Federica, Calo', Girolamo, Szymaszkiewicz, Agata, Piasecka-Zelga, Joanna, Janecka, Anna
Published in Peptides (New York, N.Y. : 1980) (01.07.2018)
Published in Peptides (New York, N.Y. : 1980) (01.07.2018)
Get full text
Journal Article
Synthesis, Pharmacological Evaluation, and Computational Studies of Cyclic Opioid Peptidomimetics Containing β 3 -Lysine
Wtorek, Karol, Lipiński, Piotr F J, Adamska-Bartłomiejczyk, Anna, Piekielna-Ciesielska, Justyna, Sukiennik, Jarosław, Kluczyk, Alicja, Janecka, Anna
Published in Molecules (Basel, Switzerland) (28.12.2021)
Get full text
Published in Molecules (Basel, Switzerland) (28.12.2021)
Journal Article
Synthesis and activity of opioid peptidomimetics with β 2 - and β 3 -amino acids
Gach-Janczak, Katarzyna, Piekielna-Ciesielska, Justyna, Adamska-Bartłomiejczyk, Anna, Perlikowska, Renata, Kruszyński, Rafał, Kluczyk, Alicja, Krzywik, Julia, Sukiennik, Jarosław, Cerlesi, Maria Camilla, Calo, Girolamo, Wasilewski, Andrzej, Zielińska, Marta, Janecka, Anna
Published in Peptides (New York, N.Y. : 1980) (01.09.2017)
Published in Peptides (New York, N.Y. : 1980) (01.09.2017)
Get full text
Journal Article