Identification of novel quinazoline derivatives as potent antiplasmodial agents
Bouchut, Anne, Rotili, Dante, Pierrot, Christine, Valente, Sergio, Lafitte, Sophia, Schultz, Johan, Hoglund, Urban, Mazzone, Roberta, Lucidi, Alessia, Fabrizi, Giancarlo, Pechalrieu, Dany, Arimondo, Paola B., Skinner-Adams, Tina S., Chua, Ming Jang, Andrews, Kathy T., Mai, Antonello, Khalife, Jamal
Published in European journal of medicinal chemistry (01.01.2019)
Published in European journal of medicinal chemistry (01.01.2019)
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Anti-Giardia Drug Discovery: Current Status and Gut Feelings
Riches, Andrew, Hart, Christopher J. S, Trenholme, Katharine R, Skinner-Adams, Tina S
Published in Journal of medicinal chemistry (25.11.2020)
Published in Journal of medicinal chemistry (25.11.2020)
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Fingerprinting the substrate specificity of M1 and M17 aminopeptidases of human malaria, Plasmodium falciparum
Poreba, Marcin, McGowan, Sheena, Skinner-Adams, Tina S, Trenholme, Katharine R, Gardiner, Donald L, Whisstock, James C, To, Joyce, Salvesen, Guy S, Dalton, John P, Drag, Marcin
Published in PloS one (16.02.2012)
Published in PloS one (16.02.2012)
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Structure–Activity and Structure–Toxicity Relationships of Peptoid‐Based Histone Deacetylase Inhibitors with Dual‐Stage Antiplasmodial Activity
Mackwitz, Marcel K. W., Hesping, Eva, Antonova‐Koch, Yevgeniya, Diedrich, Daniela, Woldearegai, Tamirat Gebru, Skinner‐Adams, Tina, Clarke, Mary, Schöler, Andrea, Limbach, Laura, Kurz, Thomas, Winzeler, Elizabeth A., Held, Jana, Andrews, Katherine T., Hansen, Finn K.
Published in ChemMedChem (06.05.2019)
Published in ChemMedChem (06.05.2019)
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Abstracts of the 2024 50th Annual NATAS Conference
Advincula, Rigoberto, Bowman, Christopher, Smith, Dennis, Schoch, Jr, Karl, Adams, Tina, Stewart, Cathy, Judovits, Lawrence, Pilato, Louis
Published in Polymers (08.10.2024)
Published in Polymers (08.10.2024)
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Discovery of 1,3,4-oxadiazoles with slow-action activity against Plasmodium falciparum malaria parasites
Andrews, Katherine T., Fisher, Gillian M., Firmin, Meaghan, Liepa, Andris J., Wilson, Tony, Gardiner, James, Mohri, Yacine, Debele, Emmanuel, Rai, Anjana, Davey, Andrew K., Masurier, Antoine, Delion, Alix, Mouratidis, Alexandros A., Hutt, Oliver E., Forsyth, Craig M., Burrows, Jeremy N., Ryan, John H., Riches, Andrew G., Skinner-Adams, Tina S.
Published in European journal of medicinal chemistry (15.11.2024)
Published in European journal of medicinal chemistry (15.11.2024)
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Journal Article
Effect of clinically approved HDAC inhibitors on Plasmodium, Leishmania and Schistosoma parasite growth
Chua, Ming Jang, Arnold, Megan S.J., Xu, Weijun, Lancelot, Julien, Lamotte, Suzanne, Späth, Gerald F., Prina, Eric, Pierce, Raymond J., Fairlie, David P., Skinner-Adams, Tina S., Andrews, Katherine T.
Published in International journal for parasitology -- drugs and drug resistance (01.04.2017)
Published in International journal for parasitology -- drugs and drug resistance (01.04.2017)
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Journal Article
Activity of alkoxyamide-based histone deacetylase inhibitors against Plasmodium falciparum malaria parasites
Dawood, Wisam A., Fisher, Gillian M., Kinnen, Franziska J.M., Anzenhofer, Christian, Skinner-Adams, Tina, Alves Avelar, Leandro, Asfaha, Yodita, Kurz, Thomas, Andrews, Katherine T.
Published in Experimental parasitology (01.03.2024)
Published in Experimental parasitology (01.03.2024)
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Journal Article
Profiling the anti-protozoal activity of anti-cancer HDAC inhibitors against Plasmodium and Trypanosoma parasites
Engel, Jessica A., Jones, Amy J., Avery, Vicky M., Sumanadasa, Subathdrage D.M., Ng, Susanna S., Fairlie, David P., Adams, Tina S., Andrews, Katherine T.
Published in International journal for parasitology -- drugs and drug resistance (01.12.2015)
Published in International journal for parasitology -- drugs and drug resistance (01.12.2015)
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Abstracts of the 2023 49th Annual NATAS Conference
LaVan, David, Yi, Feng, Adams, Tina, Tao, Ran, Pelczar, Elizabeth, Xia, Han, Hu, Xiao, Sauerbrunn, Stephen, Matisons, Janis
Published in Polymers (30.07.2023)
Published in Polymers (30.07.2023)
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Conference Proceeding
Lysine Acetylation in Sexual Stage Malaria Parasites Is a Target for Antimalarial Small Molecules
TRENHOLME, Katharine, MAREK, Linda, GOODMAN, Christopher D, MCFADDEN, Geoffrey I, SUMANADASA, Subathdrage D. M, FAIRLIE, David P, AVERY, Vicky M, KURZ, Thomas, ANDREWS, Katherine T, DUFFY, Sandra, PRADEL, Gabriele, FISHER, Gillian, HANSEN, Finn K, SKINNER-ADAMS, Tina S, BUTTERWORTH, Alice, NGWA, Che Julius, MOECKING, Jonas
Published in Antimicrobial agents and chemotherapy (01.07.2014)
Published in Antimicrobial agents and chemotherapy (01.07.2014)
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Mollemycin A: An Antimalarial and Antibacterial Glyco-hexadepsipeptide-polyketide from an Australian Marine-Derived Streptomyces sp. (CMB-M0244)
Raju, Ritesh, Khalil, Zeinab G, Piggott, Andrew M, Blumenthal, Antje, Gardiner, Donald L, Skinner-Adams, Tina S, Capon, Robert J
Published in Organic letters (21.03.2014)
Published in Organic letters (21.03.2014)
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A Subset Screen of the Compounds Australia Scaffold Library Identifies 7-Acylaminodibenzoxazepinones as Potent and Selective Hits for Anti- Giardia Drug Discovery
Hart, Christopher J S, Riches, Andrew G, Tiash, Snigdha, Clapper, Erin, Ramu, Soumya, Zuegg, Johannes, Ryan, John H, Skinner-Adams, Tina S
Published in Biomedicines (08.12.2022)
Published in Biomedicines (08.12.2022)
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Journal Article
Plasmodium falciparum neutral aminopeptidases: new targets for anti-malarials
Skinner-Adams, Tina S., Stack, Colin M., Trenholme, Katharine R., Brown, Chris L., Grembecka, Jolanta, Lowther, Jonathan, Mucha, Artur, Drag, Marcin, Kafarski, Pawel, McGowan, Sheena, Whisstock, James C., Gardiner, Donald L., Dalton, John P.
Published in Trends in biochemical sciences (Amsterdam. Regular ed.) (2010)
Published in Trends in biochemical sciences (Amsterdam. Regular ed.) (2010)
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Journal Article
Abstracts of the 2022 48th Annual NATAS Conference
Adams, Tina, Schoch, Karl F., Pelczar, Elizabeth, Xia, Han, Hu, Xiao, Reynaud, Sara, Sauerbrunn, Stephen
Published in Polymers (30.07.2022)
Published in Polymers (30.07.2022)
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Journal Article
Conference Proceeding
Structural basis for the inhibition of the essential Plasmodium falciparum M1 neutral aminopeptidase
McGowan, Sheena, Porter, Corrine J, Lowther, Jonathan, Stack, Colin M, Golding, Sarah J, Skinner-Adams, Tina S, Trenholme, Katharine R, Teuscher, Franka, Donnelly, Sheila M, Grembecka, Jolanta, Mucha, Artur, Kafarski, Pawel, DeGori, Ross, Buckle, Ashley M, Gardiner, Donald L, Whisstock, James C, Dalton, John P
Published in Proceedings of the National Academy of Sciences - PNAS (24.02.2009)
Published in Proceedings of the National Academy of Sciences - PNAS (24.02.2009)
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Journal Article
Catalyst-Controlled Stereoselective Synthesis Secures the Structure of the Antimalarial Isocyanoterpene Pustulosaisonitrile‑1
White, Andrew M, Dao, Kathy, Vrubliauskas, Darius, Könst, Zef A, Pierens, Gregory K, Mándi, Attila, Andrews, Katherine T, Skinner-Adams, Tina S, Clarke, Mary E, Narbutas, Patrick T, Sim, Desmond C.-M, Cheney, Karen L, Kurtán, Tibor, Garson, Mary J, Vanderwal, Christopher D
Published in Journal of organic chemistry (15.12.2017)
Published in Journal of organic chemistry (15.12.2017)
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Journal Article
Structural reassignment of a dibenz[b,f][1,4]oxazepin-11(10H)-one with potent antigiardial activity
Riches, Andrew G., Hart, Christopher J. S., Schmit, Matthieu, Debele, Emmanuel A., Tiash, Snigdha, Clapper, Erin, Skinner-Adams, Tina S., Ryan, John H.
Published in Australian journal of chemistry (01.01.2022)
Published in Australian journal of chemistry (01.01.2022)
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