Altered conformational sampling along an evolutionary trajectory changes the catalytic activity of an enzyme
Kaczmarski, Joe A., Mahawaththa, Mithun C., Feintuch, Akiva, Clifton, Ben E., Adams, Luke A., Goldfarb, Daniella, Otting, Gottfried, Jackson, Colin J.
Published in Nature communications (23.11.2020)
Published in Nature communications (23.11.2020)
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Journal Article
Enhanced Cytotoxicity through Conjugation of a “Clickable” Luminescent Re(I) Complex to a Cell-Penetrating Lipopeptide
Leonidova, Anna, Pierroz, Vanessa, Adams, Luke A, Barlow, Nicholas, Ferrari, Stefano, Graham, Bim, Gasser, Gilles
Published in ACS medicinal chemistry letters (10.07.2014)
Published in ACS medicinal chemistry letters (10.07.2014)
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Journal Article
Application of Fragment-Based Screening to the Design of Inhibitors of Escherichia coli DsbA
Adams, Luke A., Sharma, Pooja, Mohanty, Biswaranjan, Ilyichova, Olga V., Mulcair, Mark D., Williams, Martin L., Gleeson, Ellen C., Totsika, Makrina, Doak, Bradley C., Caria, Sofia, Rimmer, Kieran, Horne, James, Shouldice, Stephen R., Vazirani, Mansha, Headey, Stephen J., Plumb, Brent R., Martin, Jennifer L., Heras, Begoña, Simpson, Jamie S., Scanlon, Martin J.
Published in Angewandte Chemie (International ed.) (09.02.2015)
Published in Angewandte Chemie (International ed.) (09.02.2015)
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Journal Article
Pulse EPR-enabled interpretation of scarce pseudocontact shifts induced by lanthanide binding tags
Abdelkader, Elwy H., Yao, Xuejun, Feintuch, Akiva, Adams, Luke A., Aurelio, Luigi, Graham, Bim, Goldfarb, Daniella, Otting, Gottfried
Published in Journal of biomolecular NMR (01.01.2016)
Published in Journal of biomolecular NMR (01.01.2016)
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Journal Article
Genetic Encoding of N 6‑(((Trimethylsilyl)methoxy)carbonyl)‑l‑lysine for NMR Studies of Protein–Protein and Protein–Ligand Interactions
Abdelkader, Elwy H, Qianzhu, Haocheng, Tan, Yi Jiun, Adams, Luke A, Huber, Thomas, Otting, Gottfried
Published in Journal of the American Chemical Society (20.01.2021)
Published in Journal of the American Chemical Society (20.01.2021)
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Journal Article
Selective Distance Measurements Using Triple Spin Labeling with Gd3+, Mn2+, and a Nitroxide
Wu, Zuyan, Feintuch, Akiva, Collauto, Alberto, Adams, Luke A., Aurelio, Luigi, Graham, Bim, Otting, Gottfried, Goldfarb, Daniella
Published in The journal of physical chemistry letters (02.11.2017)
Published in The journal of physical chemistry letters (02.11.2017)
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Journal Article
Diastereoselective Synthesis of Cyclopropane Amino Acids Using Diazo Compounds Generated in Situ
Adams, Luke A, Aggarwal, Varinder K, Bonnert, Roger V, Bressel, Bettina, Cox, Russell J, Shepherd, Jon, de Vicente, Javier, Walter, Magnus, Whittingham, William G, Winn, Caroline L
Published in Journal of organic chemistry (28.11.2003)
Published in Journal of organic chemistry (28.11.2003)
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Journal Article
Chemical Tagging with tert‐Butyl and Trimethylsilyl Groups for Measuring Intermolecular Nuclear Overhauser Effects in a Large Protein–Ligand Complex
Jabar, Shereen, Adams, Luke A., Wang, Yao, Aurelio, Luigi, Graham, Bim, Otting, Gottfried
Published in Chemistry : a European journal (21.09.2017)
Published in Chemistry : a European journal (21.09.2017)
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Journal Article
Rapid Elaboration of Fragments into Leads Applied to Bromodomain‑3 Extra-Terminal Domain
Adams, Luke A., Wilkinson-White, Lorna E., Gunzburg, Menachem J., Headey, Stephen J., Mohanty, Biswaranjan, Scanlon, Martin J., Capuano, Ben, Mackay, Joel P., Doak, Bradley C.
Published in Journal of medicinal chemistry (27.04.2023)
Published in Journal of medicinal chemistry (27.04.2023)
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Journal Article
Small neutral Gd(iii) tags for distance measurements in proteins by double electron-electron resonance experiments
Mahawaththa, Mithun C, Lee, Michael D, Giannoulis, Angeliki, Adams, Luke A, Feintuch, Akiva, Swarbrick, James D, Graham, Bim, Nitsche, Christoph, Goldfarb, Daniella, Otting, Gottfried
Published in Physical chemistry chemical physics : PCCP (2018)
Published in Physical chemistry chemical physics : PCCP (2018)
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Journal Article
Trimethylsilyl tag for probing protein–ligand interactions by NMR
Becker, Walter, Adams, Luke A., Graham, Bim, Wagner, Gabriel E., Zangger, Klaus, Otting, Gottfried, Nitsche, Christoph
Published in Journal of biomolecular NMR (01.04.2018)
Published in Journal of biomolecular NMR (01.04.2018)
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Journal Article
Selective Distance Measurements Using Triple Spin Labeling with Gd 3+ , Mn 2+ , and a Nitroxide
Wu, Zuyan, Feintuch, Akiva, Collauto, Alberto, Adams, Luke A, Aurelio, Luigi, Graham, Bim, Otting, Gottfried, Goldfarb, Daniella
Published in The journal of physical chemistry letters (02.11.2017)
Published in The journal of physical chemistry letters (02.11.2017)
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Journal Article
Synthesis and Characterization of High-Affinity 4,4-Difluoro-4-bora-3a,4a-diaza-s-indacene-Labeled Fluorescent Ligands for Human β-Adrenoceptors
Baker, Jillian G, Adams, Luke A, Salchow, Karolina, Mistry, Shailesh N, Middleton, Richard J, Hill, Stephen J, Kellam, Barrie
Published in Journal of medicinal chemistry (13.10.2011)
Published in Journal of medicinal chemistry (13.10.2011)
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Journal Article
Application of Fragment-Based Screening to the Design of Inhibitors of Escherichia coli DsbA
Adams, Luke A., Sharma, Pooja, Mohanty, Biswaranjan, Ilyichova, Olga V., Mulcair, Mark D., Williams, Martin L., Gleeson, Ellen C., Totsika, Makrina, Doak, Bradley C., Caria, Sofia, Rimmer, Kieran, Horne, James, Shouldice, Stephen R., Vazirani, Mansha, Headey, Stephen J., Plumb, Brent R., Martin, Jennifer L., Heras, Begoña, Simpson, Jamie S., Scanlon, Martin J.
Published in Angewandte Chemie (09.02.2015)
Published in Angewandte Chemie (09.02.2015)
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Journal Article
Efficient synthesis of protected cyclopropyl beta-aspartylphosphates
Adams, LA, Charmant, JPH, Cox, RJ, Walter, M, Whittingham, WG
Published in Organic & biomolecular chemistry (21.02.2004)
Published in Organic & biomolecular chemistry (21.02.2004)
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Journal Article